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Elucidating the druggable interface of protein-protein interactions using fragment docking and coevolutionary analysis 期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2016, 卷号: 113, 期号: 50, 页码: E8051-E8058
作者:  Bai, Fang;  Morcos, Faruck;  Cheng, Ryan R.;  Jiang, Hualiang
收藏  |  浏览/下载:23/0  |  提交时间:2019/01/08
Crystal structure of FabZ-ACP complex reveals a dynamic seesaw-like catalytic mechanism of dehydratase in fatty acid biosynthesis 期刊论文
CELL RESEARCH, 2016, 卷号: 26, 期号: 12, 页码: 1330-1344
作者:  Zhang, Lin;  Xiao, Jianfeng;  Xu, Jianrong;  Fu, Tianran;  Cao, Zhiwei
收藏  |  浏览/下载:16/0  |  提交时间:2019/01/08
Potent Antitumor Activities and Structure Basis of the Chiral beta-Lactam Bridged Analogue of Combretastatin A-4 Binding to Tubulin 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 22, 页码: 10329-10334
作者:  Zhou, Pengfei;  Liu, Yan;  Zhou, Lu;  Zhu, Kongkai;  Feng, Kechang
收藏  |  浏览/下载:21/0  |  提交时间:2019/01/08
Design, Synthesis, and Biological Evaluation of Novel Tetrahydroprotoberberine Derivatives (THPBs) as Selective alpha(1A)-Adrenoceptor Antagonists 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 20, 页码: 9489-9502
作者:  Guo, Diliang;  Li, Jing;  Lin, Henry;  Zhou, Yu;  Chen, Ying
收藏  |  浏览/下载:28/0  |  提交时间:2019/01/08
Rhodium(III)-Catalyzed Site-Selective C-H Alkylation and Arylation of Pyridones Using Organoboron Reagents 期刊论文
ORGANIC LETTERS, 2016, 卷号: 18, 期号: 20, 页码: 5376-5379
作者:  Peng, Panfeng;  Wang, Jiang;  Jiang, Hualiang;  Liu, Hong
收藏  |  浏览/下载:13/0  |  提交时间:2019/01/08
Small-molecule targeting of e3 ligase adaptor spop in kidney cancer 期刊论文
Cancer cell, 2016, 卷号: 30, 期号: 3, 页码: 474-484
作者:  Guo, Zhong-Qiang;  Zheng, Tong;  Chen, Baoen;  Luo, Cheng;  Ouyang, Sisheng
收藏  |  浏览/下载:80/0  |  提交时间:2019/05/09
Small-Molecule Targeting of E3 Ligase Adaptor SPOP in Kidney Cancer 期刊论文
CANCER CELL, 2016, 卷号: 30, 期号: 3, 页码: 474-484
作者:  Guo, Zhong-Qiang;  Zheng, Tong;  Chen, Baoen;  Luo, Cheng;  Ouyang, Sisheng
收藏  |  浏览/下载:37/0  |  提交时间:2019/01/08
Crystal structures of sirt3 reveal that the alpha 2-alpha 3 loop and alpha 3-helix affect the interaction with long-chain acyl lysine 期刊论文
Febs letters, 2016, 卷号: 590, 期号: 17, 页码: 3019-3028
作者:  Gai, Wei;  Li, He;  Jiang, Hualiang;  Long, Yaqiu;  Liu, Dongxiang
收藏  |  浏览/下载:38/0  |  提交时间:2019/05/09
Discovery of novel inhibitors targeting the menin-mixed lineage leukemia interface using pharmacophore- and docking-based virtual screening 期刊论文
Journal of chemical information and modeling, 2016, 卷号: 56, 期号: 9, 页码: 1847-1855
作者:  Xu, Yuan;  Yue, Liyan;  Wang, Yulan;  Xing, Jin;  Chen, Zhifeng
收藏  |  浏览/下载:37/0  |  提交时间:2019/05/09
Probing the structure and dynamics of caveolin-1 in a caveolae-mimicking asymmetric lipid bilayer model 期刊论文
EUROPEAN BIOPHYSICS JOURNAL WITH BIOPHYSICS LETTERS, 2016, 卷号: 45, 期号: 6, 页码: 511-521
作者:  Liu, Hanqi;  Yang, Linlin;  Zhang, Qiansen;  Mao, Lingxue;  Jiang, Hualiang
收藏  |  浏览/下载:15/0  |  提交时间:2019/01/08


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