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科研机构
上海药物研究所 [76]
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期刊论文 [75]
学位论文 [1]
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2018 [8]
2017 [4]
2016 [8]
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Improved Practical Synthesis of DY-038, an Oral Available Antiplatelet Agent
期刊论文
CHEMISTRYSELECT, 2021, 卷号: 6, 期号: 13, 页码: 3183-3186
作者:
Cao, Yangzhi
;
Kong, Deyu
;
Sun, Lulu
;
Meng, Xin
;
Zhang, Yinyong
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2021/08/17
antiplatelet agent
cyclization
DY-038
process development
sulfonamides
Optimization of P2Y(12) Antagonist Ethyl 6-(4-((Benzylsulfonyl)carbarnoyl)piperidin-1-yl)-5-cyano-2-methylnicotinate (AZD1283) Led to the Discovery of an Oral Antiplatelet Agent with Improved Druglike Properties
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 6, 页码: 3088-3106
作者:
Kong, Deyu
;
Xue, Tao
;
Guo, Bin
;
Cheng, Jianjun
;
Liu, Shunyin
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  |  
浏览/下载:15/0
  |  
提交时间:2020/07/01
Inhibiting mechanism of small molecule toward the p53-MDM2 interaction: A molecular dynamic exploration
期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2018, 卷号: 92, 期号: 4, 页码: 1763-1777
作者:
Chen, Jianzhong
;
Wang, Jinan
;
Pang, Laixue
;
Zhu, Weiliang
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  |  
浏览/下载:40/0
  |  
提交时间:2019/01/08
hydrophobic contact scanning
MM-GBSA
p53-MDM2 interaction
principal component analysis
solvated interaction energy
Structural characterization of a galactan from Ophiopogon japonicus and anti-pancreatic cancer activity of its acetylated derivative
期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2018, 卷号: 113, 页码: 907-915
作者:
Gu, Dan
;
Huang, Lulin
;
Chen, Xia
;
Wu, Qianhu
;
Ding, Kan
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  |  
浏览/下载:74/0
  |  
提交时间:2019/01/08
Ophiopogon japonicus
Polysaccharide
Acetylated derivative
Apoptosis
Anti-pancreatic cancer
Design, synthesis and biological evaluation of a series of novel 2-benzamide-4-(6-oxy-N-methyl-l-naphthamide)-pyridine derivatives as potent fibroblast growth factor receptor (FGFR) inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 154, 页码: 9-28
作者:
Wei, Manman
;
Peng, Xia
;
Xing, Li
;
Dai, Yang
;
Huang, Ruimin
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  |  
浏览/下载:63/0
  |  
提交时间:2019/01/08
FGFR
VEGFR
Synergistic effect
Tumor growth inhibition
Lucitanib
Design, synthesis, and molecular docking study of 3H-imidazole[4,5-c]pyridine derivatives as CDK2 inhibitors
期刊论文
ARCHIV DER PHARMAZIE, 2018, 卷号: 351, 期号: 6
作者:
Wu, Yi-Zhe
;
Ying, Hua-Zhou
;
Xu, Lei
;
Cheng, Gang
;
Chen, Jing
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  |  
浏览/下载:33/0
  |  
提交时间:2019/01/08
cancer
CDK2 inhibitor
imidazo[4
5-c]pyridine
targeted therapy
Discovery and structure-activity relationships study of thieno[2,3-b] pyridine analogues as hepatic gluconeogenesis inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 152, 页码: 307-317
作者:
Ma, Fei
;
Liu, Jian
;
Zhou, Tingting
;
Lei, Min
;
Chen, Jing
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  |  
浏览/下载:79/0
  |  
提交时间:2019/01/08
Thienol2,3-b]pyridine derivatives
Structure-activity relationships (SARs)
Hepatic gluconeogenesis
Type 2 diabetes mellitus (T2DM)
One-step calcination preparation of worm-like ZnO@BiOI heterojunction with enhanced visible light response for mild photooxidation reaction
期刊论文
MATERIALS LETTERS, 2018, 卷号: 217, 页码: 296-299
作者:
Tong, Zhifang
;
He, Lingling
;
Ren, Chunguang
;
Wang, Zhonghua
;
Jiang, Zonglin
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2019/01/08
One-step method
ZnO@BiOI
Nanocomposites
Visible light
Oxidation, 1,4-DHP derivatives
Facile Synthesis of New Functionalized Triazacyclopenta[cd]indenones Through a Multicomponent Reaction Followed by an Intramolecular Aminolysis
期刊论文
JOURNAL OF HETEROCYCLIC CHEMISTRY, 2018, 卷号: 55, 期号: 4, 页码: 814-820
作者:
Shen, Guo-Bing
;
Yu, Ting
;
Zhang, Yong-Liang
;
Ma, Lan-Ping
;
Chen, Lin
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  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
Rapid Syntheses of Heteroaryl-Substituted Imidazo[1,5-a]indole and Pyrrolo[1,2-c]imidazole via Aerobic C2-H Functionalizations
期刊论文
ORGANIC LETTERS, 2018, 卷号: 20, 期号: 1, 页码: 284-287
作者:
Kong, Wei-Jun
;
Chen, Xingrong
;
Wang, Mingming
;
Dai, Hui-Xiong
;
Yu, Jin-Quan
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  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
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