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科研机构
西安交通大学 [29]
华中师范大学 [6]
内容类型
期刊论文 [35]
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2019 [2]
2018 [9]
2017 [5]
2016 [4]
2015 [10]
2014 [5]
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Synthesis of Aryl Trimethylstannane via BF3 center dot OEt2-Mediated Cross-Coupling of Hexaalkyl Distannane Reagent with Aryl Triazene at Room Temperature
期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2019, 卷号: 84, 页码: 463-471
作者:
Mao, Shuai
;
Chen, Zhengkai
;
Wang, Lu
;
Khadka, Daulat Bikram
;
Xin, Minhang
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2019/11/19
Discovery of potent anti-inflammatory 4-(4,5,6,7-tetrahydrofuro[3,2-c]pyridin-2-yl) pyrimidin-2-amines for use as Janus kinase inhibitors.
期刊论文
Bioorganic & medicinal chemistry, 2019, 卷号: 27, 期号: 12, 页码: 2592-2597
作者:
Wang, Yazhou*
;
Huang, Wei*
;
Xin, Minhang
;
Chen, Pan
;
Gui, Li
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2019/12/23
Anti-inflammatory
Furo[3,2-c]pyridine
JAK inhibitor
Rheumatoid arthritis
Novel 4-(2-pyrimidinylamino)benzamide derivatives as potent hedgehog signaling pathway inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 页码: 5029-5036
作者:
Xin, Minhang
;
Zhang, Liandi
;
Tu, Chongxing
;
Tang, Feng
;
Wen, Jun
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2019/11/19
SAR
In vivo
Hedgehog signaling pathway inhibitors
4-(2-Pyrimidinylamino)benzamide
Discovery of 2-(aminopyrimidin-5-yl)-4-(morpholin-4-yl)-6- substituted triazine as PI3K and BRAF dual inhibitor.
期刊论文
Future medicinal chemistry, 2018, 卷号: 10, 页码: 2445-2455
作者:
Wang Hui-Yan
;
Shen Ying
;
Zhang Hao
;
Hei Yuan-Yuan
;
Zhao Hong-Yi
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/11/19
BRAF inhibitor
drug design
PI3K inhibitor
antiproliferative effects
PI3K and BRAF dual inhibitor
The development of Bruton's tyrosine kinase (BTK) inhibitors from 2012 to 2017: A mini-review
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 151, 页码: 315-326
作者:
Liang, Chengyuan
;
Tian, Danni
;
Ren, Xiaodong
;
Ding, Shunjun
;
Jia, Minyi
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2019/11/26
Kinase inhibitor
Irreversible inhibitor
Bruton's tyrosine kinase (BTK)
Reversible covalent inhibitor
Introduction of pyrrolidineoxy or piperidineamino group at the 4-position of quinazoline leading to novel quinazoline-based phosphoinositide 3-kinase delta (PI3K delta) inhibitors
期刊论文
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2018, 卷号: 33, 页码: 651-656
作者:
Xin, Minhang
;
Duan, Weiming
;
Feng, Yifan
;
Hei, Yuan-Yuan
;
Zhang, Hao
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/11/26
selectivity
anti-proliferation
PI3K delta inhibitors
4-pyrrolidineoxy
4-piperidineamino
Synthesis and evaluation of 2,9-disubstituted 8-phenylthio/phenylsulfinyl-9H-purine as new EGFR inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 页码: 2173-2185
作者:
Hei, Yuan-Yuan
;
Shen, Ying
;
Wang, Jin
;
Zhang, Hao
;
Zhao, Hong-Yi
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2019/11/26
Antiproliferative effects
Drug design
EGFR-TK inhibitor
Anticancer agent
Purine
Synthesis and biological evaluation of irreversible EGFR tyrosine kinase inhibitors containing pyrido[3,4-d]pyrimidine scaffold
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 页码: 3619-3633
作者:
Zhang, Hao
;
Wang, Jin
;
Zhao, Hong-Yi
;
Yang, Xue-Yan
;
Lei, Hao
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2019/11/26
Pyrido[3,4-d]pyrimidine
Anticancer
Drug design
Irreversible inhibitors
EGFR-TKIs
Novel 6-aryl substituted 4-pyrrolidineaminoquinazoline derivatives as potent phosphoinositide 3-kinase delta (PI3K delta) inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 页码: 2028-2040
作者:
Xin, Minhang
;
Duan, Weiming
;
Feng, Yifan
;
Hei, Yuan-Yuan
;
Zhang, Hao
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2019/11/26
4-Pyrrolidineaminoquinazoline
Structure-activity relationship
Anti-proliferation
PI3K delta inhibitors
6-Aryl
Strategies to target the Hedgehog signaling pathway for cancer therapy
期刊论文
MEDICINAL RESEARCH REVIEWS, 2018, 卷号: 38, 页码: 870-913
作者:
Xin, Minhang
;
Ji, Xinyue
;
De La Cruz, Ladie Kimberly
;
Thareja, Suresh
;
Wang, Binghe
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2019/11/26
sonidegib
hedgehog signaling pathway
Hh inhibitor
basal cell carcinoma
vismodegib
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