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上海药物研究所 [19]
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Optogenetically engineered cell-based graphene transistor for pharmacodynamic evaluation of anticancer drugs
期刊论文
Sensors and Actuators B: Chemical, 2022, 卷号: 358, 页码: 1-11
作者:
Yang J(杨佳)
;
Li GX(李恭新)
;
Zu LP(祖立鹏)
;
Wang WX(王文学)
;
Ge ZX(葛治星)
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2022/03/07
Cell-based biosensor
Optogenetics
Photosensitive proteins
Cancer cells
Graphene transistor
Pharmacodynamic evaluation
Oxidosqualene Cyclases Involved in the Biosynthesis of Diverse Triterpenes in Camellia sasanqua
期刊论文
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2022
作者:
Huang, Liufang
;
Hu, Yonger
;
Huang, Ruoshi
;
Chen, Jiabo
;
Zhang, Xiande
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  |  
浏览/下载:0/0
  |  
提交时间:2024/03/07
oxidosqualene cyclases (OSCs)
Camellia sasanqua
triterpene biosynthesis
catalytic mechanism
Marine bacterial exopolysaccharide EPS11 inhibits migration and invasion of liver cancer cells by directly targeting collagen I
期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2021, 卷号: 297, 期号: 4, 页码: 12
作者:
Liu, Ge
;
Liu, Rui
;
Shan, Yeqi
;
Sun, Chaomin
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  |  
浏览/下载:28/0
  |  
提交时间:2022/01/05
Novel poly (ADP-ribose) polymerases inhibitor DHC-1 exhibits in vitro and in vivo anticancer activity on BRCA-deficient pancreatic cancer cells
期刊论文
FOOD AND CHEMICAL TOXICOLOGY, 2021, 卷号: 147, 页码: 10
作者:
Wu, Xiaochen
;
Li, Qiqi
;
Zhang, Fan
;
Wang, Lijun
;
Wang, Jun
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  |  
浏览/下载:38/0
  |  
提交时间:2021/04/21
PARP inhibitor
BRCA
Pancreatic cancer
Iridin Prevented Against Lipopolysaccharide-Induced Inflammatory Responses of Macrophages via Inactivation of PKM2-Mediated Glycolytic Pathways
期刊论文
JOURNAL OF INFLAMMATION RESEARCH, 2021, 卷号: 14
作者:
Ying, Zhen-Hua
;
Li, Hui-Min
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  |  
浏览/下载:29/0
  |  
提交时间:2021/04/26
isoflavone
glycolysis
Warburg effect
PKM2
JAK/STATs
NF-kappa B
Diterpenoids from Euphorbia royleana reverse P-glycoprotein-mediated multidrug resistance in cancer cells
期刊论文
PHYTOCHEMISTRY, 2020, 卷号: 176, 页码: -
作者:
Shaker, Sharpkate
;
Sang, Jun
;
Yan, Xue-Long
;
Fan, Run-Zhu
;
Tang, Gui-Hua
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  |  
浏览/下载:36/0
  |  
提交时间:2020/08/07
INGOL
LATEX
ESTERS
PLANTS
Rational Coarse-Grained Molecular Dynamics Simulations of Supramolecular Anticancer Nanotubes
期刊论文
JOURNAL OF PHYSICAL CHEMISTRY B, 2019, 卷号: 123, 期号: 50, 页码: 10582-10593
作者:
Manandhar, Anjela
;
Chakraborty, Kaushik
;
Tang, Phu K.
;
Kang, Myungshim
;
Zhang, Pengcheng
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  |  
浏览/下载:15/0
  |  
提交时间:2020/07/01
Structure-Based Discovery and Development of a Series of Potent and Selective Bromodomain and Extra-Terminal Protein Inhibitors
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 18, 页码: 8642-8663
作者:
Hu, Jianping
;
Tian, Chang-Qing
;
Damaneh, Mohammadali Soleimani
;
Li, Yanlian
;
Cao, Danyan
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  |  
浏览/下载:11/0
  |  
提交时间:2020/07/01
Design of wogonin-inspired selective cyclin-dependent kinase 9 (CDK9) inhibitors with potent in vitro and in vivo antitumor activity
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 178, 页码: 782-801
作者:
Wang, Jubo
;
Li, Tinghan
;
Zhao, Tengteng
;
Wu, Tizhi
;
Liu, Chuang
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  |  
浏览/下载:21/0
  |  
提交时间:2020/07/01
Wogonin
CDK9
AML
Flavonoid
Antitumor
Design, synthesis and biological evaluation of bromophenol-thiazolylhydrazone hybrids inhibiting the interaction of translation initiation factors eIF4E/eIF4G as multifunctional agents for cancer treatment
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 177, 页码: 153-170
作者:
Wang, Lijun
;
Guo, Chuanlong
;
Li, Xiuxue
;
Yu, Xuemin
;
Li, Xiangqian
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  |  
浏览/下载:184/0
  |  
提交时间:2019/08/29
Bromophenol-thiazolylhydrazone hybrids
Synthesis
Multifunctional agents
eIF4E/eIF4G interaction
Autophagy
ROS
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