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The Antioxidant Activity and Catalytic Mechanism of Schiff Base Diphenylamines at Elevated Temperatures
期刊论文
INDUSTRIAL & ENGINEERING CHEMISTRY RESEARCH, 2020, 卷号: 59, 期号: 3, 页码: 1031-1037
作者:
Yu, Shasha
;
Wang, Yishan
;
Wang, Shengpei
;
Zhu, Jia
;
Liu, Shenggao
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2020/12/16
HYDROCARBON AUTOXIDATION
INHIBITION
REACTIVITY
CAPACITY
Discovery of a Highly Selective and Potent kappa Opioid Receptor Agonist from N-Cyclopropylmethyl-7 alpha-phenyl-6,14-endoethanotetrahydronorthebaines with Reduced Central Nervous System (CNS) Side Effects Navigated by the Message-Address Concept
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 24, 页码: 11054-11070
作者:
Xiao, Li
;
Wang, Yujun
;
Zhang, Mumei
;
Wu, Weiwei
;
Kong, Linghui
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浏览/下载:92/0
  |  
提交时间:2020/07/01
Discovery of New Selective Butyrylcholinesterase (BChE) Inhibitors with Anti-A beta Aggregation Activity: Structure-Based Virtual Screening, Hit Optimization and Biological Evaluation
期刊论文
MOLECULES, 2019, 卷号: 24, 期号: 14, 页码: 21
作者:
Jiang, Cheng-Shi
;
Ge, Yong-Xi
;
Cheng, Zhi-Qiang
;
Wang, Yin-Yin
;
Tao, Hong-Rui
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  |  
浏览/下载:13/0
  |  
提交时间:2020/07/01
selective BChE inhibitor
virtual screening
structural optimization
molecular dynamics
anti-A beta aggregation
A Small-Molecule Compound Selectively Activates K2P Channel TASK-3 by Acting at Two Distant Clusters of Residues
期刊论文
MOLECULAR PHARMACOLOGY, 2019, 卷号: 96, 期号: 1, 页码: 26-35
作者:
Tian, Fuyun
;
Qiu, Yunguang
;
Lan, Xi
;
Li, Min
;
Yang, Huaiyu
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  |  
浏览/下载:18/0
  |  
提交时间:2020/07/01
Discovery of alkoxy benzamide derivatives as novel BPTF bromodomain inhibitors via structure-based virtual screening
期刊论文
BIOORGANIC CHEMISTRY, 2019, 卷号: 86, 页码: 494-500
作者:
Zhang, Dan
;
Han, Jie
;
Lu, Wenchao
;
Lian, Fulin
;
Wang, Jun
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  |  
浏览/下载:11/0
  |  
提交时间:2020/07/01
Lysine acetylation
Bromodomain
Virtual screening
BPTF inhibitor
Continuation of structure-activity relationship study of novel benzamide derivatives as potential antipsychotics
期刊论文
ARCHIV DER PHARMAZIE, 2019, 卷号: 352, 期号: 4, 页码: 13
作者:
Xu, Mingshuo
;
Guo, Shuang
;
Yang, Feipu
;
Wang, Yu
;
Wu, Chunhui
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  |  
浏览/下载:43/0
  |  
提交时间:2020/07/01
5-HT1A
5-HT2A
catalepsy
D-2
PCP-induced hyperactivity
Preparation and thermal properties of stearic acid-benzamide eutectic mixture expanded graphite composites as phase change materials for thermal energy storage
期刊论文
POWDER TECHNOLOGY, 2019, 卷号: 342, 页码: 131-140
作者:
Ma, Guixiang
;
Sun, Jinhe
;
Zhang, Yue
;
Jing, Yan
;
Jia, Yongzhong
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  |  
浏览/下载:0/0
  |  
提交时间:2021/11/29
Mechanistic Investigation of Au(III)-Catalyzed Cycloisomerizations of N-Propargylcarboxamides
期刊论文
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2019, 卷号: 2019, 期号: 40
作者:
Liu, Yuxia
;
Liu, Peng
;
Ling, Baoping
;
Chen, Guang
;
Chen, Tao
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  |  
浏览/下载:62/0
  |  
提交时间:2019/11/26
AuCl3 catalysis
Cycloisomerization
N-(propargyl)benzamide
Mechanism
Density functional calculations
Discovery of alkoxy benzamide derivatives as novel BPTF bromodomain inhibitors via structure-based virtual screening
期刊论文
Bioorganic chemistry, 2019, 卷号: 86, 页码: 494-500
作者:
Zhang Dan[1]
;
Han Jie[2]
;
Lu Wenchao[3]
;
Lian Fulin[4]
;
Wang Jun[5]
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2019/04/22
BPTF inhibitor
Bromodomain
Lysine acetylation
Virtual screening
1-Arylsulfonyl indoline-benzamides as a new antitubulin agents, with inhibition of histone deacetylase
期刊论文
European Journal of Medicinal Chemistry, 2019, 卷号: Vol.162, 页码: 612-630
作者:
Mei-Jung Lai
;
Ritu Ojha
;
Mei-Hsiang Lin
;
Yi-Min Liu
;
Hsueh-Yun Lee
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2019/12/13
Tubulin
Indoline
Benzamide
HDAC
Cancer
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