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A unique hormonal recognition feature of the human glucagon-like peptide-2 receptor 期刊论文
CELL RESEARCH, 2020, 页码: 11
作者:  Sun, Wen;  Chen, Li-Nan;  Zhou, Qingtong;  Zhao, Li-Hua;  Yang, Dehua
收藏  |  浏览/下载:84/0  |  提交时间:2020/12/24
Development of Bisindole-Substituted Aminopyrazoles as Novel GSK-3 beta Inhibitors with Suppressive Effects against Microglial Inflammation and Oxidative Neurotoxicity 期刊论文
ACS CHEMICAL NEUROSCIENCE, 2020, 卷号: 11, 期号: 20, 页码: 3398-3408
作者:  Liu, Jian-Guo;  Zhao, Danfeng;  Gong, Qi;  Bao, Fengxia;  Chen, Wen-Wen
收藏  |  浏览/下载:16/0  |  提交时间:2021/05/24
Structural basis for activation of the growth hormone-releasing hormone receptor 期刊论文
NATURE COMMUNICATIONS, 2020, 卷号: 11, 期号: 1, 页码: 10
作者:  Zhou, Fulai;  Zhang, Huibing;  Cong, Zhaotong;  Zhao, Li-Hua;  Zhou, Qingtong
收藏  |  浏览/下载:23/0  |  提交时间:2020/12/21
Evaluation of biased agonism mediated by dual agonists of the GLP-1 and glucagon receptors 期刊论文
BIOCHEMICAL PHARMACOLOGY, 2020, 卷号: 180, 页码: 16
作者:  Darbalaei, Sanaz;  Yuliantie, Elita;  Dai, Antao;  Chang, Rulue;  Zhao, Peishen
收藏  |  浏览/下载:19/0  |  提交时间:2020/12/21
Pharmacological characterization of mono-, dual- and tri-peptidic agonists at GIP and GLP-1 receptors 期刊论文
BIOCHEMICAL PHARMACOLOGY, 2020, 卷号: 177, 页码: 13
作者:  Yuliantie, Elita;  Darbalaei, Sanaz;  Dai, Antao;  Zhao, Peishen;  Yang, Dehua
收藏  |  浏览/下载:22/0  |  提交时间:2020/12/24
Structure-based design of antiviral drug candidates targeting the SARS-CoV-2 main protease 期刊论文
SCIENCE, 2020, 卷号: 368, 期号: 6497, 页码: 1331-+
作者:  Dai, Wenhao;  Zhang, Bing;  Jiang, Xia-Ming;  Su, Haixia;  Li, Jian
收藏  |  浏览/下载:30/0  |  提交时间:2020/12/24
Discovery of a Potent and Selective NF-kappa B-Inducing Kinase (NIK) Inhibitor That Has Anti-inflammatory Effects in Vitro and in Vivo 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 8, 页码: 4388-4407
作者:  Li, Zhiqiang;  Li, Xinzhi;  Su, Ming-Bo;  Gao, Li-Xin;  Zhou, Yu-Bo
收藏  |  浏览/下载:28/0  |  提交时间:2020/07/01
Structural basis of G(s) and G(i) recognition by the human glucagon receptor 期刊论文
SCIENCE, 2020, 卷号: 367, 期号: 6484, 页码: 1346-+
作者:  Qiao, Anna;  Han, Shuo;  Li, Xinmei;  Li, Zhixin;  Zhao, Peishen
收藏  |  浏览/下载:38/0  |  提交时间:2020/07/01
Discovery of aryl sulfonamide-selective Nav1.7 inhibitors with a highly hydrophobic ethanoanthracene core 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 卷号: 41, 期号: 3, 页码: 293-302
作者:  Wang, Jin-tao;  Zheng, Yue-ming;  Chen, Yue-ting;  Gu, Min;  Gao, Zhao-bing
收藏  |  浏览/下载:44/0  |  提交时间:2020/07/01
A Novel G Protein-Biased and Subtype-Selective Agonist for a G Protein-Coupled Receptor Discovered from Screening Herbal Extracts 期刊论文
ACS CENTRAL SCIENCE, 2020, 卷号: 6, 期号: 2, 页码: 213-225
作者:  Zhang, Bingjie;  Zhao, Simeng;  Yang, Dehua;  Wu, Yiran;  Xin, Ye
收藏  |  浏览/下载:36/0  |  提交时间:2020/07/01


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