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Discovery of Pteridin-7(8H)-one-Based Irreversible Inhibitors Targeting the Epidermal Growth Factor Receptor (EGFR) Kinase T790M/L858R Mutant 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 20
Zhou, Wei; Liu, Xiaofeng; Tu, Zhengchao; Zhang, Lianwen; Ku, Xin; Bai, Fang; Zhao, Zhenjiang; Xu, Yufang; Ding, Ke; Li, Honglin
收藏  |  浏览/下载:16/0  |  提交时间:2016/12/16
1-Phenyl-4-benzoyl-1H-1,2,3-triazoles as Orally Bioavailable Transcriptional Function Suppressors of Estrogen-Related Receptor alpha 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 11
Xu, Shilin; Zhuang, Xiaoxi; Pan, Xiaofen; Zhang, Zhang; Duan, Lei; Liu, Yingxue; Zhang, Lianwen; Ren, Xiaomei; Ding, Ke
收藏  |  浏览/下载:15/0  |  提交时间:2016/12/16
Discovery of Pteridin-7(8H)-one-Based Irreversible Inhibitors Targeting the Epidermal Growth Factor Receptor (EGFR) Kinase T790M/L858R Mutant 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 20
作者:  Tu, Zhengchao;  Liu, Xiaofeng;  Ku, Xin;  Bai, Fang;  Zhou, Wei
收藏  |  浏览/下载:14/0  |  提交时间:2018/12/13
Pyrimido[4,5-d]pyrimidin-4(1H)-one Derivatives as Selective Inhibitors of EGFR Threonine(790) to Methionine(790) (T790M) Mutants 期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2013, 卷号: 52, 期号: 32
作者:  Zhang, Lianwen;  Ding, Ke;  Wang, Shaomeng;  Ren, Xiaomei;  Li, Honglin
收藏  |  浏览/下载:39/0  |  提交时间:2018/12/13
1-Phenyl-4-benzoyl-1H-1,2,3-triazoles as Orally Bioavailable Transcriptional Function Suppressors of Estrogen-Related Receptor alpha 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 11
作者:  Liu, Yingxue;  Xu, Shilin;  Zhuang, Xiaoxi;  Pan, Xiaofen;  Zhang, Zhang
收藏  |  浏览/下载:14/0  |  提交时间:2018/12/13
Design, Synthesis, and Biological Evaluation of 2-Oxo-3,4-dihydropyrimido[4,5-d]pyrimidinyl Derivatives as New Irreversible Epidermal Growth Factor Receptor Inhibitors with Improved Pharmacokinetic Properties 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 21
作者:  Xu, Tianfeng;  Ding, Ke;  Ren, Xiaomei;  Tu, Zhengchao;  Lu, Xiaoyun
收藏  |  浏览/下载:8/0  |  提交时间:2018/12/13
Pyrimido[4,5-d]pyrimidin-4(1H)-one Derivatives as Selective Inhibitors of EGFR Threonine(790) to Methionine(790) (T790M) Mutants 期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2013, 卷号: 52, 期号: 32
Xu, Tianfeng; Zhang, Lianwen; Xu, Shilin; Yang, Chao-Yie; Luo, Jinfeng; Ding, Fang; Lu, Xiaoyun; Liu, Yingxue; Tu, Zhengchao; Li, Shiliang; Pei, Duanqing; Cai, Qian; Li, Honglin; Ren, Xiaomei; Wang, Shaomeng; Ding, Ke
收藏  |  浏览/下载:50/0  |  提交时间:2016/12/16
Design, Synthesis, and Biological Evaluation of 2-Oxo-3,4-dihydropyrimido[4,5-d]pyrimidinyl Derivatives as New Irreversible Epidermal Growth Factor Receptor Inhibitors with Improved Pharmacokinetic Properties 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 21
Xu, Shilin; Xu, Tianfeng; Zhang, Lianwen; Zhang, Zhang; Luo, Jinfeng; Liu, Yingxue; Lu, Xiaoyun; Tu, Zhengchao; Ren, Xiaomei; Ding, Ke
收藏  |  浏览/下载:14/0  |  提交时间:2016/12/16


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