×
验证码:
换一张
忘记密码?
记住我
CORC
首页
科研机构
检索
知识图谱
申请加入
托管服务
登录
注册
在结果中检索
科研机构
上海药物研究所 [10]
内容类型
期刊论文 [9]
学位论文 [1]
发表日期
2020 [1]
2017 [2]
2016 [1]
2014 [2]
2011 [1]
2010 [1]
更多...
×
知识图谱
CORC
开始提交
已提交作品
待认领作品
已认领作品
未提交全文
收藏管理
QQ客服
官方微博
反馈留言
浏览/检索结果:
共10条,第1-10条
帮助
限定条件
专题:上海药物研究所
第一署名单位
第一作者单位
通讯作者单位
已选(
0
)
清除
条数/页:
5
10
15
20
25
30
35
40
45
50
55
60
65
70
75
80
85
90
95
100
排序方式:
请选择
作者升序
作者降序
题名升序
题名降序
发表日期升序
发表日期降序
提交时间升序
提交时间降序
Phase I dose-escalation and expansion study of PARP inhibitor, fluzoparib (SHR3162), in patients with advanced solid tumors
期刊论文
CHINESE JOURNAL OF CANCER RESEARCH, 2020, 卷号: 32, 期号: 3, 页码: 370-+
作者:
Li, Huiping
;
Liu, Rongrui
;
Shao, Bin
;
Ran, Ran
;
Song, Guohong
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2020/12/24
Phase I
PARP inhibitor (fluzoparib)
solid tumor
pharmacokinetics
safety
antitumor activity
Discovery of potent 2,4-difluoro-linker poly(ADP-ribose) polymerase 1 inhibitors with enhanced water solubility and in vivo anticancer efficacy
期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 11, 页码: 1521-1532
作者:
Chen, Wen-hua
;
Song, Shan-shan
;
Qi, Ming-hui
;
Huan, Xia-juan
;
Wang, Ying-qing
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2019/01/08
PARP-1 inhibitor
olaparib
breast cancer
BRCA-deficient tumors
discoveryofpotent24difluorolinkerpolyadpribosepolymerase1inhibitorswithenhancedwatersolubilityandinvivoanticancerefficacy
期刊论文
actapharmacologicasinica, 2017, 卷号: 38, 期号: 11, 页码: 1521
作者:
Chen Wenhua
;
Song Shanshan
;
Ql Minghui
;
Huan Xiajuan
;
Wang Yingqing
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2020/07/01
PARP INHIBITORS
MEDICINAL CHEMISTRY
DRUG DISCOVERY
CANCER
THERAPY
DESIGN
FLUORINE
SUCCESS
PREDICT
METRICS
PARP-1 inhibitor
olaparib
breast cancer
BRCA-deficient tumors
Effects of alisol B 23-acetate on ovarian cancer cells: G1 phase cell cycle arrest, apoptosis, migration and invasion inhibition
期刊论文
PHYTOMEDICINE, 2016, 卷号: 23, 期号: 8, 页码: 800-809
作者:
Zhang, Le-Le
;
Xu, Yu-Lian
;
Tang, Zheng-Hai
;
Xu, Xiao-Huang
;
Chen, Xin
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2019/01/08
Ovarian cancer
Alisol B 23-acetate
Cell cycle arrest
Apoptosis
Migration
Invasion
Synthesis of isoquinolinone-based tricycles as novel poly(ADP-ribose) polymerase-1 (PARP-1) inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 12, 页码: 2669-2673
作者:
Chen, Jianyang
;
Peng, Haixia
;
He, Jinxue
;
Huan, Xiajuan
;
Miao, Zehong
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2019/01/08
Isoquinolinone-based tricycles
PARP-1 inhibitors
Antitumor
Curcusone D, a novel ubiquitin-proteasome pathway inhibitor via ROS-induced DUB inhibition, is synergistic with bortezomib against multiple myeloma cell growth
期刊论文
BIOCHIMICA ET BIOPHYSICA ACTA-GENERAL SUBJECTS, 2014, 卷号: 1840, 期号: 6, 页码: 2004-2013
作者:
Cao, Mei-Na
;
Zhou, Yu-Bo
;
Gao, An-Hui
;
Cao, Jia-Yi
;
Gao, Li-Xin
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2019/01/08
Ubiquitin-proteasome pathway
Deubiquitinase
ROS
Curcusone D
Bortezomib
Multiple myeloma
Lewis Acid Catalyzed Cyclization of Glycals/2-Deoxy-D-ribose with Arylamines: Additional Findings on Product Structure and Reaction Diastereoselectivity
期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2011, 卷号: 76, 期号: 21, 页码: 8833-8839
作者:
Du, Chengtang
;
Li, Fulong
;
Zhang, Xuefeng
;
Hu, Wenxiang
;
Yao, Qizheng
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/01/08
Investigation of the Catalytic Mechanism of Sir2 Enzyme with QM/MM Approach: SN1 vs SN2?
期刊论文
JOURNAL OF PHYSICAL CHEMISTRY B, 2010, 卷号: 114, 期号: 36, 页码: 11927-11933
作者:
Liang, Zhongjie
;
Shi, Ting
;
Ouyang, Sisheng
;
Li, Honglin
;
Yu, Kunqian
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2019/01/08
AMP-activated Protein Kinase Is Involved in Neural Stem Cell Growth Suppression and Cell Cycle Arrest by 5-Aminoimidazole-4-carboxamide-1-beta-D-ribofuranoside and Glucose Deprivation by Down-regulating Phospho-retinoblastoma Protein and Cyclin D
期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2009, 卷号: 284, 期号: 10, 页码: 6175-6184
作者:
Zang, Yi
;
Yu, Li-Fang
;
Nan, Fa-Jun
;
Feng, Lin-Yin
;
Li, Jia
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2019/01/08
©版权所有 ©2017 CSpace - Powered by
CSpace