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科研机构
北京大学 [10]
内容类型
期刊论文 [9]
其他 [1]
发表日期
2017 [2]
2016 [1]
2015 [2]
2014 [3]
2012 [1]
2006 [1]
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专题:北京大学
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Statistical Analysis and Prediction of Covalent Ligand Targeted Cysteine Residues
期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2017
Zhang, Weilin
;
Pei, Jianfeng
;
Lai, Luhua
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2017/12/03
AMINO-ACID ALPHABET
PROTEIN DATA-BANK
ALLOSTERIC DRUGS
RATIONAL DESIGN
BINDING-SITES
DOCKING
DISCOVERY
IDENTIFICATION
INHIBITORS
INFORMATION
Rational Design of Selective Allosteric Inhibitors of PHGDH and Serine Synthesis with Anti-tumor Activity
期刊论文
CELL CHEMICAL BIOLOGY, 2017
Wang, Qian
;
Liberti, Maria V.
;
Liu, Pei
;
Deng, Xiaobing
;
Liu, Ying
;
Locasale, Jason W.
;
Lai, Luhua
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2017/12/03
PHOSPHOGLYCERATE DEHYDROGENASE
CANCER METABOLISM
SYNTHESIS PATHWAY
ACCURATE DOCKING
BINDING-SITES
DRUG DESIGN
BIOSYNTHESIS
DISCOVERY
CELLS
COMBINATION
Discovery of Novel 15-Lipoxygenase Activators To Shift the Human Arachidonic Acid Metabolic Network toward Inflammation Resolution
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016
Meng, Hu
;
McClendon, Christopher L.
;
Dai, Ziwei
;
Li, Kenan
;
Zhang, Xiaoling
;
He, Shan
;
Shang, Erchang
;
Liu, Ying
;
Lai, Luhua
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2017/12/03
INHIBITION
ENZYMES
MODEL
SITE
BIOSYNTHESIS
PROSTACYCLIN
PROTEINS
EFFECTOR
SYNTHASE
LIGANDS
Ainsliadimer A selectively inhibits IKK alpha/beta by covalently binding a conserved cysteine
期刊论文
NATURE COMMUNICATIONS, 2015
Dong, Ting
;
Li, Chao
;
Wang, Xing
;
Dian, Longyang
;
Zhang, Xiuguo
;
Li, Lin
;
Chen, She
;
Cao, Ran
;
Li, Li
;
Huang, Niu
;
He, Sudan
;
Lei, Xiaoguang
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2017/12/03
NF-KAPPA-B
BIOMIMETIC SYNTHESES
ALLOSTERIC SITE
CANCER-THERAPY
BCL-X
ACTIVATION
PHOSPHORYLATION
INFLAMMATION
KINASE
UBIQUITINATION
Diverse Ways of Perturbing the Human Arachidonic Acid Metabolic Network To Control Inflammation
期刊论文
ACCOUNTS OF CHEMICAL RESEARCH, 2015
Meng, Hu
;
Liu, Ying
;
Lai, Luhua
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2017/12/03
PROSTAGLANDIN E-2 SYNTHASE-1
TRADITIONAL CHINESE MEDICINE
LEUKOTRIENE A(4) HYDROLASE
DUAL INHIBITORS
DRUG DESIGN
LTA(4) HYDROLASE
5-LIPOXYGENASE
DISCOVERY
DERIVATIVES
CYCLOOXYGENASE-2
Discovery of Novel Allosteric Effectors Based on the Predicted Allosteric Sites for Escherichia coli D-3-Phosphoglycerate Dehydrogenase
期刊论文
plos one, 2014
Wang, Qian
;
Qi, Yifei
;
Yin, Ning
;
Lai, Luhua
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2015/11/13
SERINE BIOSYNTHESIS
3-PHOSPHOGLYCERATE DEHYDROGENASE
PHOSPHOGLYCERATE DEHYDROGENASE
MYCOBACTERIUM-TUBERCULOSIS
HYBRID TETRAMERS
BINDING
MODEL
METABOLISM
MECHANISM
PATHWAYS
Discovery of Novel Allosteric Inhibitors for D-3-Phosphoglycerate Dehydrogenase
其他
2014-01-01
刘培
;
王倩
;
刘莹
;
来鲁华
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2015/10/24
PHGDH Metabolic enzymes Virtual screening Allosteric inhibitors Synthesis
Break CDK2/Cyclin E1 Interface Allosterically with Small Peptides
期刊论文
plos one, 2014
Chen, Hao
;
Zhao, Yunjie
;
Li, Haotian
;
Zhang, Dongyan
;
Huang, Yanzhao
;
Shen, Qi
;
Van Duyne, Rachel
;
Kashanchi, Fatah
;
Zeng, Chen
;
Liu, Shiyong
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2015/11/11
PROTEIN-PROTEIN INTERACTIONS
CYCLIN-DEPENDENT KINASE-2
MOLECULAR-DYNAMICS
COMPUTATIONAL DESIGN
STRUCTURAL BASIS
BINDING
ACTIVATION
INHIBITORS
MDM2
P53
Identifying Allosteric Binding Sites in Proteins with a Two-State G(o)over-bar Model for Novel Allosteric Effector Discovery
期刊论文
journal of chemical theory and computation, 2012
Qi, Yifei
;
Wang, Qian
;
Tang, Bo
;
Lai, Luhua
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2015/11/12
LOCAL MOTIONS
D-3-PHOSPHOGLYCERATE DEHYDROGENASE
MOLECULAR-DYNAMICS
SUBSTRATE-BINDING
POPULATION-SHIFT
ENERGY LANDSCAPE
DRUG DISCOVERY
NETWORK MODEL
INHIBITION
KINASE
Gossypol induces Bax/Bak-independent activation of apoptosis and cytochrome c release via a conformational change in Bcl-2
期刊论文
faseb journal, 2006
Lei, Xiaobo
;
Chen, Yingyu
;
Du, Guanhua
;
Yu, Wenyu
;
Wang, Xiaohui
;
Qu, Hong
;
Xia, Bin
;
He, Hongping
;
Mao, Jianhua
;
Zong, Weixing
;
Liao, Xudong
;
Mehrpour, Maryam
;
Hao, Xiaojiang
;
Chen, Quan
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2015/11/16
mitochondria
Bcl-2 inhibitors
drug screening
PERMEABILITY TRANSITION PORE
CELL-DEATH
MITOCHONDRIAL DYSFUNCTION
X-L
CASPASE ACTIVATION
ARSENIC TRIOXIDE
FAMILY PROTEINS
CANCER-CELLS
BAX
AUTOPHAGY
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