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Synthesis and Biological Evaluation of Oxopyrido[2,3-d] Pyrimidine-7-ones Derivatives as Covalent L85812/T790M Mutant Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors 期刊论文
LETTERS IN DRUG DESIGN & DISCOVERY, 2019, 卷号: 16, 期号: 8, 页码: 826-834
作者:  Niu, Ao;  Wang, Yang;  Yang, Yushe;  Wei, Jianhai;  Ding, Jian
收藏  |  浏览/下载:12/0  |  提交时间:2020/07/01
Synthesis and Biological Activities of Novel 2-Aminobenzimidazoles EGFR~(T790M) Inhibitors 期刊论文
Chinese Journal of Synthetic Chemistry, 2018, 卷号: 26, 期号: 9, 页码: 637-646
作者:  Duan Jingyi;  Zhang Yinyong;  Qian Anran;  Tong Linjiang;  Xie Hua
收藏  |  浏览/下载:28/0  |  提交时间:2019/01/08
The CRISPR/Cas9 system targeting EGFR exon 17 abrogates NF-κB activation via epigenetic modulation of UBXN1 in EGFRwt/vIII glioma cells 期刊论文
Cancer Letters, 2017, 卷号: 388, 页码: 269-280
作者:  Huang K.;  Yang C.;  Wang Q.-X.;  Li Y.-S.;  Fang C.
收藏  |  浏览/下载:1/0  |  提交时间:2019/12/12
The CRISPR/Cas9 system targeting EGFR exon 17 abrogates NF-kappa B activation via epigenetic modulation of UBXN1 in EGFRwt/vIII glioma cells 期刊论文
CANCER LETTERS, 2017, 卷号: 388, 页码: 269-280
作者:  Huang, Kai;  Yang, Chao;  Wang, Qi-xue;  Li, Yan-sheng;  Fang, Chuan
收藏  |  浏览/下载:2/0  |  提交时间:2019/12/12
Synthesis and evaluation of novel non-covalent binding quinazoline glycoside derivatives targeting the L858R and T790M variants of EGFR 期刊论文
RSC ADVANCES, 2016, 卷号: 6, 期号: 43, 页码: 36857-36862
作者:  Zhang, Renshuai;  Chen, Shaopeng;  Zhang, Xiaowei;  Yu, Rilei;  Wan, Shengbiao
收藏  |  浏览/下载:11/0  |  提交时间:2019/01/08
EGFRT790M/IGF1R双重抑制剂的设计、合成及成药性研究 学位论文
广州生物院: 中国科学院大学, 2015
作者:  陳成斌
收藏  |  浏览/下载:61/0  |  提交时间:2018/12/25
Antitumor efficacy of D2C7-(scdsFv)-PE38KDEL, a novel immunotoxin targeting EGFRwt and EGFRvIII, by convection-enhanced delivery in orthotopic brain tumor mouse models 期刊论文
Journal for ImmunoTherapy of Cancer, 2013
作者:  Bao X., Chandramohan V., Keir S.T., Pegram C.N., McLendon R.E., Kuan C.-T., Pastan I.H., Bigner D.D.
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/19
Construction of an Immunotoxin, D2C7-(scdsFv)-PE38KDEL, Targeting EGFRwt and EGFRvIII for Brain Tumor Therapy 期刊论文
CLINICAL CANCER RESEARCH, 2013, 卷号: 19, 期号: 17
作者:  Chandramohan, Vidyalakshmi;  Bao, Xuhui;  Keir, Stephen T.;  Pegram, Charles N.;  Szafranski, Scott E.
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/19
Identification of an Exon 4-Deletion Variant of Epidermal Growth Factor Receptor with Increased Metastasis-Promoting Capacity 期刊论文
Neoplasia, 2011, 卷号: 13, 期号: 5, 页码: 461-IN12
作者:  Wang, Hai;  Zhou, Min;  Shi, Bizhi;  Zhang, Qingli;  Jiang, Hua
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/27


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