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Pharmacologic characterization of SHR8443, a novel dual inhibitor of phosphatidylinositol 3-kinase and mammalian target of rapamycin 期刊论文
ONCOTARGET, 2017, 卷号: 8, 期号: 64, 页码: 107977-107990
作者:  Xie, Chengying;  Chen, Xiangling;  Zheng, Mingyue;  Liu, Xiaohong;  Wang, Hongbin
收藏  |  浏览/下载:27/0  |  提交时间:2019/01/08
Aspirin Inhibits Cancer Metastasis and Angiogenesis via Targeting Heparanase 期刊论文
CLINICAL CANCER RESEARCH, 2017, 卷号: 23, 期号: 20, 页码: 6267-6278
作者:  Dai, Xiaoyang;  Yan, Juan;  Fu, Xuhong;  Pan, Qiuming;  Sun, Danni
收藏  |  浏览/下载:32/0  |  提交时间:2019/01/08
Design, Synthesis, and Pharmacological Evaluation of Novel Multisubstituted Pyridin-3-amine Derivatives as Multitargeted Protein Kinase Inhibitors for the Treatment of Non-Small Cell Lung Cancer 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 14, 页码: 6018-6035
作者:  Zhu, Wei;  Chen, Hui;  Wang, Yulan;  Wang, Jiang;  Peng, Xia
收藏  |  浏览/下载:20/0  |  提交时间:2019/01/08
RD-Metabolizer: an integrated and reaction types extensive approach to predict metabolic sites and metabolites of drug-like molecules 期刊论文
CHEMISTRY CENTRAL JOURNAL, 2017, 卷号: 11
作者:  Meng, Jiajia;  Li, Shiliang;  Liu, Xiaofeng;  Zheng, Mingyue;  Li, Honglin
收藏  |  浏览/下载:17/0  |  提交时间:2019/01/08
Machine-Learning-Assisted Approach for Discovering Novel Inhibitors Targeting Bromodomain-Containing Protein 4 期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2017, 卷号: 57, 期号: 7, 页码: 1677-1690
作者:  Xing, Jing;  Lu, Wenchao;  Liu, Rongfeng;  Wang, Yulan;  Xie, Yiqian
收藏  |  浏览/下载:23/0  |  提交时间:2019/01/08
青蒿素及其衍生物的抗疟构效关系研究和治疗新适应症衍生物的发现 期刊论文
科学通报, 2017, 卷号: 62, 期号: 18, 页码: 1948-1963
作者:  郑明月;  刘刚;  唐炜;  左建平;  张翱
收藏  |  浏览/下载:44/0  |  提交时间:2019/01/08
Structure-activity relationships of the antimalarial agent artemisinin and the research progress on the artemisinin analogues with novel pharmacological actions 期刊论文
Kexue Tongbao/Chinese Science Bulletin, 2017, 卷号: 62, 期号: 18, 页码: 1948-1963
作者:  Zheng, Mingyue;  Liu, Gang;  Tang, Wei;  Zuo, Jianping;  Zhang, Ao
收藏  |  浏览/下载:13/0  |  提交时间:2019/01/08
Discovery of novel trimethoxy-ring BRD4 bromodomain inhibitors: AlphaScreen assay, crystallography and cell-based assay 期刊论文
MEDCHEMCOMM, 2017, 卷号: 8, 期号: 6, 页码: 1322-1331
作者:  Chen, Zhifeng;  Zhang, Hao;  Liu, Shien;  Xie, Yiqian;  Jiang, Hao
收藏  |  浏览/下载:90/0  |  提交时间:2019/01/08
Discovery and optimization of selective inhibitors of protein arginine methyltransferase 5 by docking-based virtual screening 期刊论文
ORGANIC & BIOMOLECULAR CHEMISTRY, 2017, 卷号: 15, 期号: 17, 页码: 3648-3661
作者:  Ye, Yan;  Zhang, Bidong;  Mao, Ruifeng;  Zhang, Chenhua;  Wang, Yulan
收藏  |  浏览/下载:22/0  |  提交时间:2019/01/08
舵机折叠翼展开性能及实验 期刊论文
机械强度, 2017, 页码: 230-234
作者:  刘断尘;  韩雪峰;  张跃;  张明月;  刘晓东
收藏  |  浏览/下载:21/0  |  提交时间:2018/04/09


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