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The Development of Inhibitors Targeting the Mixed Lineage Leukemia 1 (MLL1)-WD Repeat Domain 5 Protein (WDR5) Protein-Protein Interaction 期刊论文
CURRENT MEDICINAL CHEMISTRY, 2020, 卷号: 27, 期号: 33, 页码: 5530-5542
作者:  Ye, Xiaoqing;  Chen, Gang;  Jin, Jia;  Zhang, Binzhong;  Wang, Yinda
收藏  |  浏览/下载:14/0  |  提交时间:2020/12/24
The identification of novel small-molecule inhibitors targeting WDR5-MLL1 interaction through fluorescence polarization based high-throughput screening 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 4, 页码: 638-645
作者:  Ye, Xiaoqing;  Zhang, Rukang;  Lian, Fulin;  Zhang, Weiyao;  Lu, Wenchao
收藏  |  浏览/下载:3/0  |  提交时间:2020/07/01
Discovery of potent DOT1L inhibitors by AlphaLISA based High Throughput Screening assay 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 8, 页码: 1751-1758
作者:  Song, Yakai;  Li, Linjuan;  Chen, Yantao;  Liu, Jingqiu;  Xiao, Senhao
收藏  |  浏览/下载:42/0  |  提交时间:2019/01/08
Piperidine Alkaloids with Diverse Skeletons from Anacyclus pyrethrum 期刊论文
JOURNAL OF NATURAL PRODUCTS, 2018, 卷号: 81, 期号: 6, 页码: 1474-1482
作者:  Chen, QB (Chen, Qi-Bin);  Gao, J (Gao, Jie);  Zou, GA (Zou, Guo-An);  Xin, XL (Xin, Xue-Lei);  Aisa, HA (Aisa, Haji Akber)
收藏  |  浏览/下载:25/0  |  提交时间:2018/07/16
Melatonin inhibits MLL-rearranged leukemia via RBFOX3/hTERT and NF-κB/COX-2 signaling pathways. 期刊论文
Cancer letters, 2018
作者:  Tang Yan-Lai;  Sun Xi;  Huang Li-Bin;  Liu Xiao-Jian;  Qin Ge
收藏  |  浏览/下载:12/0  |  提交时间:2019/12/26
Piribedil disrupts the MLL1-WDR5 interaction and sensitizes MLL-rearranged acute myeloid leukemia (AML) to doxorubicin-induced apoptosis 期刊论文
CANCER LETTERS, 2018, 卷号: 431, 页码: 150-160
作者:  Zhang, Xiong;  Zheng, Xingling;  Yang, Hong;  Yan, Juan;  Fu, Xuhong
收藏  |  浏览/下载:37/0  |  提交时间:2019/01/08
Development of Potent Type I Protein Arginine Methyltransferase (PRMT) Inhibitors of Leukemia Cell Proliferation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 21, 页码: 8888-8905
作者:  Wang, Chen;  Jiang, Hao;  Jin, Jia;  Xie, Yiqian;  Chen, Zhifeng
收藏  |  浏览/下载:113/0  |  提交时间:2019/01/08
Discovery of Novel Disruptor of Silencing Telomeric 1-Like (DOTI L) Inhibitors using a Target-Specific Scoring Function for the (S)-Adenosyl-L-methionine (SAM)-Dependent Methyltransferase Family 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 5, 页码: 2026-2036
作者:  Wang, Yulan;  Li, Linjuan;  Zhang, Bidong;  Xing, Jing;  Chen, Shijie
收藏  |  浏览/下载:23/0  |  提交时间:2019/01/08
Alkaloid constituents from Viola tianschanica 期刊论文
PHYTOCHEMISTRY, 2017, 卷号: 144, 期号: 12, 页码: 233-242
作者:  Chen, QB (Chen, Qi-Bin);  Aisa, HA (Aisa, Haji Akber);  Aisa, HA
收藏  |  浏览/下载:20/0  |  提交时间:2018/01/19
Aleukemic extramedullary T lymphoid/myeloid bilineage hematopoietic and lymphoid malignancy with progression to bilineage leukemia at relapse: A case report 期刊论文
ONCOLOGY LETTERS, 2017, 卷号: 14, 期号: 6
作者:  Wu, Mengyao;  Li, Xiaoqiu;  Tang, Feng;  Zhu, Ping;  Ding, Tianling
收藏  |  浏览/下载:11/0  |  提交时间:2019/12/05


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