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上海药物研究所 [29]
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Design, synthesis and bioactivity study of evodiamine derivatives as multifunctional agents for the treatment of hepatocellular carcinoma
期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 114
作者:
Fan, Xiaohong
;
Deng, Jiedan
;
Shi, Tao
;
Wen, Huaixiu
;
Li, Junfang
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2021/11/18
Hepatocellular carcinoma
Topo I
Evodiamine
Cancer-associated fibroblasts (CAFs)
Eucalypglobulusals A-J, Formyl-Phloroglucinol-Terpene Meroterpenoids from Eucalyptus globulus Fruits
期刊论文
JOURNAL OF NATURAL PRODUCTS, 2018, 卷号: 81, 期号: 12, 页码: 2638-2646
作者:
Qin, Xu-Jie
;
Jin, Ling-Yu
;
Yu, Qian
;
Liu, Hui
;
Khan, Afsar
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2019/03/18
A series of camptothecin prodrugs exhibit HDAC inhibition activity
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 16, 页码: 4706-4715
作者:
Zhu, Qiwen
;
Yu, Xumeng
;
Shen, Qianqian
;
Zhang, Qiumeng
;
Su, Mingbo
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2019/01/08
Camptothecin
HDAC
SAHA
Prodrug
New tanshinone I derivatives S222 and S439 similarly inhibit topoisomerase I/II but reveal different p53-dependency in inducing G2/M arrest and apoptosis
期刊论文
BIOCHEMICAL PHARMACOLOGY, 2018, 卷号: 154, 页码: 255-264
作者:
Tian, Qian-Ting
;
Ding, Chun-Yong
;
Song, Shan-Shan
;
Wang, Ying-Qing
;
Zhang, Ao
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  |  
浏览/下载:42/0
  |  
提交时间:2019/01/08
Tanshinone-1
S222
S439
Anticancer targets
DNA topoisomerases
P53
Topoisomerase I inhibitory and photocleavage activity of non-dppz DNA "light switches\' based on ruthenium complexes containing nitro group
期刊论文
APPLIED ORGANOMETALLIC CHEMISTRY, 2018, 卷号: Vol.32 No.8
作者:
Liu, XueWen
;
Huang, Jie
;
Tang, YuXuan
;
Shen, YouMing
;
Lu, JiLin
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2019/12/26
DNA "light switch\'
nitro group
non-dppz
ruthenium complex
topo I inhibition
New designed DNA light switch Ruthenium complexes as DNA photocleavers and Topoisomerase I inhibitors
期刊论文
Applied Organometallic Chemistry, 2018, 卷号: Vol.32 No.4
作者:
Liu, Xue-Wen
;
Xiao, Yang
;
Peng, Wei-Gen
;
Zhao, Li-Jin
;
Shen, You-Ming
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2019/12/26
light switch
phenazine
photocleavage
Ruthenium complex
topo I inhibition
Antiproliferative activities of Amaryllidaceae alkaloids from Lycoris radiata targeting DNA topoisomerase I
期刊论文
SCIENTIFIC REPORTS, 2016, 卷号: 6, 页码: 10
作者:
Chen, Gui-Lin
;
Tian, Yong-Qiang
;
Wu, Jian-Lin
;
Li, Na
;
Guo, Ming-Quan
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  |  
浏览/下载:62/0
  |  
提交时间:2018/12/29
Novel synthetic acridine-based derivatives as topoisomerase Ⅰ inhibitors
期刊论文
2016, 2016
Bin Li
;
Chun-Mei Gao
;
Qin-Sheng Sun
;
Lu-Lu Li
;
Chun-Yan Tan
;
Hong-Xia Liu
;
Yu-Yang Jiang
;
Bin Li
;
Chun-Mei Gao
;
Qin-Sheng Sun
;
Lu-Lu Li
;
Chun-Yan Tan
;
Hong-Xia Liu
;
Yu-Yang Jiang
收藏
  |  
浏览/下载:5/0
Down-regulation of G9a triggers DNA damage response and inhibits colorectal cancer cells proliferation
期刊论文
ONCOTARGET, 2015, 卷号: 6, 期号: 5, 页码: 2917-+
作者:
Zhang, Jie
;
He, Pengxing
;
Xi, Yong
;
Geng, Meiyu
;
Chen, Yi
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08
colorectal cancer
G9a
epigenetics
DNA damage response (DDR)
SN38/CPT
synergistic effect
DNA Interaction, Photocleavage and Topoisomerase I Inhibition by Ru Complex with a New Ligand Possessing Phenazine Unit.
期刊论文
JOURNAL OF FLUORESCENCE, 2015, 卷号: Vol.25 No.5, 页码: 1527-1535
作者:
Liu, Xue-Wen
;
Shen, You-Ming
;
Shu, Jun-Shi
;
Xiao, Yang
;
Zhang, Song-Bai
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/31
Ru(II)
complex
DNA-binding
Photocleavage
Topoisomerase
inhibition
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