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Discovery of an Inhibitor for the TREK-1 Channel Targeting an Intermediate Transition State of Channel Gating 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 19, 页码: 10972-10983
作者:  Ma, Yuqin;  Luo, Qichao;  Fu, Jie;  Che, Yanxin;  Guo, Fei
收藏  |  浏览/下载:11/0  |  提交时间:2021/05/24
TREK Channel Family Activator with a Well-Defined Structure-Activation Relationship for Pain and Neurogenic Inflammation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 7, 页码: 3665-3677
作者:  Qiu, Yunguang;  Huang, Lu;  Fu, Jie;  Han, Chenxia;  Fang, Jing
收藏  |  浏览/下载:45/0  |  提交时间:2020/07/01
A Small-Molecule Compound Selectively Activates K2P Channel TASK-3 by Acting at Two Distant Clusters of Residues 期刊论文
MOLECULAR PHARMACOLOGY, 2019, 卷号: 96, 期号: 1, 页码: 26-35
作者:  Tian, Fuyun;  Qiu, Yunguang;  Lan, Xi;  Li, Min;  Yang, Huaiyu
收藏  |  浏览/下载:18/0  |  提交时间:2020/07/01
An allosteric ligand-binding site in the extracellular cap of K2P channels 期刊论文
NATURE COMMUNICATIONS, 2017, 卷号: 8
作者:  Luo, Qichao;  Chen, Liping;  Cheng, Xi;  Ma, Yuqin;  Li, Xiaona
收藏  |  浏览/下载:17/0  |  提交时间:2019/01/08
TREK1 channel blockade induces an antidepressant-like response synergizing with 5-HT1A receptor signaling 期刊论文
EUROPEAN NEUROPSYCHOPHARMACOLOGY, 2015, 卷号: 25, 期号: 12, 页码: 2426-2436
作者:  Ye, Dongqing;  Li, Yang;  Zhang, Xiangrong;  Guo, Fei;  Geng, Leiyu
收藏  |  浏览/下载:20/0  |  提交时间:2019/01/08
TREK1亚型双孔钾离子通道参与抗抑郁治疗的分子机制研究 会议论文
作者:  叶冬青;  李扬;  向荣;  张志珺
收藏  |  浏览/下载:12/0  |  提交时间:2019/01/08
TREK1 potassium channels and depression 期刊论文
Acta Pharmaceutica Sinica, 2012, 卷号: 47, 期号: 11, 页码: 1403-1408
作者:  Ye Dongqing;  Zhang Zhijun;  Li Yang
收藏  |  浏览/下载:9/0  |  提交时间:2019/01/08
trek1钾通道与抑郁症 期刊论文
药学学报, 2012, 卷号: 47, 期号: 11, 页码: 1403
作者:  李扬;  叶冬青;  张志珺
收藏  |  浏览/下载:7/0  |  提交时间:2020/07/01


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