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TSL-1502, a glucuronide prodrug of a poly (ADP-ribose) polymerase (PARP) inhibitor, exhibits potent anti-tumor activity in preclinical models 期刊论文
AMERICAN JOURNAL OF CANCER RESEARCH, 2021, 卷号: 11, 期号: 4, 页码: 1632-1645
作者:  Wang, Lei;  Zhu, Xi;  Li, Lili;  Li, Lin;  Fu, Li
收藏  |  浏览/下载:75/0  |  提交时间:2021/06/11
A pentapeptide enabled AL3810 liposome-based glioma-targeted therapy with immune opsonic effect attenuated 期刊论文
ACTA PHARMACEUTICA SINICA B, 2021, 卷号: 11, 期号: 1, 页码: 283-299
作者:  Li, Jinyang;  Lu, Jiasheng;  Guo, Haiyan;  Zhou, Jianfen;  Wang, Songli
收藏  |  浏览/下载:28/0  |  提交时间:2021/05/24
Bufalin exerts antitumor effects in neuroblastoma via the induction of reactive oxygen species-mediated apoptosis by targeting the electron transport chain 期刊论文
INTERNATIONAL JOURNAL OF MOLECULAR MEDICINE, 2020, 卷号: 46, 期号: 6, 页码: 2137-2149
作者:  Pan, Lijia;  Nie, Litong;  Yao, Sheng;  Bi, Aiwei;  Ye, Yang
收藏  |  浏览/下载:26/0  |  提交时间:2020/12/24
SAF-189s, a potent new-generation ROS1 inhibitor, is active against crizotinib-resistant ROS1 mutant-driven tumors 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 7
作者:  Xia, Zong-jun;  Ji, Yin-chun;  Sun, De-qiao;  Peng, Xia;  Gao, Ying-lei
收藏  |  浏览/下载:75/0  |  提交时间:2020/12/21
Cancer Cell Membrane-Camouflaged Nanorods with Endoplasmic Reticulum Targeting for Improved Antitumor Therapy 期刊论文
ACS APPLIED MATERIALS & INTERFACES, 2019, 卷号: 11, 期号: 50, 页码: 46614-46625
作者:  Zhang, Wei;  Yu, Miaorong;  Xi, Ziyue;  Nie, Di;  Dai, Zhuo
收藏  |  浏览/下载:38/0  |  提交时间:2020/07/01
Activation and function of receptor tyrosine kinases in human clear cell renal cell carcinomas 期刊论文
BMC CANCER, 2019, 卷号: 19, 期号: 1, 页码: 13
作者:  Zhang, Qing;  Liu, Jian-He;  Liu, Jing-Li;  Qi, Chun-Ting;  Yan, Lei
收藏  |  浏览/下载:60/0  |  提交时间:2020/07/01
1-Phenyl-dihydrobenzoindazoles as novel colchicine site inhibitors: Structural basis and antitumor efficacy 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 177, 页码: 448-456
作者:  Jiang, Junhang;  Zhang, Hao;  Wang, Chongqing;  Zhang, Qingsen;  Fang, Shaoyu
收藏  |  浏览/下载:16/0  |  提交时间:2020/07/01
Preclinical evaluation of 3D185, a novel potent inhibitor of FGFR1/2/3 and CSF-1R, in FGFR-dependent and macrophage-dominant cancer models 期刊论文
JOURNAL OF EXPERIMENTAL & CLINICAL CANCER RESEARCH, 2019, 卷号: 38, 期号: 1, 页码: 16
作者:  Peng, Xia;  Hou, Pengcong;  Chen, Yi;  Dai, Yang;  Ji, Yinchun
收藏  |  浏览/下载:6/0  |  提交时间:2020/07/01
Inhibition of G9a by a small molecule inhibitor, UNC0642, induces apoptosis of human bladder cancer cells 期刊论文
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 8, 页码: 1076-1084
作者:  Cao, Yue-peng;  Sun, Jing-ya;  Li, Mei-qian;  Dong, Yu;  Zhang, Yuan-heng
收藏  |  浏览/下载:17/0  |  提交时间:2020/07/01
Inhibition of the BET family reduces its new target gene IDO1 expression and the production of L-kynurenine 期刊论文
CELL DEATH & DISEASE, 2019, 卷号: 10, 页码: 13
作者:  Tian, Chang-Qing;  Chen, Lin;  Chen, Hua-Dong;  Huan, Xia-Juan;  Hu, Jian-Ping
收藏  |  浏览/下载:19/0  |  提交时间:2020/07/01


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