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| New 1-(1-ethyl-piperidin-4-yl)-1-(phenyl or heterocyclyl)-alkanol derivatives, are 5-HT(2A) receptor antagonists useful e.g. for treating schizophrenia, depression, memory disorders or eating disorders 专利 作者: PRUECHER HELMUT; BOETTCHER HENNING; ACKERMANN KARL-AUGUST; GOTTSCHLICH RUDOLF; GREINER HARTMUT 收藏  |  浏览/下载:1/0  |  提交时间:2019/12/05 |
| 2-PHENYL-INDOLES AS PROSTAGLANDIN D2 RECEPTOR ANTAGONISTS 专利 作者: YANG ZHAOXIA; REILING STEPHAN; NIEDUZAK THADDEUS R; MATHEW ROSE M; JACKSON SHARON 收藏  |  浏览/下载:3/0  |  提交时间:2019/12/05 |
| Indole derivatives as CRTH2 receptor antagonists in combination with a second active ingredient 专利 作者: Berthelette Carl; Boyd Michael; Colucci John; Villeneuve Karine; Methot Joey 收藏  |  浏览/下载:2/0  |  提交时间:2019/12/05 |
| USE OF B LYMPHOCYTE STIMULATOR PROTEIN ANTAGONISTS TO TREAT ASTHMA AND OTHER ALLERGIC AND INFLAMMATORY CONDITIONS OF THE RESPIRATORY SYSTEM 专利 作者: WASSERMAN Heather; CARLSON Timothy; MIGONE Thi sau; DEVALARAJA Madhav 收藏  |  浏览/下载:8/0  |  提交时间:2019/12/05 |
| AMIDINE-CONTAINING COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS 专利 作者: YuHua Ji; Craig HUSFELD; YongQi MU; Cameron Smith 收藏  |  浏览/下载:3/0  |  提交时间:2019/12/05 |
| As a receptor antagonists mGlu5 polypyridine-4-and-imidazolecarboxylic ethynylbenzoic pyrazolecarboxylic 专利 作者: ビュッテルマン,ベルント; チェッカレッリ,シモーナ・マリーア; ヤーシュケ,ゲオルク; コルツェヴスキ,サビーネ; ポーター,リチャード・ヒュー・フィリップ 收藏  |  浏览/下载:2/0  |  提交时间:2019/12/05 |
| CONDENSED PYRIDINE DERIVATIVES USEFUL AS A28 ADENOSINE RECEPTOR ANTAGONISTS 专利 作者: VIDAL JUAN Bernat; EASTWOOD Paul Robert; GONZALEZ RODRIGUEZ Jacob 收藏  |  浏览/下载:1/0  |  提交时间:2019/12/05 |
| New heteroaryl-substituted piperidine compounds are protease-activated receptor antagonists useful for the treatment and/or prophylaxis of e.g. cardiovascular diseases, thromboembolic diseases, tumors, stroke, hypertension and asthma 专利 作者: Heimbach, Dirk, Dr., 40629 Düsseldorf, DE; Röhrig, Susanne, Dr., 40724 Hilden, DE; Schneider, Dirk, 42115 Wuppertal, DE; Rester, Ulrich, Dr., 42115 Wuppertal, DE; Bender, Eckhard, Dr., 40764 Langenfeld, DE 收藏  |  浏览/下载:4/0  |  提交时间:2019/12/05 |
| IMMUNOMODULATING TUMOR NECROSIS FACTOR RECEPTOR 25 (TNFR25) AGONISTS, ANTAGONISTS AND IMMUNOTOXINS 专利 作者: PODACK, ECKHARD; DEYEV, VADIM; LEVY, ROBERT 收藏  |  浏览/下载:0/0  |  提交时间:2019/12/05 |
| 4-AZETIDINYL-1-HETEROARYL-CYCLOHEXANE ANTAGONISTS OF CCR2 专利 作者: ZHANG Xuqing; HUFNAGEL Heather; CAI Chaozhong; LANTER James; MARKOTAN Thomas 收藏  |  浏览/下载:2/0  |  提交时间:2019/12/05 |