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上海药物研究所 [6]
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吉林大学白求恩第一医... [1]
复旦大学上海医学院 [1]
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期刊论文 [9]
专利 [1]
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Cryo-EM Structure of the Human Cannabinoid Receptor CB2-G(i) Signaling Complex
期刊论文
CELL, 2020, 卷号: 180, 期号: 4, 页码: 645-+
作者:
Xing, Changrui
;
Zhuang, Youwen
;
Xu, Ting-Hai
;
Feng, Zhiwei
;
Zhou, X. Edward
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2020/07/01
Developing pyridazine-3-carboxamides to be CB2 agonists: The design, synthesis, structure-activity relationships and docking studies
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 137, 页码: 598-611
作者:
Qian, Hai-Yan
;
Wang, Zhi-Long
;
Xie, Xiao-Yu
;
Pan, You-Lu
;
Li, Gang-Jian
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2019/01/08
Pyridazine-3-carboxamides
CB2 agonist
Structure-activity relationships
Molecular docking
logP
Amidoalkylindoles as Potent and Selective Cannabinoid Type 2 Receptor Agonists with in Vivo Efficacy in a Mouse Model of Multiple Sclerosis
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 16, 页码: 7067-7083
作者:
Shi, Ying
;
Duan, Yan-Hui
;
Ji, Yue-Yang
;
Wang, Zhi-Long
;
Wu, Yan-Ran
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2019/01/08
Development of Quinazoline/Pyrimidine-2,4(1H,3H)-diones as Agonists of Cannabinoid Receptor Type 2
期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 8, 期号: 6, 页码: 678-681
作者:
Qian, Hai-Yan
;
Wang, Zhi-Long
;
Pan, You-Lu
;
Chen, Li-Li
;
Xie, Xin
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
Cannabinoid receptors
CB2 agonist
structure-activity relationship
molecular modeling
Development of Quinoline-2,4(1H,3H)-diones as Potent and Selective Ligands of the Cannabinoid Type 2 Receptor
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 58, 期号: 15, 页码: 5751-5769
作者:
Han, Shuang
;
Zhang, Fei-Fei
;
Qian, Hai-Yan
;
Chen, Li-Li
;
Pu, Jian-Bin
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  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08
Species Differences in Cannabinoid Receptor 2 and Receptor Responses to Cocaine Self-Administration in Mice and Rats
期刊论文
neuropsychopharmacology, 2015
Zhang, Hai-Ying
;
Bi, Guo-Hua
;
Li, Xia
;
Li, Jie
;
Qu, Hong
;
Zhang, Shi-Jian
;
Li, Chuan-Yun
;
Onaivi, Emmanuel S.
;
Gardner, Eliot L.
;
Xi, Zheng-Xiong
;
Liu, Qing-Rong
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2015/11/13
PROTEIN-COUPLED RECEPTORS
CB2 RECEPTOR
PHARMACOLOGICAL CHARACTERIZATION
SWISS-MODEL
ENDOCANNABINOID SYSTEM
INTRANASAL DELIVERY
SELECTIVE LIGANDS
PLACE PREFERENCE
MESSENGER-RNA
BRAIN
Antinociceptive Effects of Central Administration of the Endogenous Cannabinoid Receptor Type 1 Agonist VDPVNFKLLSH-OH [(m)VD-hemopressin(alpha)], an N-Terminally Extended Hemopressin Peptide
期刊论文
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2014, 卷号: 348, 期号: 2, 页码: 316-323
作者:
Han, ZL
;
Fang, Q
;
Wang, ZL
;
Li, XH
;
Li, N
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2015/12/22
SUPPRESSION OF OUTWARD K+ CURRENTS BY WIN55212-2 IN RAT RETINAL GANGLION CELLS IS INDEPENDENT OF CB1/CB2 RECEPTORS
期刊论文
NEUROSCIENCE, 2013, 卷号: 253
作者:
Zhang, C. -Q.
;
Wu, H. -J.
;
Wang, S. -Y.
;
Yin, S.
;
Lu, X-J.
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/19
cannabinoid receptor
CB1/CB2 receptor agonist
TEA-sensitive K+ current
anandamide
patch-clamp
Presence and regulation of cannabinoid receptors in human retinal pigment epithelial cells
期刊论文
MOLECULAR VISION, 2009, 卷号: 15, 期号: 132-33, 页码: 1243-1251
作者:
Wei, Yan
;
Wang, Xu
;
Wang, Ling
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08
COMPOSED DERIVATIVES OF ARILETERSULFONAMIDAS, THEIR SALTS, EQUIPMENT LIKE AGONIST OF RECEIVER CB1 AND CB2 IN THE TREATMENT OF NEURODEGENERATIVE DISEASES, ISCHEMIAS CEREBRAL, CRANEO-ENCEPHALIC TRAUMATISM, PAINFUL STATES, EMESIS, BACTERIAL OR VIRAL GLAUCOMA, ASTHMA, ANOREXY, INFECTIONS (DIVISIONAL OF CL 37? 98).
专利
作者:
null
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  |  
浏览/下载:3/0
  |  
提交时间:2019/12/05
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