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上海药物研究所 [15]
中南大学 [2]
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武汉大学 [1]
上海中医药大学 [1]
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期刊论文 [21]
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2020 [6]
2019 [2]
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Discovery of nitazoxanide-based derivatives as autophagy activators for the treatment of Alzheimer's disease
期刊论文
ACTA PHARMACEUTICA SINICA B, 2020, 卷号: 10, 期号: 4, 页码: 646-666
作者:
Li, Xiaokang
;
Lu, Jian
;
Xu, Yixiang
;
Wang, Jiaying
;
Qiu, Xiaoxia
收藏
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浏览/下载:45/0
  |  
提交时间:2020/07/01
Alzheimer's disease
Autophagy
Nitazoxanide
beta-amyloid
Tau protein
Repurposing antimycotic ciclopirox olamine as a promising anti-ischemic stroke agent
期刊论文
ACTA PHARMACEUTICA SINICA B, 2020, 卷号: 10, 期号: 3, 页码: 434-446
作者:
Feng, Hongxuan
;
Hu, Linghao
;
Zhu, Hongwen
;
Tao, Lingxue
;
Wu, Lei
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2020/07/01
Blood-brain barrier
Brain ischemia
Cell cycle
Inflammation
Neuroprotection
Development of Novel N-hydroxypyridone Derivatives as Potential Anti-Ischemic Stroke Agents
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 3, 页码: 1051-1067
作者:
Hu, Linghao
;
Feng, Hongxuan
;
Zhang, Hongguang
;
Yu, Songda
;
Zhao, Qinyuan
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2020/07/01
Discovery of synergistic activity of fluoroquinolones in combination with antimicrobial peptides against clinical polymyxin-resistant Pseudomonas aeruginosa DK2
期刊论文
CHINESE CHEMICAL LETTERS, 2020, 卷号: 31, 期号: 2, 页码: 413-417
作者:
Zheng, Xinyu
;
Cao, Qiao
;
Cao, Qin
;
Mao, Fei
;
Li, Xiaokang
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2020/07/01
Polymyxin B
Pseudomonas aeruginosa
Fluoroquinolones
Synergy
Cystic fibrosis
Antimicrobial peptides
K2S2O8-promoted direct thiocyanation of pyrazolin-5-ones with ammonium thiocyanate at room temperature
期刊论文
ORGANIC CHEMISTRY FRONTIERS, 2020, 卷号: 7, 期号: 2, 页码: 350-354
作者:
Mao, Xiaokang
;
Ni, Jiabin
;
Xu, Bin
;
Ding, Chunyong
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  |  
浏览/下载:9/0
  |  
提交时间:2020/07/01
Targeting virulence factors as an antimicrobial approach: Pigment inhibitors
期刊论文
MEDICINAL RESEARCH REVIEWS, 2020, 卷号: 40, 期号: 1, 页码: 293-338
作者:
Ni, Shuaishuai
;
Li, Baoli
;
Xu, Yixiang
;
Mao, Fei
;
Li, Xiaokang
收藏
  |  
浏览/下载:62/0
  |  
提交时间:2020/07/01
antimicrobial
colored pathogens
CrtN inhibitor
staphyloxanthin
virulence factor pigment
Copper-Catalyzed Synthesis of gem-Bisarylthio Enamines under Redox-Neutral Conditions
期刊论文
ADVANCED SYNTHESIS & CATALYSIS, 2019, 卷号: 361, 期号: 9, 页码: 2004-2008
作者:
Ni, Jiabin
;
Mao, Xiaokang
;
Zhanga, Ao
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2020/07/01
copper
oxime acetates
disulfides
redox-neutral
gem-bisarylthio enamines
Understanding the topic evolution of scientific literatures like an evolving city: Using Google Word2Vec model and spatial autocorrelation analysis
期刊论文
INFORMATION PROCESSING & MANAGEMENT, 2019, 卷号: 56, 期号: 4
作者:
Hu Kai
;
Luo Qing
;
Qi Kunlun
;
Yang Siluo
;
Mao Jin
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/12/06
Semantic relatedness
Topic evolution
Spatial clustering
Spatial autocorrelation
Word2Vec
Rational Design of Novel Selective Dual-Target Inhibitors of Acetylcholinesterase and Monoamine Oxidase B as Potential Anti-Alzheimer's Disease Agents
期刊论文
ACS chemical neuroscience, 2018
作者:
Xu, Yixiang
;
Zhang, Jian
;
Wang, Huan
;
Mao, Fei
;
Bao, Keting
收藏
  |  
浏览/下载:84/0
  |  
提交时间:2019/01/08
Design, synthesis and evaluation of vilazodone-tacrine hybrids as multitarget-directed ligands against depression with cognitive impairment
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 12, 页码: 3117-3125
作者:
Liu, Wenwen
;
Wang, Huan
;
Li, Xiaokang
;
Xu, Yixiang
;
Zhang, Jian
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2019/01/08
Depression
Cognitive impairment
Multitarget-directed ligand
5-HT1A agonist
5-HT reuptake inhibition
ChE inhibition
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