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Discovery of aryl sulfonamide-selective Nav1.7 inhibitors with a highly hydrophobic ethanoanthracene core 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 卷号: 41, 期号: 3, 页码: 293-302
作者:  Wang, Jin-tao;  Zheng, Yue-ming;  Chen, Yue-ting;  Gu, Min;  Gao, Zhao-bing
收藏  |  浏览/下载:44/0  |  提交时间:2020/07/01
Antiepileptic geissoschizine methyl ether is an inhibitor of multiple neuronal channels 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 9
作者:  Xie, Zhu-qing;  Tian, Xiao-ting;  Zheng, Yue-ming;  Zhan, Li;  Chen, Xue-qin
收藏  |  浏览/下载:23/0  |  提交时间:2020/07/01
discoveryofarylsulfonamideselectivenav17inhibitorswithahighlyhydrophobicethanoanthracenecore 期刊论文
actapharmacologicasinica, 2020, 卷号: 41, 期号: 3, 页码: 293
作者:  Wang Jintao;  Zheng Yueming;  Chen Yueting;  Gu Min;  Gao Zhaobing
收藏  |  浏览/下载:24/0  |  提交时间:2020/07/01
Quercetin Reduces Cortical GABAergic Transmission and Alleviates MK-801-Induced Hyperactivity 期刊论文
EBioMedicine, 2018, 卷号: 34, 页码: 201-213
作者:  Fan, Hui-Ran;  Du, Wei-Feng;  Zhu, Tao;  Wu, Yan-Jiao;  Liu, Yan-Mei
收藏  |  浏览/下载:34/0  |  提交时间:2019/01/08
An allosteric ligand-binding site in the extracellular cap of K2P channels 期刊论文
NATURE COMMUNICATIONS, 2017, 卷号: 8
作者:  Luo, Qichao;  Chen, Liping;  Cheng, Xi;  Ma, Yuqin;  Li, Xiaona
收藏  |  浏览/下载:17/0  |  提交时间:2019/01/08
Propofol inhibits hERG K+ channels and enhances the inhibition effects on its mutations in HEK293 cells 期刊论文
EUROPEAN JOURNAL OF PHARMACOLOGY, 2016, 卷号: 791, 页码: 168-178
作者:  Han, Sheng-Na;  Jing, Ying;  Yang, Lin-Lin;  Zhang, Zhao;  Zhang, Li-Rong
收藏  |  浏览/下载:42/0  |  提交时间:2019/01/08
Timosaponin derivative YY-23 acts as a non-competitive NMDA receptor antagonist and exerts a rapid antidepressant-like effect in mice 期刊论文
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 2, 页码: 166-176
作者:  Zhang, Qi;  Guo, Fei;  Fu, Zhi-wen;  Zhang, Bing;  Huang, Cheng-gang
收藏  |  浏览/下载:14/0  |  提交时间:2019/01/08
Novel KCNQ2 channel activators discovered using fluorescence-based and automated patch-clamp-based high-throughput screening techniques 期刊论文
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 1, 页码: 105-110
作者:  Yue, Jin-feng;  Qiao, Guan-hua;  Liu, Ni;  Chen, Xue-qin;  Nan, Fa-jun
收藏  |  浏览/下载:17/0  |  提交时间:2019/01/08
Lead compound optimization strategy (5) - reducing the hERG cardiac toxicity in drug development 期刊论文
Acta Pharmaceutica Sinica, 2016, 卷号: 51, 期号: 10, 页码: 1530-1539
作者:  Zhou Shengbin;  Wang Jiang;  Liu Hong
收藏  |  浏览/下载:45/0  |  提交时间:2019/01/08
timosaponinderivativeyy23actsasanoncompetitivenmdareceptorantagonistandexertsarapidantidepressantlikeeffectinmice 期刊论文
actapharmacologicasinica, 2016, 卷号: 000, 期号: 002, 页码: 166
作者:  QiZHANG;  Fei GUO;  Zhi-wen FU;  Bing ZHANG;  Cheng-gang HUANG
收藏  |  浏览/下载:2/0  |  提交时间:2020/07/01
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