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北京大学 [3]
上海药物研究所 [3]
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武汉大学 [2]
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期刊论文 [16]
学位论文 [2]
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Discovery of Potent and Selective CDK9 Degraders for Targeting Transcription Regulation in Triple-Negative Breast Cancer
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 19, 页码: 14822-14847
作者:
Wei, Dan
;
Wang, Hanlin
;
Zeng, Qinghe
;
Wang, Wenjing
;
Hao, Bingbing
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2021/12/16
Tideglusib and Its Analogues As Inhibitors of Staphylococcus aureus SrtA
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 15, 页码: 8442-8457
作者:
Yang, Teng
;
Zhang, Tao
;
Guan, Xiang-Na
;
Dong, Ze
;
Lan, Lefu
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2020/12/24
以病毒样颗粒为“底盘”的流感疫苗仿生合成
学位论文
: 中国科学院大学, 2020
作者:
魏江雪
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2021/09/07
流感疫苗,病毒样颗粒,仿生合成,疫苗合成学,加热装载
FDA-approved drug screen identifies proteasome as a synthetic lethal target in MYC-driven neuroblastoma
期刊论文
ONCOGENE, 2019, 卷号: 38, 期号: 41
作者:
Wang, Jingchao
;
Jiang, Jue
;
Chen, Hui
;
Wang, Liyuan
;
Guo, Hao
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2019/12/05
Developmental toxicity of synthetic phenolic antioxidants to the early life stage of zebrafish
期刊论文
SCIENCE OF THE TOTAL ENVIRONMENT, 2018, 卷号: 643, 页码: 559-568
作者:
Shi, Guoqing
;
Yang, Xiaoxi
;
Sun, Zhendong
;
Wang, Wanyi
;
Zhou, Qunfang
收藏
  |  
浏览/下载:55/0
  |  
提交时间:2019/06/20
Synthetic phenolic antioxidants
Zebrafish embryo (Danio rerio)
Developmental toxicity
Hypothalamic-pituitary-thyroid axis (HPT axis)
Pluripotency biomarker
Phospho-ERK is a biomarker of response to a synthetic lethal drug combination of sorafenib and MEK inhibition in liver cancer
期刊论文
JOURNAL OF HEPATOLOGY, 2018, 卷号: 69, 期号: 5
作者:
Wang, Cun
;
Jin, Haojie
;
Gao, Dongmei
;
Lieftink, Cor
;
Evers, Bastiaan
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/12/05
Hepatocellular carcinoma
CRISPR screen
Sorafenib
MAPK1
Cell-Cycle-Targeting MicroRNAs as Therapeutic Tools against Refractory Cancers
其他
2017-01-01
Hydbring, Per
;
Wang, Yinan
;
Fassl, Anne
;
Li, Xiaoting
;
Matia, Veronica
;
Otto, Tobias
;
Choi, Yoon Jong
;
Sweeney, Katharine E.
;
Suski, Jan M.
;
Yin, Hao
;
Bogorad, Roman L.
;
Goel, Shom
;
Yuzugullu, Haluk
;
Kauffman, Kevin J.
;
Yang, Junghoon
;
Jin, Chong
;
Li, Yingxiang
;
Floris, Davide
;
Swanson, Richard
;
Ng, Kimmie
;
Sicinska, Ewa
;
Anders, Lars
;
Zhao, Jean J.
;
Polyak, Kornelia
;
Anderson, Daniel G.
;
Li, Cheng
;
Sicinski, Piotr
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2017/12/03
BREAST-CANCER
TUMOR-SUPPRESSOR
SYNTHETIC LETHAL
PROSTATE-CANCER
MIR-193A-3P
MYC
TUMORIGENESIS
PROGRESSION
METASTASIS
INHIBITION
CHD1 loss sensitizes prostate cancer to DNA damaging therapy by promoting error-prone double-strand break repair
期刊论文
ANNALS OF ONCOLOGY, 2017
Shenoy, T. R.
;
Boysen, G.
;
Wang, M. Y.
;
Xu, Q. Z.
;
Guo, W.
;
Koh, F. M.
;
Wang, C.
;
Zhang, L. Z.
;
Wang, Y.
;
Gil, V.
;
Aziz, S.
;
Christova, R.
;
Rodrigues, D. N.
;
Crespo, M.
;
Rescigno, P.
;
Tunariu, N.
;
Riisnaes, R.
;
Zafeiriou, Z.
;
Flohr, P.
;
Yuan, W.
;
Knight, E.
;
Swain, A.
;
Ramalho-Santos, M.
;
Xu, D. Y.
;
de Bono, J.
;
Wu, H.
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2017/12/03
chromatin remodeler CHD1
PCa
DDR
homologous recombination
non-homologous end joining
synthetic lethality
REGULATES 53BP1 STABILITY
MAMMALIAN-CELLS
PATHWAY CHOICE
MOUSE MODEL
CHROMATIN
TRANSCRIPTION
CASTRATION
PROTEIN
PTEN
RECRUITMENT
SLC25A22 Promotes Proliferation and Survival of Colorectal Cancer Cells With KRAS Mutations and Xenograft Tumor Progression in Mice via Intracellular Synthesis of Aspartate
期刊论文
GASTROENTEROLOGY, 2016
Wong, Chi Chun
;
Qian, Yun
;
Li, Xiaona
;
Xu, Jiaying
;
Kang, Wei
;
Tong, Joanna H.
;
To, Ka-Fai
;
Jin, Ye
;
Li, Weilin
;
Chen, Huarong
;
Go, Minnie Y. Y.
;
Wu, Jian-Lin
;
Cheng, Ka Wing
;
Ng, Simon S. M.
;
Sung, Joseph J. Y.
;
Cai, Zongwei
;
Yu, Jun
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2017/12/04
Glutamic-Oxaloacetic Transaminase 1
Solute Carrier Family 25 Member 22
Colon Cancer
Glutaminolysis
PHOSPHATE-ACTIVATED GLUTAMINASE
INNER MITOCHONDRIAL-MEMBRANE
ONCOGENIC KRAS
LOCALIZATION
METABOLISM
BRAIN
GLUCOSE
GROWTH
TUMORIGENESIS
BIOSYNTHESIS
microRNA-206 impairs c-Myc-driven cancer in a synthetic lethal manner by directly inhibiting MAP3K13
期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 13
作者:
Han, Han
;
Chen, Yuxing
;
Cheng, Li
;
Prochownik, Edward V.
;
Li, Youjun
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2019/12/05
Myc
microRNA
MAP3K13
breast cancer
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