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科研机构
上海药物研究所 [15]
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期刊论文 [15]
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2020 [1]
2019 [1]
2018 [1]
2013 [1]
2012 [3]
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An in vitro Fo''rster resonance energy transfer-based high-throughput screening assay identifies inhibitors of SUMOylation E2 Ubc9
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 10
作者:
Wang, Yu-zhe
;
Liu, Xiao
;
Way, George
;
Madarha, Vipul
;
Zhou, Qing-tong
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2020/07/01
SUMOylation inhibitor
WNN0605-F008
high-throughput screening
Ubc9
PIAS1
Fo''rster resonance energy transfer
surface plasmon resonance
Discovery of betulinaldehyde as a natural ROR gamma t agonist
期刊论文
FITOTERAPIA, 2019, 卷号: 137, 页码: 8
作者:
Yang, Feng
;
Zhang, Ruihan
;
Ni, Dongxuan
;
Luo, Xiaomin
;
Chen, Shijie
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2020/07/01
ROR gamma t
Receptor agonist
Triterpenoids
Alpha screen
Molecular docking
HS218 as an FXR antagonist suppresses gluconeogenesis by inhibiting FXR binding to PGC-1 alpha promoter
期刊论文
METABOLISM-CLINICAL AND EXPERIMENTAL, 2018, 卷号: 85, 页码: 126-138
作者:
Xu, Xin
;
Shi, Xiaofan
;
Chen, Yidi
;
Zhou, Tingting
;
Wang, Jiaying
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2020/07/01
T2DM
Gluconeogenesis
FXR antagonist
PGC-1 alpha
Drug lead compound
Marine natural product des-O-methyllasiodiplodin effectively lowers the blood glucose level in db/db mice via ameliorating inflammation
期刊论文
ACTA PHARMACOLOGICA SINICA, 2013, 卷号: 34, 期号: 10, 页码: 1325-1336
作者:
Zhou, Rong
;
Lin, Zhong-hui
;
Jiang, Cheng-shi
;
Gong, Jing-xu
;
Chen, Li-li
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
des-O-methyllasiodiplodin
diabetes
db/db mice
pro-inflammatory cytokine
ROS
mineralocorticoid receptor
aldosterone
blood glucose
glycosylated hemoglobin (HbA1c)
L655,240, acting as a competitive BACE1 inhibitor, efficiently decreases beta-amyloid peptide production in HEK293-APPswe cells
期刊论文
ACTA PHARMACOLOGICA SINICA, 2012, 卷号: 33, 期号: 12, 页码: 1459-1468
作者:
Lu, Qin
;
Chen, Wu-yan
;
Zhu, Zhi-yuan
;
Chen, Jing
;
Xu, Ye-chun
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
L655,240
Alzheimer's disease
BACE1
beta-amyloid peptide
HEK293-APPswe cells
l655240actingasacompetitivebace1inhibitorefficientlydecreasespamyloidpeptideproductioninhek293appswecells
期刊论文
actapharmacologicasinica, 2012, 卷号: 33, 期号: 12, 页码: 1459
作者:
Lu Qin
;
Chen Wuyan
;
Zhu Zhiyuan
;
Chen Jing
;
Xu Yechun
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2020/07/01
L655
240
Alzheimer's disease
BACE1
-amyloid peptide
HEK293-APPswe cells
L655,240, acting as a competitive BACE1 inhibitor, efficiently decreases p-amyloid peptide production in HEK293-APPswe cells
期刊论文
Acta Pharmacologica Sinica, 2012, 卷号: 33, 期号: 12, 页码: 1459
作者:
Lu Qin
;
Chen Wuyan
;
Zhu Zhiyuan
;
Chen Jing
;
Xu Yechun
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2020/12/24
L655
240
Alzheimer's disease
BACE1
-amyloid peptide
HEK293-APPswe cells
Sulfated polymannuroguluronate inhibits Tat-induced SLK cell adhesion via a novel binding site, a KKR spatial triad
期刊论文
ACTA PHARMACOLOGICA SINICA, 2011, 卷号: 32, 期号: 5, 页码: 647-654
作者:
Wu, Yan-lin
;
Ai, Jing
;
Zhao, Jing-ming
;
Xiong, Bing
;
Xin, Xiao-jie
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2019/01/08
sulfated polymannuroguluronate
transactivating factor of the HIV-1 virus (Tat)
binding site
Kaposi's sarcoma
heparin
mutation
HIV-1
7-Chloroarctinone-b as a new selective PPAR gamma antagonist potently blocks adipocyte differentiation
期刊论文
ACTA PHARMACOLOGICA SINICA, 2009, 卷号: 30, 期号: 9, 页码: 1351-1358
作者:
Li, Yong-tao
;
Li, Li
;
Chen, Jing
;
Hu, Tian-cen
;
Huang, Jin
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2019/01/08
peroxisome proliferator-activated receptor
antagonist
surface plasmon resonance
recruitment of the coactivator
adipocyte differentiation
S9, a Novel Anticancer Agent, Exerts Its Anti-Proliferative Activity by Interfering with Both PI3K-Akt-mTOR Signaling and Microtubule Cytoskeleton
期刊论文
PLOS ONE, 2009, 卷号: 4, 期号: 3
作者:
Zhang, Chao
;
Yang, Na
;
Yang, Chun-hao
;
Ding, Hua-sheng
;
Luo, Cheng
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2019/01/08
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