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Identification and Structure-Activity Relationship (SAR) of potent and selective oxadiazole-based agonists of sphingosine-1-phosphate receptor (S1P(1)) 期刊论文
2019, 卷号: 82, 页码: 41-57
作者:  Liu, Tianqi;  Jin, Jing;  Chen, Yonghui;  Xi, Qiumu;  Hu, Jinping
收藏  |  浏览/下载:17/0  |  提交时间:2020/01/03
The involvement of blood cells in the phosphorylation of the selective sphingosine-1-phosphate receptor 1 agonist SYL-927 期刊论文
2019, 卷号: 74, 期号: 2, 页码: 107-110
作者:  Yang, Shy;  Hu, Jin-Ping;  Li, Yan
收藏  |  浏览/下载:3/0  |  提交时间:2020/01/03
CYP2J2 is the major enzyme in human liver microsomes responsible for hydroxylation of SYL-927, a novel and selective sphingosine 1-phosphate receptor 1 (S1P(1)) agonist 期刊论文
2018, 卷号: 39, 期号: 9, 页码: 431-436
作者:  Yang, Shu;  Hu, Jinping;  Li, Yan;  Zhao, Zhigang
收藏  |  浏览/下载:4/0  |  提交时间:2020/01/03
Identification of cytochrome P450 isoforms involved in the metabolism of Syl930, a selective S1PR(1) agonist acting as a potential therapeutic agent for autoimmune encephalitis 期刊论文
2017, 卷号: 32, 期号: 1, 页码: 53-60
作者:  Mi, Jiaqi;  Zhao, Manman;  Yang, Shu;  Jia, Yufei;  Wang, Yan
收藏  |  浏览/下载:5/0  |  提交时间:2020/01/04
NS11821, a partial subtype-selective GABAA agonist, elicits selective effects on the central nervous system in randomized controlled trial with healthy subjects 期刊论文
2016, 卷号: 30, 期号: 3, 页码: 253-62
作者:  Zuiker Rob G J A;  Chen Xia;  Østerberg Ole;  Mirza Naheed R;  Muglia Pierandrea
收藏  |  浏览/下载:5/0  |  提交时间:2020/01/04
IDENTIFICATION OF THE MAJOR METABOLITES OF SYL-927, A SELECTIVE SPHINGOSINE 1-PHOSPHATE RECEPTOR 1 AGONIST IN RATS AND HUMAN LIVER MICROSOMES 会议论文
DRUG METABOLISM REVIEWS, 2015-11-20
作者:  Li, Yan;  Yang, Shu;  Hu, Jinping;  Wang, Xiaojiang;  Xiao, Qiong
收藏  |  浏览/下载:8/0  |  提交时间:2020/01/04
Identification of a novel selective agonist of PPAR gamma with no promotion of adipogenesis and less inhibition of osteoblastogenesis 期刊论文
2015, 卷号: 5, 页码: 9530
作者:  Liu, Chang;  Feng, Tingting;  Zhu, Ningyu;  Liu, Peng;  Han, Xiaowan
收藏  |  浏览/下载:5/0  |  提交时间:2020/01/13
IDENTIFICATION OF THE MAJOR METABOLITES OF SYL-927, A SELECTIVE SPHINGOSINE 1-PHOSPHATE RECEPTOR 1 AGONIST IN RATS AND HUMAN LIVER MICROSOMES 期刊论文
2015, 卷号: 47, 期号: ,SI, 页码: 195-196
作者:  Li, Yan;  Yang, Shu;  Hu, Jinping;  Wang, Xiaojiang;  Xiao, Qiong
收藏  |  浏览/下载:3/0  |  提交时间:2020/01/13
Discovery of SYL933: A 2-aminopropane-1, 3-diol derivative as potent and selective S1P(1) receptor agonist (prodrug) 期刊论文
2014, 卷号: 247
作者:  Tian, Yulin;  Jin, Jing;  Han, Weijuan;  Hu, Jinping;  Zhou, Wanqi
收藏  |  浏览/下载:8/0  |  提交时间:2020/01/13
Discovery of SYL933: A 2-aminopropane-1, 3-diol derivative as potent and selective S1P(1) receptor agonist (prodrug) 会议论文
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014-03-16
作者:  Tian, Yulin;  Jin, Jing;  Han, Weijuan;  Hu, Jinping;  Zhou, Wanqi
收藏  |  浏览/下载:12/0  |  提交时间:2020/01/13


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