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科研机构
合肥物质科学研究院 [3]
北京大学 [1]
华南理工大学 [1]
安徽大学 [1]
内容类型
期刊论文 [6]
发表日期
2017 [6]
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Discovery of 1-(4-(4-Amino-3-(4-(2-morpholinoethoxy)-phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)phenyl)-3-(5-(tert-butyl)isoxazol-3-yl)urea (CHMFL-FLT3-213) as a Highly Potent Type II FLT3 Kinase Inhibitor Capable of Overcoming a Variety of FLT3 Kinase Mutants in FLT3-ITD Positive AML
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 20, 页码: 8407-8424
作者:
Wang, Aoli
;
Li, Xixiang
;
Chen, Cheng
;
Wu, Hong
;
Qi, Ziping
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2019/06/17
Discovery of N-(3-(5-((3-acrylamido-4-(morpholine-4-carbonyl) phenyl)amino)-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl)-4-(tert-butyl)benzamide (CHMFL-BTK-01) as a highly selective irreversible Bruton's tyrosine kinase (BTK) inhibitor
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 131, 页码: 107-125
作者:
Liang, Qianmao
;
Chen, Yongfei
;
Yu, Kailin
;
Chen, Cheng
;
Zhang, Shouxiang
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2018/07/26
Btk
Irreversible Inhibitor
Kinase Inhibitor
Structure-activity Relationship
B-cell Lymphoma
Discovery of 2-((3-Acrylamido-4-methylphenyl)amino)-N-(2-methyl5-(3,4,5-trimethoxybenzamido)phenyI)-4-(methylamino)pyrimidine-5-carboxamide (CHMFL-BMX-078) as a Highly Potent and Selective Type II Irreversible Bone Marrow Kinase in the X Chromosome (BMX) Kinase Inhibitor
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 5, 页码: 1793-1816
作者:
Liang, Xiaofei
;
Lv, Fengchao
;
Wang, Beilei
;
Yu, Kailin
;
Wu, Hong
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  |  
浏览/下载:724/0
  |  
提交时间:2018/07/04
Discovery of 2-((3-Acrylamido-4-methylphenyl)amino)-N-(2-methyl5-(3,4,5-trimethoxyben zamido)phenyI)-4-(methylamino)pyrimidine-5-carboxamide (CHMFL-BMX-078) as a Highly Potent and Selective Type II Irreversible Bone Marrow Kinase in the X Chro
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017
Liang, Xiaofei
;
Lv, Fengchao
;
Wang, Beilei
;
Yu, Kailin
;
Wu, Hong
;
Qi, Ziping
;
Jiang, Zongru
;
Chen, Cheng
;
Wang, Aoli
;
Miao, Weili
;
Wang, Wenchao
;
Hu, Zhenquan
;
Liu, Juan
;
Liu, Xiaochuan
;
Zhao, Zheng
;
Wang, Li
;
Zhang, Shanchuan
;
Ye, Zi
;
Wang, Chu
;
Ren, Tao
;
Wang, Yinsheng
;
Liu, Qingsong
;
Liu, Jing
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2017/12/03
GROWTH-FACTOR RECEPTOR
TYROSINE KINASE
COVALENT
ETK/BMX
FAMILY
CELLS
GENE
BTK
ACTIVATION
EXPRESSION
Novel reassortment of avian influenza A(H7N9) virus with subtype H6N6 and H5N6 viruses circulating in Guangdong Province, China
期刊论文
Journal of Infection, 2017, 卷号: Vol.75 No.2, 页码: 179-182
作者:
Hu,Mingda
;
Liang,Long
;
Ren,Hongguang
;
Yue,Junjie
;
Jin,Yuan
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  |  
浏览/下载:7/0
  |  
提交时间:2019/04/22
Nickel hexacyanoferrate/carbon composite as a high-rate and long-life cathode material for aqueous hybrid energy storage
期刊论文
CHEMICAL COMMUNICATIONS, 2017, 卷号: 53, 页码: 10556-10559
作者:
Zhang, Dapeng[1]
;
Zhang, Junshu[1]
;
Yang, Zengxu[1]
;
Ren, Xiaochuan[2]
;
Mao, Hongzhi[1]
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/04/24
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