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Metabolic profiling of tyrosine kinase inhibitor nintedanib using metabolomics 期刊论文
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2020
作者:  Zhou, Zi-Meng;  Wang, Yi-Kun;  Yan, Dong-Mei;  Fang, Jian-He;  Xiao, Xue-Rong
收藏  |  浏览/下载:10/0  |  提交时间:2021/01/05
The discovery of novel and selective fatty acid binding protein 4 inhibitors by virtual screening and biological evaluation 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 18, 页码: 4310-4317
作者:  Song, Ming;  Xu, Yong;  Zhang, Yan;  Nie, Tao;  Zhou, Yang
收藏  |  浏览/下载:21/0  |  提交时间:2018/12/13
Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5911-5916
Wang, Zhen; Bian, Huan; Bartual, Sergio G.; Du, Wenting; Luo, Jinfeng; Zhao, Hu; Zhang, Shasha; Mo, Cheng; Zhou, Yang; Xu, Yong; Tu, Zhengchao; Ren, Xiaomei; Lu, Xiaoyun; Brekken, Rolf A.; Yao, Libo; Bullock, Alex N.; Su, Jin; Ding, Ke
收藏  |  浏览/下载:51/0  |  提交时间:2016/12/16
Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5911-5916
作者:  Yao, Libo;  Ding, Ke;  Su, Jin;  Bullock, Alex N.;  Brekken, Rolf A.
收藏  |  浏览/下载:33/0  |  提交时间:2018/12/13
Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 4, 页码: 1565-1579
作者:  Tu, Zhengchao;  Zhou, Yulai;  Ding, Ke;  Xu, Yong;  Xue, Xiaoqian
收藏  |  浏览/下载:25/0  |  提交时间:2018/12/13
Identification of N-phenyl-2-(N-phenylphenylsulfonamido) acetamides as new ROR gamma inverse agonists: Virtual screening, structure-based optimization, and biological evaluation 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 116, 页码: 13-26
作者:  Xue, Xiaoqian;  Song, Yu;  Qian, Chao-Nan;  Yan, Weiqun;  Xing, Yanli
收藏  |  浏览/下载:23/0  |  提交时间:2018/12/13
Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 4, 页码: 1565-1579
Xue, Xiaoqian; Zhang, Yan; Liu, Zhaoxuan; Song, Ming; Xing, Yanli; Xiang, Qiuping; Wang, Zhen; Tu, Zhengchao; Zhou, Yulai; Ding, Ke; Xu, Yong
收藏  |  浏览/下载:20/0  |  提交时间:2016/12/16
The discovery of novel and selective fatty acid binding protein 4 inhibitors by virtual screening and biological evaluation 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 18, 页码: 4310-4317
Zhou, Yang; Nie, Tao; Zhang, Yan; Song, Ming; Li, Kuai; Ding, Mengxiao; Ding, Ke; Wu, Donghai; Xu, Yong
收藏  |  浏览/下载:21/0  |  提交时间:2016/12/16
Identification of N-phenyl-2-(N-phenylphenylsulfonamido) acetamides as new ROR gamma inverse agonists: Virtual screening, structure-based optimization, and biological evaluation 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 116, 页码: 13-26
Song, Yu; Xue, Xiaoqian; Wu, Xishan; Wang, Rui; Xing, Yanli; Yan, Weiqun; Zhou, Yulai; Qian, Chao-Nan; Zhang, Yan; Xu, Yong
收藏  |  浏览/下载:29/0  |  提交时间:2016/12/16
Psora-4, a Kv1.3 Blocker, Enhances Differentiation and Maturation in Neural Progenitor Cells 期刊论文
CNS NEUROSCIENCE & THERAPEUTICS, 2015, 卷号: 21, 期号: 7, 页码: 558-567
作者:  Zheng, Hui;  Zhou, Yu-Ye;  Hou, Guo-Qiang;  He, Song-Wei;  Li, Zhi-Yuan
收藏  |  浏览/下载:18/0  |  提交时间:2018/12/13


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