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上海药物研究所 [32]
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Design, synthesis, in vitro evaluation of a new pyrrolo[1,2-a]thiazolo[5,4-d]pyrimidinone derivatives as cholinesterase inhibitors against Alzheimer's disease
期刊论文
JOURNAL OF HETEROCYCLIC CHEMISTRY, 2022, 卷号: 59, 期号: 6, 页码: 1086-1101
作者:
Zeng, Y (Zeng, Yan) [1] , [2]
;
Nie, LF (Nie, Lifei) [1]
;
Liu, L (Liu, Liu) [1]
;
Niu, C (Niu, Chao) [1] , [2]
;
Li, Y (Li, Yi) [1] , [2]
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2022/06/21
Twin drug design, synthesis and evaluation of diosgenin derivatives as multitargeted agents for the treatment of vascular dementia
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 37, 页码: 16
作者:
Yang, Gui-Xiang
;
Sun, Jia-Min
;
Zheng, Lu-Lu
;
Zhang, Li
;
Li, Jie
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  |  
浏览/下载:71/0
  |  
提交时间:2021/06/11
Vascular dementia
Diosgenin
Antioxidant
Anti-cholinesterase
Multi-target-directed ligands
Short-term exposure to norfloxacin induces oxidative stress, neurotoxicity and microbiota alteration in juvenile large yellow croaker Pseudosciaena crocea
期刊论文
ENVIRONMENTAL POLLUTION, 2020, 卷号: 267, 页码: 9
作者:
Wang, Xinghuo
;
Hu, Menghong
;
Gu, Huaxin
;
Zhang, Libin
;
Shang, Yueyong
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  |  
浏览/下载:21/0
  |  
提交时间:2021/04/12
AChE
Fish
Intestinal microbiota
Norfloxacin
Oxidative stress
Design, synthesis and cholinesterase inhibitory activity of alpha-mangostin derivatives
期刊论文
NATURAL PRODUCT RESEARCH, 2020
作者:
Chi, Xiao-Qian
;
Hou, Bo
;
Yang, Liu
;
Zi, Cheng-Ting
;
Lv, Yong-Feng
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  |  
浏览/下载:17/0
  |  
提交时间:2021/01/05
Discovery of new multifunctional selective acetylcholinesterase inhibitors: structure-based virtual screening and biological evaluation
期刊论文
JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN, 2019, 卷号: 33, 期号: 5, 页码: 521-530
作者:
Jiang, Cheng-Shi
;
Ge, Yong-Xi
;
Cheng, Zhi-Qiang
;
Song, Jia-Li
;
Wang, Yin-Yin
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2020/07/01
AChE inhibitor
Pharmacophore model
Molecular docking
Anti-A aggregation
Neuroprotective activity
New 4-N-phenylaminoquinoline derivatives as antioxidant, metal chelating and cholinesterase inhibitors for Alzheimer's disease.
期刊论文
Bioorganic chemistry, 2019, 卷号: Vol.93, 页码: 103328
作者:
Rong Cai
;
Li-Ning Wang
;
Jing-Jing Fan
;
Shang-Qi Geng
;
Yu-Ming Liu
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  |  
浏览/下载:9/0
  |  
提交时间:2019/11/21
4-N-phenylaminoquinoline
Alzheimer’s disease
Anti-cholinesterase activity
Antioxidant
Metal chelator
Cholinesterase inhibitory isoquinoline alkaloids from Corydalis mucronifera
期刊论文
2019, 卷号: Vol.159, 页码: 199-207
作者:
Jun Zhang
;
Chen Zhang
;
Fu-Chun Xu
;
Quesheng
;
Qing-Ying Zhang
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  |  
浏览/下载:5/0
  |  
提交时间:2019/04/15
Corydalis
mucronifera
Maxim.
Isoquinoline
alkaloids
Cholinesterase
inhibitory
activity
Enzymatic reaction modulated synthesis of quantum dots for visual detection of cholinesterase activity and inhibitor
期刊论文
2019, 卷号: 292, 页码: 180-186
作者:
Deng, Wenqing[1]
;
Chen, Piaopiao[3,4,5]
;
Hu, Pingyue[1]
;
He, Ziying[1]
;
Zhang, Mei[2]
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/12/06
Structure-activity study of fluorine or chlorine-substituted cinnamic acid derivatives with tertiary amine side chain in acetylcholinesterase and butyrylcholinesterase inhibition
期刊论文
DRUG DEVELOPMENT RESEARCH, 2019, 卷号: Vol.80 No.4, 页码: 438-445
作者:
Gao, XH
;
Tang, JJ
;
Liu, HR
;
Liu, LB
;
Liu, YZ
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2019/12/17
cholinesterase inhibitors
cinnamic acid
halogen
Low Plasma Cholinesterase Activity is Associated With Postoperative Delirium After Noncardiac Surgery in Elderly Patients: A Prospective Observational Study
期刊论文
PSYCHOSOMATICS, 2019, 卷号: 60, 期号: 2, 页码: 190-196
作者:
Zhao, Bao
;
Ni, Yuhua
;
Tian, Xingsong
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  |  
浏览/下载:3/0
  |  
提交时间:2019/12/11
Delirium
PSY0250
Old age
Cholinesterase activity
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