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Discovery of novel BET inhibitors by drug repurposing of nitroxoline and its analogues 期刊论文
ORGANIC & BIOMOLECULAR CHEMISTRY, 2017, 卷号: 15, 期号: 44, 页码: 9352-9361
作者:  Jiang, Hao;  Xing, Jing;  Wang, Chen;  Zhang, Hao;  Yue, Liyan
收藏  |  浏览/下载:108/0  |  提交时间:2019/01/08
PI-273, a Substrate-Competitive, Specific Small-Molecule Inhibitor of PI4KII alpha, Inhibits the Growth of Breast Cancer Cells 期刊论文
CANCER RESEARCH, 2017, 卷号: 77, 期号: 22, 页码: 6253-6266
作者:  Li, Jiangmei;  Gao, Zhen;  Zhao, Dan;  Zhang, Lunfeng;  Qiao, Xinhua
收藏  |  浏览/下载:24/0  |  提交时间:2019/01/08
Development of Potent Type I Protein Arginine Methyltransferase (PRMT) Inhibitors of Leukemia Cell Proliferation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 21, 页码: 8888-8905
作者:  Wang, Chen;  Jiang, Hao;  Jin, Jia;  Xie, Yiqian;  Chen, Zhifeng
收藏  |  浏览/下载:113/0  |  提交时间:2019/01/08
Discovery of potent 2,4-difluoro-linker poly(ADP-ribose) polymerase 1 inhibitors with enhanced water solubility and in vivo anticancer efficacy 期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 11, 页码: 1521-1532
作者:  Chen, Wen-hua;  Song, Shan-shan;  Qi, Ming-hui;  Huan, Xia-juan;  Wang, Ying-qing
收藏  |  浏览/下载:26/0  |  提交时间:2019/01/08
Label-free brainwide visualization of senile plaque using cryo-micro-optical sectioning tomography 期刊论文
OPTICS LETTERS, 2017, 卷号: 42, 期号: 21, 页码: 4247-4250
作者:  Luo, Yilin;  Wang, Anle;  Liu, Mengmeng;  Lei, Tian;  Zhang, Xiaochuan
收藏  |  浏览/下载:30/0  |  提交时间:2019/01/08
Computational Studies on Acetylcholinesterases 期刊论文
MOLECULES, 2017, 卷号: 22, 期号: 8
作者:  Xu, Yechun;  Cheng, Shanmei;  Sussman, Joel L.;  Silman, Israel;  Jiang, Hualiang
收藏  |  浏览/下载:17/0  |  提交时间:2019/01/08
Potent, Selective, and Cell Active Protein Arginine Methyltransferase 5 (PRMT5) Inhibitor Developed by Structure-Based Virtual Screening and Hit Optimization 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 14, 页码: 6289-6304
作者:  Mao, Ruifeng;  Shao, Jingwei;  Zhu, Kongkai;  Zhang, Yuanyuan;  Ding, Hong
收藏  |  浏览/下载:91/0  |  提交时间:2019/01/08
Machine-Learning-Assisted Approach for Discovering Novel Inhibitors Targeting Bromodomain-Containing Protein 4 期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2017, 卷号: 57, 期号: 7, 页码: 1677-1690
作者:  Xing, Jing;  Lu, Wenchao;  Liu, Rongfeng;  Wang, Yulan;  Xie, Yiqian
收藏  |  浏览/下载:23/0  |  提交时间:2019/01/08
Structure-activity relationships of the antimalarial agent artemisinin and the research progress on the artemisinin analogues with novel pharmacological actions 期刊论文
Kexue Tongbao/Chinese Science Bulletin, 2017, 卷号: 62, 期号: 18, 页码: 1948-1963
作者:  Zheng, Mingyue;  Liu, Gang;  Tang, Wei;  Zuo, Jianping;  Zhang, Ao
收藏  |  浏览/下载:13/0  |  提交时间:2019/01/08
Structure of the full-length glucagon class b g-protein-coupled receptor 期刊论文
Nature, 2017, 卷号: 546, 期号: 7657, 页码: 259-+
作者:  Zhang, Haonan;  Qiao, Anna;  Yang, Dehua;  Yang, Linlin;  Dai, Antao
收藏  |  浏览/下载:48/0  |  提交时间:2019/04/23


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