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An Improved Protocol for the Virtual Screening Discovery of Novel Histone Deacetylase Inhibitors 期刊论文
CHEMICAL & PHARMACEUTICAL BULLETIN, 2019, 卷号: 67, 期号: 10, 页码: 1076-1081
作者:  Song, Qiuhang;  Liu, Tingting;  Liu, Yucui;  Wang, Shuyue;  Fan, Cong
收藏  |  浏览/下载:9/0  |  提交时间:2019/12/11
Effects of histone deacetylase inhibitor Scriptaid and parathyroid hormone on osteocyte functions and metabolism 期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2019, 卷号: 294, 期号: 25, 页码: 9722-9733
作者:  Sun, Ningyuan;  Uda, Yuhei;  Azab, Ehab;  Kochen, Alejandro;  Santos, Roberto Nunes Campos E.
收藏  |  浏览/下载:26/0  |  提交时间:2019/12/11
Histone deacetylase 6 inhibitor enhances resistance to Mycobacterium tuberculosis infection through innate and adaptive immunity in mice 期刊论文
PATHOGENS AND DISEASE, 2018, 卷号: 76, 期号: 6
作者:  Wang, Xiaolei;  Tang, Xiaowei;  Zhou, Zheng;  Huang, Qing
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/11
Hyper-acetylation contributes to the sensitivity of chemo-resistant prostate cancer cells to histone deacetylase inhibitor Trichostatin A 期刊论文
JOURNAL OF CELLULAR AND MOLECULAR MEDICINE, 2018, 卷号: 22, 期号: 3, 页码: 1909-1922
作者:  Xu, Qingqing;  Liu, Xiaofei;  Zhu, Shiqin;  Hu, Xuelei;  Niu, Huanmin
收藏  |  浏览/下载:7/0  |  提交时间:2019/12/11
Discovery of meta-sulfamoyl N-hydroxybenzamides as HDAC8 selective inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 页码: 282-291
作者:  
收藏  |  浏览/下载:12/0  |  提交时间:2019/12/11
Histone deacetylase inhibitor SAHA-induced epithelial-mesenchymal transition by upregulating Slug in lung cancer cells 期刊论文
ANTI-CANCER DRUGS, 2018, 卷号: 29, 期号: 1, 页码: 80-88
作者:  Wang, Jun;  Xu, Mei-qing;  Jiang, Xian-liang;  Mei, Xin-yu;  Liu, Xue-gang
收藏  |  浏览/下载:7/0  |  提交时间:2019/12/11
Design, synthesis, and preliminary bioactivity evaluation of N-benzylpyrimidin-2-amine derivatives as novel histone deacetylase inhibitor 期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2017, 卷号: 90, 期号: 5, 页码: 936-942
作者:  Zhou, Yi;  Dun, Yanyan;  Fu, Huansheng;  Wang, Lei;  Pan, Xiaole
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/16
Preclinical and Clinical Studies of Chidamide (CS055/HBI-8000), An Orally Available Subtype-selective HDAC Inhibitor for Cancer Therapy 期刊论文
ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY, 2017, 卷号: 17, 期号: 6, 页码: 802-812
作者:  Gao, Shuai;  Li, Xiaoyang;  Zang, Jie;  Xu, Wenfang;  Zhang, Yingjie
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/12
Valproic acid induces autophagy by suppressing the Akt/mTOR pathway in human prostate cancer cells 期刊论文
ONCOLOGY LETTERS, 2016, 卷号: 12, 期号: 3, 页码: 1826-1832
作者:  Xia, Qinghua;  Zheng, Yi;  Jiang, Wei;  Huang, Zhongxian;  Wang, Muwen
收藏  |  浏览/下载:2/0  |  提交时间:2019/12/16
PXD101 analogs with L-phenylglycine-containing branched cap as histone deacetylase inhibitors 期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2016, 卷号: 88, 期号: 4, 页码: 574-584
作者:  Li, Jingyao;  Li, Xiaoyang;  Wang, Xue;  Hou, Jinning;  Zang, Jie
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/16


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