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上海药物研究所 [3]
中国医学科学院 北京... [2]
南华大学 [1]
四川大学 [1]
山东大学 [1]
华南理工大学 [1]
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期刊论文 [13]
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2021 [1]
2019 [1]
2018 [3]
2017 [2]
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2015 [1]
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Discovery of a highly potent kinase inhibitor capable of overcoming multiple imatinib-resistant ABL mutants for chronic myeloid leukemia (CML)
期刊论文
EUROPEAN JOURNAL OF PHARMACOLOGY, 2021, 卷号: 897
作者:
Lu, Tingting
;
Cao, Jiangyan
;
Zou, Fengming
;
Li, Xixiang
;
Wang, Aoli
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2021/04/26
BCR-ABL
ABL mutants
Chronic myeloid leukemia
Kinase inhibitor
Imatinib resistance
Deciphering the mechanism of Indirubin and its derivatives in the inhibition of Imatinib resistance using a "drug target prediction-gene microarray analysis-protein network construction" strategy
期刊论文
BMC COMPLEMENTARY AND ALTERNATIVE MEDICINE, 2019, 卷号: 19
作者:
Li, Huayao
;
Liu, Lijuan
;
Zhuang, Jing
;
Liu, Cun
;
Zhou, Chao
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/11
Indirubin
Derivatives
Imatinib resistance
Drug target prediction
Gene microarray analysis
Protein network construction
Comparison of Frequency and Sensitivity of BCR-ABL1 Kinase Domain Mutations in Asian and White Patients With Imatinib-resistant Chronice-Phase Chronic Myeloid Leukemia
期刊论文
CLINICAL LYMPHOMA MYELOMA & LEUKEMIA, 2018, 卷号: 18, 期号: 10
作者:
Cui, Jiu Wei
;
Kim, Hawk
;
Kim, SooHyun
;
Kim, Hyeoung-Joon
;
Kim, Yeo-Kyeoung
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/12/05
Asian countries
BCR-ABL1 mutation
CML
Drug resistance
Imatinib
Co-delivery of doxorubicin and imatinib by pH sensitive cleavable PEGylated nanoliposomes with folate-mediated targeting to overcome multidrug resistance
期刊论文
INTERNATIONAL JOURNAL OF PHARMACEUTICS, 2018, 卷号: 542, 期号: 1-2
作者:
Chen, Yan
;
Cheng, Yao
;
Zhao, Pengxuan
;
Zhang, Shasha
;
Li, Minsi
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2019/12/05
Doxorubicin
Imatinib
Drug resistance
pH-sensitive
Liposomes
LncRNA MALAT1 promotes cell proliferation and imatinib resistance by sponging miR-328 in chronic myelogenous leukemia
期刊论文
Biochemical and Biophysical Research Communications, 2018, 卷号: 507, 期号: 1-4, 页码: 1-8
作者:
Wen, Feng*
;
Cao, Yi-Xiong
;
Luo, Ze-Yu
;
Liao, Pei
;
Lu, Zhong-Wei
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/27
*Chronic myeloid leukemia
*Imatinib resistance
*LncRNA MALAT1
*Proliferation
*miR-328
[The Roles of Glut5 in Imatinib Resistance in the Ph+ Acute Lymphoblastic Leukemia Cell].
期刊论文
Sichuan Da Xue Xue Bao Yi Xue Ban, 2017, 卷号: Vol.48 No.3, 页码: 389-393
作者:
Yan TY
;
Naren DL
;
Gong YP.
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2019/03/01
Fructose
Glucose
transport
5
Imatinib
resistance
Ph+
acute
lymphoblastic
leukemia
The role of long noncoding RNA HOTAIR in the acquired multidrug resistance to imatinib in chronic myeloid leukemia cells
期刊论文
2017, 卷号: 22, 期号: 4, 页码: 208-216
作者:
Wang, Haiying
;
Li, Qian
;
Tang, Shusen
;
Li, Meifang
;
Feng, Anhua
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2020/01/04
Chronic myeloid leukemia
imatinib resistance
long noncoding RNA HOTAIR
PI3K/Akt pathway
Y-632 inhibits heat shock protein 90 (Hsp90) function by disrupting the interaction between Hsp90 and Hsp70/Hsp90 organizing protein, and exerts antitumor activity in vitro and in vivo
期刊论文
CANCER SCIENCE, 2016, 卷号: 107, 期号: 6, 页码: 782-790
作者:
Wang, Wenqian
;
Liu, Yang
;
Zhao, Zhixin
;
Xie, Chengying
;
Xu, Yongping
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08
Hop
Hsp90
imatinib resistance
thiol oxidation
Y-632
Characteristics of the TCR V beta repertoire in imatinib-resistant chronic myeloid leukemia patients with ABL mutations (SCI收录)
期刊论文
SCIENCE CHINA-LIFE SCIENCES, 2015, 卷号: 58, 页码: 1276-1281
作者:
Xu Ling[1]
;
Lu YuHong[2]
;
Lai Jing[1,2]
;
Yu Wei[3]
;
Zhang YiKai[1]
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/04/25
T cell repertoire
chronic myeloid leukemia
blast crisis
imatinib resistance
BCR-ABL mutation
Curcumin derivative C817 inhibits proliferation of imatinib-resistant chronic myeloid leukemia cells with wild-type or mutant Bcr-Abl in vitro
期刊论文
ACTA PHARMACOLOGICA SINICA, 2014, 卷号: 35, 期号: 3, 页码: 401-409
作者:
Wu, Li-xian
;
Wu, Ying
;
Chen, Rui-jia
;
Liu, Yang
;
Huang, Li-sen
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2019/01/08
chronic myelogenous leukemia
imatinib resistance
Bcr-Abl
mutantion
curcumin
C817
leukemia stem cell
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