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科研机构
山东大学 [42]
内容类型
期刊论文 [41]
会议论文 [1]
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2019 [2]
2018 [4]
2017 [2]
2016 [3]
2015 [11]
2014 [2]
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专题:山东大学
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An Improved Protocol for the Virtual Screening Discovery of Novel Histone Deacetylase Inhibitors
期刊论文
CHEMICAL & PHARMACEUTICAL BULLETIN, 2019, 卷号: 67, 期号: 10, 页码: 1076-1081
作者:
Song, Qiuhang
;
Liu, Tingting
;
Liu, Yucui
;
Wang, Shuyue
;
Fan, Cong
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2019/12/11
histone deacetylase inhibitor
pharmacophore
docking
molecular dynamic
simulation
ovarian cancer
Effects of histone deacetylase inhibitor Scriptaid and parathyroid hormone on osteocyte functions and metabolism
期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2019, 卷号: 294, 期号: 25, 页码: 9722-9733
作者:
Sun, Ningyuan
;
Uda, Yuhei
;
Azab, Ehab
;
Kochen, Alejandro
;
Santos, Roberto Nunes Campos E.
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2019/12/11
parathyroid hormone
histone deacetylase (HDAC)
osteocyte
glucose
transporter type 4 (GLUT4)
bone
cell metabolism
MEF2
Scriptaid
SOST
Histone deacetylase 6 inhibitor enhances resistance to Mycobacterium tuberculosis infection through innate and adaptive immunity in mice
期刊论文
PATHOGENS AND DISEASE, 2018, 卷号: 76, 期号: 6
作者:
Wang, Xiaolei
;
Tang, Xiaowei
;
Zhou, Zheng
;
Huang, Qing
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/11
pulmonary mycobacterial infection
immune response
IL-10
HDAC6
inflammation
Hyper-acetylation contributes to the sensitivity of chemo-resistant prostate cancer cells to histone deacetylase inhibitor Trichostatin A
期刊论文
JOURNAL OF CELLULAR AND MOLECULAR MEDICINE, 2018, 卷号: 22, 期号: 3, 页码: 1909-1922
作者:
Xu, Qingqing
;
Liu, Xiaofei
;
Zhu, Shiqin
;
Hu, Xuelei
;
Niu, Huanmin
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2019/12/11
chemo-resistant mCRPC
HDAC inhibitors
apoptosis
hyper-acetylation
acetyl-CoA
ER stress
Discovery of meta-sulfamoyl N-hydroxybenzamides as HDAC8 selective inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 页码: 282-291
作者:
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2019/12/11
Histone deacetylase
Anticancer
HDAC8 inhibitor
T-cell leukemia
Neuroblastoma
Histone deacetylase inhibitor SAHA-induced epithelial-mesenchymal transition by upregulating Slug in lung cancer cells
期刊论文
ANTI-CANCER DRUGS, 2018, 卷号: 29, 期号: 1, 页码: 80-88
作者:
Wang, Jun
;
Xu, Mei-qing
;
Jiang, Xian-liang
;
Mei, Xin-yu
;
Liu, Xue-gang
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2019/12/11
epithelial-mesenchymal transitions
metastasis
SAHA
Slug
Design, synthesis, and preliminary bioactivity evaluation of N-benzylpyrimidin-2-amine derivatives as novel histone deacetylase inhibitor
期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2017, 卷号: 90, 期号: 5, 页码: 936-942
作者:
Zhou, Yi
;
Dun, Yanyan
;
Fu, Huansheng
;
Wang, Lei
;
Pan, Xiaole
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/12/16
anticancer
histone deacetylase
inhibitor
tumor
Preclinical and Clinical Studies of Chidamide (CS055/HBI-8000), An Orally Available Subtype-selective HDAC Inhibitor for Cancer Therapy
期刊论文
ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY, 2017, 卷号: 17, 期号: 6, 页码: 802-812
作者:
Gao, Shuai
;
Li, Xiaoyang
;
Zang, Jie
;
Xu, Wenfang
;
Zhang, Yingjie
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/12
Epigenetic
histone deacetylase inhibitors
chidamide
hematologic and
solid cancers
preclinical and clinical trials
Valproic acid induces autophagy by suppressing the Akt/mTOR pathway in human prostate cancer cells
期刊论文
ONCOLOGY LETTERS, 2016, 卷号: 12, 期号: 3, 页码: 1826-1832
作者:
Xia, Qinghua
;
Zheng, Yi
;
Jiang, Wei
;
Huang, Zhongxian
;
Wang, Muwen
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2019/12/16
valproic acid
histone deacetylase inhibitor
prostate cancer
autophagy
Akt/mammalian target of rapamycin pathway
PXD101 analogs with L-phenylglycine-containing branched cap as histone deacetylase inhibitors
期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2016, 卷号: 88, 期号: 4, 页码: 574-584
作者:
Li, Jingyao
;
Li, Xiaoyang
;
Wang, Xue
;
Hou, Jinning
;
Zang, Jie
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/12/16
antiproliferative activity
HDAC inhibitory activity
HDAC isoform
selectivity
HDACs
inhibitor
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