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1-Phenyl-dihydrobenzoindazoles as novel colchicine site inhibitors: Structural basis and antitumor efficacy 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 177, 页码: 448-456
作者:  Jiang, Junhang;  Zhang, Hao;  Wang, Chongqing;  Zhang, Qingsen;  Fang, Shaoyu
收藏  |  浏览/下载:17/0  |  提交时间:2020/07/01
The Structure of MT189-Tubulin Complex Provides Insights into Drug Design 期刊论文
LETTERS IN DRUG DESIGN & DISCOVERY, 2019, 卷号: 16, 期号: 9, 页码: 1069-1073
作者:  Li, Zhongping;  Ma, Lingling;  Wu, Chengyong;  Meng, Tao;  Ma, Lanping
收藏  |  浏览/下载:8/0  |  提交时间:2020/07/01
Potent Antitumor Activities and Structure Basis of the Chiral beta-Lactam Bridged Analogue of Combretastatin A-4 Binding to Tubulin 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 22, 页码: 10329-10334
作者:  Zhou, Pengfei;  Liu, Yan;  Zhou, Lu;  Zhu, Kongkai;  Feng, Kechang
收藏  |  浏览/下载:21/0  |  提交时间:2019/01/08
Discovery of novel 2-phenyl-imidazo[1,2-a]pyridine analogues targeting tubulin polymerization as antiproliferative agents 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 112, 页码: 367-372
作者:  An, Weiteng;  Wang, Wei;  Yu, Ting;  Zhang, Yongliang;  Miao, Zehong
收藏  |  浏览/下载:13/0  |  提交时间:2019/01/08
Dual targeting of microtubule and topoisomerase II by alpha-carboline derivative YCH337 for tumor proliferation and growth inhibition 期刊论文
ONCOTARGET, 2015, 卷号: 6, 期号: 11, 页码: 8960-8973
作者:  Yi, Jun-Mei;  Zhang, Xiao-Fei;  Huan, Xia-Juan;  Song, Shan-Shan;  Wang, Wei
收藏  |  浏览/下载:17/0  |  提交时间:2019/01/08
MCL-1 Degradation Mediated by JNK Activation via MEKK1/TAK1-MKK4 Contributes to Anticancer Activity of New Tubulin Inhibitor MT189 期刊论文
MOLECULAR CANCER THERAPEUTICS, 2014, 卷号: 13, 期号: 6, 页码: 1480-1491
作者:  Wang, Wei;  Wang, Ying-Qing;  Meng, Tao;  Yi, Jun-Mei;  Huan, Xia-Juan
收藏  |  浏览/下载:22/0  |  提交时间:2019/01/08
Synthesis and biological evaluation of 6H-pyrido[2 ',1 ':2,3] imidazo[4,5-c] isoquinolin-5(6H)-ones as antimitotic agents and inhibitors of tubulin polymerization 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2014, 卷号: 22, 期号: 2, 页码: 848-855
作者:  Meng, Tao;  Wang, Wei;  Zhang, Zhixiang;  Ma, Lanping;  Zhang, Yongliang
收藏  |  浏览/下载:15/0  |  提交时间:2019/01/08
YHHU0895, a novel synthetic small-molecule microtubule-destabilizing agent, effectively overcomes P-glycoprotein-mediated tumor multidrug resistance 期刊论文
CANCER LETTERS, 2012, 卷号: 314, 期号: 1, 页码: 54-62
作者:  Zhao, Hongbing;  Quan, Haitian;  Xie, Chengying;  Xu, Yongping;  Xie, Fuchun
收藏  |  浏览/下载:15/0  |  提交时间:2019/01/08
MT119, a new planar-structured compound, targets the colchicine site of tubulin arresting mitosis and inhibiting tumor cell proliferation 期刊论文
INTERNATIONAL JOURNAL OF CANCER, 2011, 卷号: 129, 期号: 1, 页码: 214-224
作者:  Zhang, Zhixiang;  Meng, Tao;  Yang, Na;  Wang, Wei;  Xiong, Bing
收藏  |  浏览/下载:11/0  |  提交时间:2019/01/08
Synthesis and Biological Evaluation of 2,4,5-Substituted Pyrimidines as a New Class of Tubulin Polymerization Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2011, 卷号: 54, 期号: 9, 页码: 3200-3205
作者:  Xie, Fuchun;  Zhao, Hongbing;  Li, Dewen;  Chen, Hong;  Quan, Haitian
收藏  |  浏览/下载:15/0  |  提交时间:2019/01/08


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