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Darinaparsin (ZIO-101) enhances the sensitivity of small-cell lung cancer to PARP inhibitors 期刊论文
ACTA PHARMACOLOGICA SINICA, 2022
作者:  Cao, Guo-Zhen;  Ma, Li-Ying;  Zhang, Zong-Hui;  Wang, Xiao-Lin;  Hua, Jing-Han
收藏  |  浏览/下载:25/0  |  提交时间:2022/12/22
Vanguard is a Glucose Deprivation-Responsive Long Non-Coding RNA Essential for Chromatin Remodeling-Reliant DNA Repair 期刊论文
ADVANCED SCIENCE, 2022
作者:  Zhang, Ben;  Thorne, Rick Francis;  Zhang, Pengfei;  Wu, Mian;  Liu, Lianxin
收藏  |  浏览/下载:15/0  |  提交时间:2022/12/23
The dual HDAC-PI3K inhibitor CUDC-907 displays single-agent activity and synergizes with PARP inhibitor olaparib in small cell lung cancer 期刊论文
JOURNAL OF EXPERIMENTAL & CLINICAL CANCER RESEARCH, 2020, 卷号: 39
作者:  Ma, Liying;  Bian, Xing;  Lin, Wenchu
收藏  |  浏览/下载:38/0  |  提交时间:2020/11/30
The MYC Paralog-PARP1 Axis as a Potential TherapeuticTarget in MYC Paralog-Activated Small Cell Lung Cancer 期刊论文
FRONTIERS IN ONCOLOGY, 2020, 卷号: 10
作者:  Bian, Xing;  Wang, Xiaolin;  Zhang, Qiuyan;  Ma, Liying;  Cao, Guozhen
收藏  |  浏览/下载:57/0  |  提交时间:2020/11/30
BTH-8, a novel poly (ADP-ribose) polymerase-1 (PARP-1) inhibitor, causes DNA double-strand breaks and exhibits anticancer activities in vitro and in vivo 期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2020, 卷号: 150, 页码: 238-245
作者:  Guo, Chuanlong;  Zhang, Fan;  Wu, Xiaochen;  Yu, Xuemin;  Wu, Xianggen
收藏  |  浏览/下载:32/0  |  提交时间:2020/09/23
USP9X stabilizes BRCA1 and confers resistance to DNA-damaging agents in human cancer cells 期刊论文
CANCER MEDICINE, 2019, 卷号: 8, 期号: 15, 页码: 6730-6740
作者:  Lu, Qin;  Zhang, Fang-Lin;  Lu, Da-Yun;  Shao, Zhi-Ming;  Li, Da-Qiang
收藏  |  浏览/下载:23/0  |  提交时间:2020/07/01
海洋溴酚化合物抗肿瘤活性筛选及作用机制研究 学位论文
中国科学院海洋研究所: 中国科学院大学, 2019
作者:  郭传龙
收藏  |  浏览/下载:78/0  |  提交时间:2019/06/17
Synthesis, preliminarily biological evaluation and molecular docking study of new Olaparib analogues as multifunctional PARP-1 and cholinesterase inhibitors 期刊论文
Journal of enzyme inhibition and medicinal chemistry, 2019, 卷号: 34, 页码: 150-162
作者:  Gao Cheng-Zhi[1];  Dong Wei[2];  Cui Zhi-Wen[3];  Yuan Qiong[4];  Hu Xia-Min[5]
收藏  |  浏览/下载:34/0  |  提交时间:2019/04/22
Synthesis, preliminarily biological evaluation and molecular docking study of new Olaparib analogues as multifunctional PARP-1 and cholinesterase inhibitors 期刊论文
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2019, 卷号: 34, 期号: 1
作者:  Gao, Cheng-Zhi;  Dong, Wei;  Cui, Zhi-Wen;  Yuan, Qiong;  Hu, Xia-Min
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/06
Design and synthesis of 2-(4,5,6,7-tetrahydrothienopyridin-2-yl)-benzoimidazole carboxamides as novel orally efficacious Poly(ADP-ribose)polymerase (PARP) inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 145, 页码: 389-403
作者:  Chen, Xuxing;  Huan, Xiajuan;  Liu, Qiufeng;  Wang, Yuqin;  He, Qian
收藏  |  浏览/下载:32/0  |  提交时间:2019/01/08


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