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Phase I dose-escalation and expansion study of PARP inhibitor, fluzoparib (SHR3162), in patients with advanced solid tumors 期刊论文
CHINESE JOURNAL OF CANCER RESEARCH, 2020, 卷号: 32, 期号: 3, 页码: 370-+
作者:  Li, Huiping;  Liu, Rongrui;  Shao, Bin;  Ran, Ran;  Song, Guohong
收藏  |  浏览/下载:22/0  |  提交时间:2020/12/24
Discovery of potent 2,4-difluoro-linker poly(ADP-ribose) polymerase 1 inhibitors with enhanced water solubility and in vivo anticancer efficacy 期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 11, 页码: 1521-1532
作者:  Chen, Wen-hua;  Song, Shan-shan;  Qi, Ming-hui;  Huan, Xia-juan;  Wang, Ying-qing
收藏  |  浏览/下载:26/0  |  提交时间:2019/01/08
discoveryofpotent24difluorolinkerpolyadpribosepolymerase1inhibitorswithenhancedwatersolubilityandinvivoanticancerefficacy 期刊论文
actapharmacologicasinica, 2017, 卷号: 38, 期号: 11, 页码: 1521
作者:  Chen Wenhua;  Song Shanshan;  Ql Minghui;  Huan Xiajuan;  Wang Yingqing
收藏  |  浏览/下载:5/0  |  提交时间:2020/07/01
Effects of alisol B 23-acetate on ovarian cancer cells: G1 phase cell cycle arrest, apoptosis, migration and invasion inhibition 期刊论文
PHYTOMEDICINE, 2016, 卷号: 23, 期号: 8, 页码: 800-809
作者:  Zhang, Le-Le;  Xu, Yu-Lian;  Tang, Zheng-Hai;  Xu, Xiao-Huang;  Chen, Xin
收藏  |  浏览/下载:19/0  |  提交时间:2019/01/08
Synthesis of isoquinolinone-based tricycles as novel poly(ADP-ribose) polymerase-1 (PARP-1) inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 12, 页码: 2669-2673
作者:  Chen, Jianyang;  Peng, Haixia;  He, Jinxue;  Huan, Xiajuan;  Miao, Zehong
收藏  |  浏览/下载:19/0  |  提交时间:2019/01/08
Curcusone D, a novel ubiquitin-proteasome pathway inhibitor via ROS-induced DUB inhibition, is synergistic with bortezomib against multiple myeloma cell growth 期刊论文
BIOCHIMICA ET BIOPHYSICA ACTA-GENERAL SUBJECTS, 2014, 卷号: 1840, 期号: 6, 页码: 2004-2013
作者:  Cao, Mei-Na;  Zhou, Yu-Bo;  Gao, An-Hui;  Cao, Jia-Yi;  Gao, Li-Xin
收藏  |  浏览/下载:33/0  |  提交时间:2019/01/08
Lewis Acid Catalyzed Cyclization of Glycals/2-Deoxy-D-ribose with Arylamines: Additional Findings on Product Structure and Reaction Diastereoselectivity 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2011, 卷号: 76, 期号: 21, 页码: 8833-8839
作者:  Du, Chengtang;  Li, Fulong;  Zhang, Xuefeng;  Hu, Wenxiang;  Yao, Qizheng
收藏  |  浏览/下载:13/0  |  提交时间:2019/01/08
Investigation of the Catalytic Mechanism of Sir2 Enzyme with QM/MM Approach: SN1 vs SN2? 期刊论文
JOURNAL OF PHYSICAL CHEMISTRY B, 2010, 卷号: 114, 期号: 36, 页码: 11927-11933
作者:  Liang, Zhongjie;  Shi, Ting;  Ouyang, Sisheng;  Li, Honglin;  Yu, Kunqian
收藏  |  浏览/下载:24/0  |  提交时间:2019/01/08
AMP-activated Protein Kinase Is Involved in Neural Stem Cell Growth Suppression and Cell Cycle Arrest by 5-Aminoimidazole-4-carboxamide-1-beta-D-ribofuranoside and Glucose Deprivation by Down-regulating Phospho-retinoblastoma Protein and Cyclin D 期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2009, 卷号: 284, 期号: 10, 页码: 6175-6184
作者:  Zang, Yi;  Yu, Li-Fang;  Nan, Fa-Jun;  Feng, Lin-Yin;  Li, Jia
收藏  |  浏览/下载:9/0  |  提交时间:2019/01/08


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