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A general strategy to the intracellular sensing of glycosidases using AIE-based glycoclusters 期刊论文
CHEMICAL SCIENCE, 2021, 卷号: 13, 期号: 1, 页码: 247-256
作者:  Dong, Lei;  Zhang, Min-Yu;  Han, Hai-Hao;  Zang, Yi;  Chen, Guo-Rong
收藏  |  浏览/下载:31/0  |  提交时间:2022/01/18
Conformational polymorphs of isotretinoin and their impact on physicochemical and biological properties 期刊论文
INTERNATIONAL JOURNAL OF PHARMACEUTICS, 2021, 卷号: 610, 页码: 10
作者:  Cheng, Yinxiang;  Rong, Xiaoyi;  Xia, Mengyuan;  Zhang, Zaiyong;  Wang, Jian-Rong
收藏  |  浏览/下载:73/0  |  提交时间:2022/01/04
Distal mutation V486M disrupts the catalytic activity of DPP4 by affecting the flap of the propeller domain 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 9
作者:  Li, Teng-teng;  Peng, Cheng;  Wang, Ji-qiu;  Xu, Zhi-jian;  Su, Ming-bo
收藏  |  浏览/下载:42/0  |  提交时间:2022/01/18
Theoretical study and application of 2-phenyl-1,3,4-thiadiazole derivatives with optical and inhibitory activity against SHP1 期刊论文
PHYSICAL CHEMISTRY CHEMICAL PHYSICS, 2021, 页码: 14
作者:  Zhang, Chun;  Sun, Yi-Tao;  Gao, Li-Xin;  Feng, Bo;  Yan, Xue
收藏  |  浏览/下载:21/0  |  提交时间:2022/01/18
Nanomedicine Strategies to Circumvent Intratumor Extracellular Matrix Barriers for Cancer Therapy 期刊论文
ADVANCED HEALTHCARE MATERIALS, 2021, 页码: 25
作者:  Xu, Xiaoxuan;  Wu, Yao;  Qian, Xindi;  Wang, Yuqi;  Wang, Jiaoying
收藏  |  浏览/下载:43/0  |  提交时间:2021/12/16
Synthesis and biological evaluation of 2,5-diaryl-1,3,4-oxadiazole derivatives as novel Src homology 2 domain-containing protein tyrosine phosphatase 2 (SHP2) inhibitors 期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 116, 页码: 13
作者:  Meng, Xiang-Dong;  Gao, Li-Xin;  Wang, Zhi-Jia;  Feng, Bo;  Zhang, Chun
收藏  |  浏览/下载:31/0  |  提交时间:2021/12/01
Improving Stability of Vitamin B5 Through Double Salt Formation 期刊论文
CRYSTAL GROWTH & DESIGN, 2021, 卷号: 21, 期号: 9, 页码: 4997-5005
作者:  Liang, Xuan;  Zhang, Qi;  Zhang, Zaiyong;  Ding, Qiaoce;  Mei, Xuefeng
收藏  |  浏览/下载:35/0  |  提交时间:2021/11/04
Discovery of pyrrolo[2,3-d]pyrimidine derivatives as potent Axl inhibitors: Design, synthesis and biological evaluation 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 220, 页码: 18
作者:  Xu, Dandan;  Sun, Deqiao;  Wang, Wei;  Peng, Xia;  Zhan, Zhengsheng
收藏  |  浏览/下载:46/0  |  提交时间:2021/08/17
Design, Synthesis, and Biological Evaluation of Novel Pyrimido[4,5-b]indole Derivatives Against Gram-Negative Multidrug-Resistant Pathogens 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 12, 页码: 8644-8665
作者:  Kong, Qidi;  Pan, Wei;  Xu, Heng;  Xue, Yaru;  Guo, Bin
收藏  |  浏览/下载:38/0  |  提交时间:2021/08/17
Graph neural networks for automated de novo drug design 期刊论文
DRUG DISCOVERY TODAY, 2021, 卷号: 26, 期号: 6, 页码: 1382-1393
作者:  Xiong, Jiacheng;  Xiong, Zhaoping;  Chen, Kaixian;  Jiang, Hualiang;  Zheng, Mingyue
收藏  |  浏览/下载:19/0  |  提交时间:2021/08/17


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