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Pharmacokinetics-Driven Optimization of 4(3H)-Pyrimidinones as Phosphodiesterase Type 5 Inhibitors Leading to TPN171, a Clinical Candidate for the Treatment of Pulmonary Arterial Hypertension 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 10, 页码: 4979-4990
作者:  Wang, Zhen;  Jiang, Xiangrui;  Zhang, Xianglei;  Tian, Guanghui;  Yang, Rulei
收藏  |  浏览/下载:39/0  |  提交时间:2020/07/01
New and Practical Synthesis of N-(3-Cyano-7-ethoxy-4-oxo-1, 4-dihydroquinolin-6-yl)acetamide 期刊论文
JOURNAL OF HETEROCYCLIC CHEMISTRY, 2014, 卷号: 51, 期号: 3, 页码: 866-868
作者:  Ma, Wenpeng;  Mao, Yongjun;  Xie, Kai;  Zhu, Qifeng;  Zhang, Rongxia
收藏  |  浏览/下载:51/0  |  提交时间:2019/01/08
Design, Synthesis, and Pharmacological Evaluation of Monocyclic Pyrimidinones as Novel Inhibitors of PDE5 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2012, 卷号: 55, 期号: 23, 页码: 10540-10550
作者:  Wang, Guan;  Liu, Zheng;  Chen, Tiantian;  Wang, Zhen;  Yang, Huaiyu
收藏  |  浏览/下载:21/0  |  提交时间:2019/01/08
A New and Improved Process for N-(4-Chloro-3-cyano-7-ethoxyquinolin-6-yl)acetamide 期刊论文
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2012, 卷号: 16, 期号: 12, 页码: 1970-1973
作者:  Mao, Yongjun;  Liu, Zheng;  Yang, Xiaojun;  Xia, Xiangfei;  Zhang, Rongxia
收藏  |  浏览/下载:22/0  |  提交时间:2019/01/08
Improved Preparation of 3-(1,1-Dimethylallyl)decursinol 期刊论文
JOURNAL OF HETEROCYCLIC CHEMISTRY, 2009, 卷号: 46, 期号: 3, 页码: 560-562
作者:  Jiang, Xiangrui;  Li, Jianfeng;  Zhang, Rongxia;  Guo, Hongli;  Huang, Shaolei
收藏  |  浏览/下载:13/0  |  提交时间:2019/01/08
An improved preparation process for gemcitabine 期刊论文
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2008, 卷号: 12, 期号: 5, 页码: 888-891
作者:  Jiang, Xiangrui;  Li, Jianfeng;  Zhang, Rongxia;  Zhu, Yi;  Shen, Jingshan
收藏  |  浏览/下载:16/0  |  提交时间:2019/01/08


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