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Allosteric Modulators Enhancing GLP-1 Binding to GLP-1R via a Transmembrane Site 期刊论文
ACS CHEMICAL BIOLOGY, 2021, 卷号: 16, 期号: 11, 页码: 2444-2452
作者:  Wang, Jiang;  Yang, Dehua;  Cheng, Xi;  Yang, Linlin;  Wang, Zhaohui
收藏  |  浏览/下载:26/0  |  提交时间:2022/01/04
Discovery of an Inhibitor for the TREK-1 Channel Targeting an Intermediate Transition State of Channel Gating 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 19, 页码: 10972-10983
作者:  Ma, Yuqin;  Luo, Qichao;  Fu, Jie;  Che, Yanxin;  Guo, Fei
收藏  |  浏览/下载:11/0  |  提交时间:2021/05/24
Selective N-glycan editing on living cell surfaces to probe glycoconjugate function 期刊论文
NATURE CHEMICAL BIOLOGY, 2020, 页码: 15
作者:  Tang, Feng;  Zhou, Mang;  Qin, Ken;  Shi, Wei;  Yashinov, Ansor
收藏  |  浏览/下载:72/0  |  提交时间:2020/07/01
TREK Channel Family Activator with a Well-Defined Structure-Activation Relationship for Pain and Neurogenic Inflammation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 7, 页码: 3665-3677
作者:  Qiu, Yunguang;  Huang, Lu;  Fu, Jie;  Han, Chenxia;  Fang, Jing
收藏  |  浏览/下载:44/0  |  提交时间:2020/07/01
Selective activation of TWIK-related acid-sensitive K+ 3 subunit-containing channels is analgesic in rodent models 期刊论文
SCIENCE TRANSLATIONAL MEDICINE, 2019, 卷号: 11, 期号: 519, 页码: 12
作者:  Liao, Ping;  Qiu, Yunguang;  Mo, Yiqing;  Fu, Jie;  Song, Zhenpeng
收藏  |  浏览/下载:30/0  |  提交时间:2020/07/01
A Small-Molecule Compound Selectively Activates K2P Channel TASK-3 by Acting at Two Distant Clusters of Residues 期刊论文
MOLECULAR PHARMACOLOGY, 2019, 卷号: 96, 期号: 1, 页码: 26-35
作者:  Tian, Fuyun;  Qiu, Yunguang;  Lan, Xi;  Li, Min;  Yang, Huaiyu
收藏  |  浏览/下载:18/0  |  提交时间:2020/07/01
Structure-Based Discovery of a Subtype-Selective Inhibitor Targeting a Transient Receptor Potential Vanilloid Channel 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 3, 页码: 1373-1384
作者:  Chai, Hao;  Cheng, Xi;  Zhou, Bin;  Zhao, Lifen;  Lin, Xianhua
收藏  |  浏览/下载:36/0  |  提交时间:2020/07/01
Nano-Structural Effects on Gene Transfection: Large, Botryoid-Shaped Nanoparticles Enhance DNA Delivery via Macropinocytosis and Effective Dissociation 期刊论文
THERANOSTICS, 2019, 卷号: 9, 期号: 6, 页码: 1580-1598
作者:  Zhang, Wenyuan;  Kang, Xuejia;  Yuan, Bo;  Wang, Huiyuan;  Zhang, Tao
收藏  |  浏览/下载:20/0  |  提交时间:2020/07/01
Concentration Dependent Effects of Ca~(2+) and Mg~(2+) on the Phosphatidylethanolamine-Phosphatidylglycerol Bilayer 期刊论文
Acta Physica-Chimica Sinica, 2019, 卷号: 35, 期号: 8, 页码: 840
作者:  Zhang Tao;  Qiu Yunguang;  Luo Qichao;  Cheng Xi;  Zhao Lifen
收藏  |  浏览/下载:11/0  |  提交时间:2020/12/24
Design, synthesis, and biological evaluation of 2-(phenoxyaryl)-3-urea derivatives as novel P2Y(1) receptor antagonists 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 158, 页码: 302-310
作者:  Peng, Jingjing;  Zhao, Lifen;  Wang, Lanlan;  Chen, Hui;  Qiu, Yunguang
收藏  |  浏览/下载:47/0  |  提交时间:2019/01/08


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