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Identification of Betulinic Acid Derivatives as Potent TGR5 Agonists with Antidiabetic Effects via Humanized TGR5(H88Y) Mutant Mice 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 16, 页码: 12181-12199
作者:  Yun, Ying;  Zhang, Chenlu;  Guo, Shimeng;  Liang, Xiaoying;  Lan, Yuan
收藏  |  浏览/下载:43/0  |  提交时间:2021/11/04
A novel GPR120-selective agonist promotes insulin secretion and improves chronic inflammation 期刊论文
LIFE SCIENCES, 2021, 卷号: 269, 页码: 8
作者:  Yang, Liu;  Lei, Xian-Tao;  Huang, Qi;  Wang, Ting;  Sun, Hong-Bin
收藏  |  浏览/下载:24/0  |  提交时间:2021/05/24
Secretion of glucagon-like peptide-1 induced by Cynanchum pregnane derivatives: Preliminary hypotheses regarding key structural elements 期刊论文
PHYTOCHEMISTRY LETTERS, 2021, 卷号: 41, 页码: 88-91
作者:  Huguet, Clement;  Real, Eleonore;  Zhao, Wei-Min;  Urbain, Aurelie
收藏  |  浏览/下载:12/0  |  提交时间:2021/11/04
Determination of the antidiabetic chemical basis of Phellodendri Chinensis Cortex by integrating hepatic disposition in vivo and hepatic gluconeogenese inhibition in vitro 期刊论文
JOURNAL OF ETHNOPHARMACOLOGY, 2020, 卷号: 263, 页码: 10
作者:  Tian, Xiaoting;  Xu, Zhou;  Hu, Pei;  Yu, Yanyan;  Li, Zhixiong
收藏  |  浏览/下载:74/0  |  提交时间:2020/12/21
Cinnamtannin D1 Protects Pancreatic beta-Cells from Glucolipotoxicity-Induced Apoptosis by Enhancement of Autophagy In Vitro and In Vivo 期刊论文
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2020, 卷号: 68, 期号: 45, 页码: 12617-12630
作者:  Wang, Xin-Yi;  Zhu, Bo-Rong;  Jia, Qi;  Li, Yi-Ming;  Wang, Ting
收藏  |  浏览/下载:24/0  |  提交时间:2021/05/24
DGAT1 inhibitors protect pancreatic beta-cells from palmitic acid-induced apoptosis 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 8
作者:  Huang, Jun-shang;  Guo, Bin-bin;  Wang, Gai-hong;  Zeng, Li-min;  Hu, You-hong
收藏  |  浏览/下载:57/0  |  提交时间:2020/12/24
Synthesis and biological evaluation of novel potent FFA1 agonists containing 2,3-dihydrobenzo[b][1,4]dioxine 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 6, 页码: 848-852
作者:  Kong, Deyu;  Guo, Shimeng;  Yang, Yushe;  Guo, Bin;  Xie, Xin
收藏  |  浏览/下载:29/0  |  提交时间:2020/07/01
Discovery of a Natural-Product-Derived Preclinical Candidate for Once-Weekly Treatment of Type 2 Diabetes 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 5, 页码: 2348-2361
作者:  Li, Shiliang;  Qin, Chun;  Cui, Shichao;  Xu, Hongling;  Wu, Fangshu
收藏  |  浏览/下载:22/0  |  提交时间:2020/07/01
Design, synthesis and structure activity relationship studies of GPR40 agonists containing amide linker 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 152, 页码: 175-194
作者:  Chen, Tingting;  Ning, Mengmeng;  Ye, Yangliang;  Wang, Kai;  Leng, Ying
收藏  |  浏览/下载:32/0  |  提交时间:2019/01/08
5,4 '-Dihydroxy-7,8-dimethoxyflavanone and Aliarin from Dodonaea viscosa Are Activators of PPAR gamma 期刊论文
PLANTA MEDICA, 2018, 卷号: 84, 期号: 8, 页码: 500-506
作者:  Zhu, Jing-jie;  Ji, Jun;  Hou, Ai-Jun;  Wang, He-Yao
收藏  |  浏览/下载:30/0  |  提交时间:2019/01/08


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