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Predicting and overcoming resistance to CDK9 inhibitors for cancer therapy 期刊论文
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13
作者:  Hua, Chen;  Shena, Lijuan;  Zoua, Fengming;  Wua, Yun;  Wanga, Beilei
收藏  |  浏览/下载:11/0  |  提交时间:2023/11/10
CDK9 inhibitors in cancer research 期刊论文
RSC MEDICINAL CHEMISTRY, 2022
作者:  Huang, Zhi;  Wang, Tianqi;  Wang, Cheng;  Fan, Yan
收藏  |  浏览/下载:7/0  |  提交时间:2022/12/23
Role of FUS-CHOP in Myxoid Liposarcoma via miR-486/CDK4 Axis 期刊论文
BIOCHEMICAL GENETICS, 2021
作者:  Wu, Hao;  Xia, Liming;  Xu, Haichao
收藏  |  浏览/下载:37/0  |  提交时间:2022/01/10
Anti-DLBCL efficacy of DCZ0825 in vitro and in vivo: involvement of the PI3K-AKT-mTOR/JNK pathway 期刊论文
ACTA BIOCHIMICA ET BIOPHYSICA SINICA, 2021, 卷号: 53, 期号: 5, 页码: 575-583
作者:  Hu, Ke;  Li, Bo;  Ma, Ruye;  Yi, Hongfei;  Xu, Zhijian
收藏  |  浏览/下载:68/0  |  提交时间:2021/06/11
Cyclin-dependent kinase inhibitor roscovitine attenuates liver inflammation and fibrosis by influencing initiating steps of liver injury 期刊论文
CLINICAL SCIENCE, 2021, 卷号: 135, 期号: 7, 页码: 925-941
作者:  Liu, Yanjun;  Li, Jiacheng;  Liao, Liping;  Huang, Heming;  Fan, Shijie
收藏  |  浏览/下载:21/0  |  提交时间:2021/08/17
Discovery of selective CDK9 degraders with enhancing antiproliferative activity through PROTAC conversion 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 211, 页码: 11
作者:  Qiu, Xiaqiu;  Li, Yuanqing;  Yu, Bin;  Ren, Jie;  Huang, Huidan
收藏  |  浏览/下载:20/0  |  提交时间:2021/05/24
CDK9  Antitumor  PROTAC  AML  Degrader  
LncRNA UCA1 Antagonizes Arsenic-Induced Cell Cycle Arrest through Destabilizing EZH2 and Facilitating NFATc2 Expression 期刊论文
ADVANCED SCIENCE, 2020, 卷号: 7, 期号: 11, 页码: 1-16
作者:  Dong, Zheng;  Gao, Ming;  Li, Changying;  Xu, Ming;  Liu, Sijin
收藏  |  浏览/下载:22/0  |  提交时间:2021/09/14
ULK1-ATG13 and their mitotic phospho-regulation by CDK1 connect autophagy to cell cycle 期刊论文
PLOS BIOLOGY, 2020, 卷号: 18
作者:  Li, Zhiyuan;  Tian, Xiaofei;  Ji, Xinmiao;  Wang, Junjun;  Chen, Hanxiao
收藏  |  浏览/下载:94/0  |  提交时间:2020/10/29
Design of wogonin-inspired selective cyclin-dependent kinase 9 (CDK9) inhibitors with potent in vitro and in vivo antitumor activity 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 178, 页码: 782-801
作者:  Wang, Jubo;  Li, Tinghan;  Zhao, Tengteng;  Wu, Tizhi;  Liu, Chuang
收藏  |  浏览/下载:21/0  |  提交时间:2020/07/01
DCZ0801, a novel compound, induces cell apoptosis and cell cycle arrest via MAPK pathway in multiple myeloma 期刊论文
ACTA BIOCHIMICA ET BIOPHYSICA SINICA, 2019, 卷号: 51, 期号: 5, 页码: 517-523
作者:  Zhang, Ting;  Li, Bo;  Feng, Qilin;  Xu, Zhijian;  Huang, Cheng
收藏  |  浏览/下载:14/0  |  提交时间:2020/07/01


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