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科研机构
上海药物研究所 [40]
内容类型
期刊论文 [40]
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2021 [2]
2020 [3]
2019 [3]
2018 [1]
2017 [2]
2016 [2]
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Antimicrobial and Immunomodulating Activities of Two Endemic Nepeta Species and Their Major Iridoids Isolated from Natural Sources
期刊论文
PHARMACEUTICALS, 2021, 卷号: 14, 期号: 5, 页码: 22
作者:
Anicic, Neda
;
Gasic, Uros
;
Lu, Feng
;
Ciric, Ana
;
Ivanov, Marija
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2021/08/17
Nepeta
nepetalactone
1,5,9-epideoxyloganic acid
antimicrobial activity
antibiofilm
immunomodulatory effects
In Vivo Efficacy and Metabolism of the Antimalarial Cycleanine and Improved In Vitro Antiplasmodial Activity of Semisynthetic Analogues
期刊论文
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 2021, 卷号: 65, 期号: 2, 页码: 11
作者:
Uche, Fidelia Ijeoma
;
Guo, Xiaozhen
;
Okokon, Jude
;
Ullah, Imran
;
Horrocks, Paul
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  |  
浏览/下载:26/0
  |  
提交时间:2021/05/24
malaria
Plasmodium falciparum
Plasmodium berghei
bisbenzylisoquinoline alkaloids
cycleanine
metabolism
in vivo activity
antimalarial agents
drug metabolism
Capsaicin derivatives with nitrothiophene substituents: Design, synthesis and antibacterial activity against multidrug-resistant S. aureus
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 198, 页码: 11
作者:
Wang, Zhi-Cheng
;
Wei, Bingyan
;
Pei, Fang-Ning
;
Yang, Teng
;
Tang, Jie
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2020/12/24
Capsaicin
Nitrothiophene
Multidrug-resistant S. aureus
Antibacterial agent
Quantitative analysis of fourteen bufadienolides in Venenum Bufonis crude drug and its Chinese patent medicines by ultra-high performance liquid chromatography coupled with tandem mass spectrometry
期刊论文
JOURNAL OF ETHNOPHARMACOLOGY, 2020, 卷号: 251, 页码: 8
作者:
Wei, Wen-long
;
An, Ya-ling
;
Zhang, Yan-zhi
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  |  
浏览/下载:26/0
  |  
提交时间:2020/07/01
Venenum Bufonis
Multi-component quantification
Quality evaluation
UHPLC-QqQ-MS/MS
Synthesis and Structure-Activity Relationship of Palmatine Derivatives as a Novel Class of Antibacterial Agents against Helicobacter pylori
期刊论文
MOLECULES, 2020, 卷号: 25, 期号: 6, 页码: 12
作者:
Fan, Tianyun
;
Guo, Xixi
;
Zeng, Qingxuan
;
Wei, Wei
;
You, Xuefu
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2020/07/01
Helicobacter pylori
palmatine
synthesis
structure-activity relationship
urease
Callistemonols A and B, Potent Antimicrobial Acylphloroglucinol Derivatives with Unusual Carbon Skeletons from Callistemon viminalis
期刊论文
JOURNAL OF NATURAL PRODUCTS, 2019, 卷号: 82, 期号: 7, 页码: 1917-1922
作者:
Wu, Jie-Wei
;
Li, Bai-Lin
;
Tang, Chunping
;
Ke, Chang-Qang
;
Zhu, Nan-Lin
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  |  
浏览/下载:18/0
  |  
提交时间:2020/07/01
Synthesis and Cdc25B/PTP1B Inhibitory Activity Evaluation of Novel Acylhydrazone Derivatives Containing Carbazole Moity
期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2019, 卷号: 39, 期号: 2, 页码: 491-499
作者:
Li Yingjun
;
Wang Siyuan
;
Jin Kun
;
Gao Lixin
;
Sheng Li
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2020/07/01
acylhydrazone
carbazole
synthesis
Cdc25B and PTP1B inhibitor
molecular docking
synthesisandcdc25bptp1binhibitoryactivityevaluationofnovelacylhydrazonederivativescontainingcarbazolemoity
期刊论文
chinesejournaloforganicchemistry, 2019, 卷号: 39, 期号: 2, 页码: 491
作者:
Li YJ(李英俊)
;
Wang SY(王思远)
;
Jin K(靳焜)
;
Gao LX(高立信)
;
Sheng L(盛丽)
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2020/07/01
BIOLOGICAL EVALUATION
ANTITUBERCULOSIS ACTIVITY
PHOSPHATASE INHIBITORS
ANTIMICROBIAL ACTIVITY
DOCKING
OPTIMIZATION
MECHANISM
ANALOGS
DESIGN
AGENTS
acylhydrazone
carbazole
synthesis
Cdc25B and PTP1B inhibitor
molecular docking
Protein Acylation Affects the Artificial Biosynthetic Pathway for Pinosylvin Production in Engineered E. coli
期刊论文
ACS CHEMICAL BIOLOGY, 2018, 卷号: 13, 期号: 5, 页码: 1200-1208
作者:
Xu, Jun-Yu
;
Xu, Ya
;
Chu, Xiaohe
;
Tan, Minjia
;
Ye, Bang-Ce
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/01/08
Prenylated flavonoids from the stems and roots of Tripterygiwn wilfordii
期刊论文
FITOTERAPIA, 2017, 卷号: 119, 页码: 64-68
作者:
Chen, Yang
;
Zhao, Jianping
;
Qiu, Yixing
;
Yuan, Hanwen
;
Khan, Shabana I.
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2019/01/08
Tripterygium wilfordii
Celastraceae
Flavanone
Antimicrobial
Antimalarial
NMR
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