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Optimization of the Antiviral Potency and Lipophilicity of Halogenated 2,6-Diarylpyridinamines as a Novel Class of HIV-1 NNRTIS 期刊论文
CHEMMEDCHEM, 2014, 卷号: 9, 期号: 7
作者:  Wu, Zhi-Yuan;  Liu, Na;  Qin, Bingjie;  Huang, Li;  Yu, Fei
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/19
Physicochemical property-driven optimization of diarylaniline compounds as potent HIV-1 non-nucleoside reverse transcriptase inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 16
作者:  Liu, Na;  Qin, Bingjie;  Sun, Lian-Qi;  Yu, Fei;  Lu, Lu
收藏  |  浏览/下载:2/0  |  提交时间:2019/12/19
Small molecule fusion inhibitors: Design, synthesis and biological evaluation of (Z)-3-(5-(3-benzyl-4-oxo-2-thioxothiazolidinylidene)methyl)-N-(3-carboxy-4-hydroxy)phenyl-2,5-dimethylpyrroles and related derivatives targeting HIV-1 gp41 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2013, 卷号: 21, 期号: 23
作者:  He, Xiao-Yang;  Lu, Lu;  Qiu, Jiayin;  Zou, Peng;  Yu, Fei
收藏  |  浏览/下载:6/0  |  提交时间:2019/12/19
L-Selectin and P-Selectin Are Novel Biomarkers of Cervicovaginal Inflammation for Preclinical Mucosal Safety Assessment of Anti-HIV-1 Microbicide 期刊论文
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 2012, 卷号: 56, 期号: 6
作者:  Zhong, Maohua;  He, Benxia;  Yang, Jingyi;  Bao, Rong;  Zhang, Yan
收藏  |  浏览/下载:8/0  |  提交时间:2019/12/19
Synthesis and Anti-HIV Activity of Aryl-2-[(4-cyanophenyl)amino]-4-pyrimidinone hydrazones as Potent Non-nucleoside Reverse Transcriptase Inhibitors 期刊论文
CHEMMEDCHEM, 2011, 卷号: 6, 期号: 12
作者:  Ma, Xiao-Dong;  Yang, Shi-Qiong;  Gu, Shuang-Xi;  He, Qiu-Qin;  Chen, Fen-Er
收藏  |  浏览/下载:2/0  |  提交时间:2019/12/19
Anti-AIDS agents 87. New bio-isosteric dicamphanoyl-dihydropyranochromone (DCP) and dicamphanoyl-khellactone (DCK) analogues with potent anti-HIV activity 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 卷号: 21, 期号: 19
作者:  Liu, Hong-Shan;  Xu, Shi-Qing;  Cheng, Ming;  Chen, Ying;  Xia, Peng
收藏  |  浏览/下载:9/0  |  提交时间:2019/12/19
Design, synthesis and biological evaluation of 3-substituted 2,5-dimethyl-N-(3-(1H-tetrazol-5-yl)phenyl)pyrroles as novel potential HIV-1 gp41 inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2011, 卷号: 19, 期号: 22
作者:  He, Xiao-Yang;  Zou, Peng;  Qiu, Jiayin;  Hou, Ling;  Jiang, Shibo
收藏  |  浏览/下载:2/0  |  提交时间:2019/12/19
Anti-AIDS agents 86. Synthesis and anti-HIV evaluation of 2 ',3 '-seco-3 '-nor DCP and DCK analogues 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2011, 卷号: 46, 期号: 10
作者:  Chen, Ying;  Cheng, Ming;  Liu, Fa-Qiang;  Xia, Peng;  Qian, Keduo
收藏  |  浏览/下载:2/0  |  提交时间:2019/12/19
Anti-AIDS agents 82: Synthesis of seco-(3 ' R,4 ' R)-3 ',4 '-di-O-(S)-camphanoyl-(+)-cis-khellactone (DCK) derivatives as novel anti-HIV agents 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2010, 卷号: 18, 期号: 12
作者:  Tang, Jian;  Qian, Keduo;  Zhang, Bei-Na;  Chen, Ying;  Xia, Peng
收藏  |  浏览/下载:6/0  |  提交时间:2019/12/19
Anti-AIDS agents 84. Synthesis and anti-human immunodeficiency virus (HIV) activity of 2 '-monomethyl-4-methyl- and 1 '-thia-4-methyl-(3 ' R,4 ' R)-3 ',4 '-di-O-(S)-camphanoyl-(+)-cis-khellactone (DCK) analogs 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2010, 卷号: 18, 期号: 20
作者:  Xu, Shi-Qing;  Yan, Xin;  Chen, Ying;  Xia, Peng;  Qian, Keduo
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/19


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