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Distal mutation V486M disrupts the catalytic activity of DPP4 by affecting the flap of the propeller domain 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 9
作者:  Li, Teng-teng;  Peng, Cheng;  Wang, Ji-qiu;  Xu, Zhi-jian;  Su, Ming-bo
收藏  |  浏览/下载:42/0  |  提交时间:2022/01/18
Cryo-EM structures of PI3K alpha reveal conformational changes during inhibition and activation 期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2021, 卷号: 118, 期号: 45, 页码: 9
作者:  Liu, Xiao;  Yang, Su;  Hart, Jonathan R.;  Xu, Yingna;  Zou, Xinyu
收藏  |  浏览/下载:39/0  |  提交时间:2022/01/04
Covalent sortase A inhibitor ML346 prevents Staphylococcus aureus infection of Galleria mellonella 期刊论文
RSC MEDICINAL CHEMISTRY, 2021, 页码: 12
作者:  Guan, Xiang-Na;  Zhang, Tao;  Yang, Teng;  Dong, Ze;  Yang, Song
收藏  |  浏览/下载:20/0  |  提交时间:2021/12/16
Synthesis and bioactivity studies of covalent inhibitors derived from (-)-Chaetominine 期刊论文
JOURNAL OF MOLECULAR STRUCTURE, 2021, 卷号: 1241, 页码: 14
作者:  Zhou, Xian;  Feng, Xuexin;  Wang, Dachi;  Chen, Deheng;  Wu, Gaoxing
收藏  |  浏览/下载:84/0  |  提交时间:2021/08/17
Novel tetrahydrobenzo[b]thiophen-2-yl)urea derivatives as novel alpha-glucosidase inhibitors: Synthesis, kinetics study, molecular docking, and in vivo anti-hyperglycemic evaluation 期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 115, 页码: 17
作者:  Xie, Hong-Xu;  Zhang, Juan;  Li, Yue;  Zhang, Jin-He;  Liu, Shan-Kui
收藏  |  浏览/下载:68/0  |  提交时间:2021/11/04
Structural insights into the activation of human calcium-sensing receptor 期刊论文
ELIFE, 2021, 卷号: 10, 页码: 24
作者:  Chen, Xiaochen;  Wang, Lu;  Cui, Qianqian;  Ding, Zhanyu;  Han, Li
收藏  |  浏览/下载:66/0  |  提交时间:2021/11/04
Metal-drug nanoparticles-mediated osteolytic microenvironment regulation for enhanced radiotherapy of orthotopic osteosarcoma 期刊论文
CHEMICAL ENGINEERING JOURNAL, 2021, 卷号: 417, 页码: 11
作者:  Geng, Huan;  Zhou, Mengxue;  Li, Bin;  Liu, Liang;  Yang, Xu
收藏  |  浏览/下载:23/0  |  提交时间:2021/08/17
Metabolically controlled histone H4K5 acylation/acetylation ratio drives BRD4 genomic distribution 期刊论文
CELL REPORTS, 2021, 卷号: 36, 期号: 4, 页码: 22
作者:  Gao, Mengqing;  Wang, Jin;  Rousseaux, Sophie;  Tan, Minjia;  Pan, Lulu
收藏  |  浏览/下载:65/0  |  提交时间:2021/11/04
D3DistalMutation: a Database to Explore the Effect of Distal Mutations on Enzyme Activity 期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2021, 卷号: 61, 期号: 5, 页码: 2499-2508
作者:  Wang, Xiaoyu;  Zhang, Xinben;  Peng, Cheng;  Shi, Yulong;  Li, Huiyu
收藏  |  浏览/下载:13/0  |  提交时间:2021/08/17
Strigolactone mimic 2-nitrodebranone is highly active in Arabidopsis growth and development 期刊论文
PLANT JOURNAL, 2021, 页码: 10
作者:  Li, Suhua;  Li, Yuwen;  Chen, Linhai;  Zhang, Chi;  Wang, Fei
收藏  |  浏览/下载:43/0  |  提交时间:2021/08/17


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