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USP9X stabilizes BRCA1 and confers resistance to DNA-damaging agents in human cancer cells 期刊论文
CANCER MEDICINE, 2019, 卷号: 8, 期号: 15, 页码: 6730-6740
作者:  Lu, Qin;  Zhang, Fang-Lin;  Lu, Da-Yun;  Shao, Zhi-Ming;  Li, Da-Qiang
收藏  |  浏览/下载:23/0  |  提交时间:2020/07/01
Molecular Mechanism of Binding Selectivity of Inhibitors toward BACE1 and BACE2 Revealed by Multiple Short Molecular Dynamics Simulations and Free-Energy Predictions 期刊论文
ACS CHEMICAL NEUROSCIENCE, 2019, 卷号: 10, 期号: 10, 页码: 4303-4318
作者:  Chen, Jianzhong;  Wang, Jinan;  Yin, Baohua;  Pang, Laixue;  Wang, Wei
收藏  |  浏览/下载:116/0  |  提交时间:2020/07/01
Quantitative visualization and detection of acetylcholinesterase activity and its inhibitor based on the oxidation character of ultrathin MnO2 nanosheets. Analytical Methods, Analytical Methods, 2019, 期刊论文
Analytical Methods, 2019, 卷号: 11, 期号: -, 页码: 4931–4938
作者:  Cai-Hong Li;  Jun-Li Yang;  Wei-Feng Wang;  Won Keun Oh;  Dang Lan Huong
收藏  |  浏览/下载:57/0  |  提交时间:2019/11/11
Synthesis and PTP1B/TCPTP Inhibitory Activity Evaluation of Novel 2,5-Disubstituted-1,3,4-thiadiazolamide Derivatives Containing Carbazole/Benzimidazole Moity 期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2019, 卷号: 39, 期号: 9, 页码: 2599-2608
作者:  Li Yingjun;  Zhao Yue;  Jin Kun;  Gao Lixin;  Sheng Li
收藏  |  浏览/下载:35/0  |  提交时间:2020/07/01
Pharmacological characterization of TQ05310, a potent inhibitor of isocitrate dehydrogenase 2 R140Q and R172K mutants 期刊论文
CANCER SCIENCE, 2019, 页码: 9
作者:  Gao, Mingzhao;  Zhu, Hongmei;  Fu, Li;  Li, Yun;  Bao, Xubin
收藏  |  浏览/下载:17/0  |  提交时间:2020/07/01
AG-221  IDH2  leukemia  R140Q  R172K  
Inhibition of the BET family reduces its new target gene IDO1 expression and the production of L-kynurenine 期刊论文
CELL DEATH & DISEASE, 2019, 卷号: 10, 页码: 13
作者:  Tian, Chang-Qing;  Chen, Lin;  Chen, Hua-Dong;  Huan, Xia-Juan;  Hu, Jian-Ping
收藏  |  浏览/下载:21/0  |  提交时间:2020/07/01
Discovery of New Selective Butyrylcholinesterase (BChE) Inhibitors with Anti-A beta Aggregation Activity: Structure-Based Virtual Screening, Hit Optimization and Biological Evaluation 期刊论文
MOLECULES, 2019, 卷号: 24, 期号: 14, 页码: 21
作者:  Jiang, Cheng-Shi;  Ge, Yong-Xi;  Cheng, Zhi-Qiang;  Wang, Yin-Yin;  Tao, Hong-Rui
收藏  |  浏览/下载:14/0  |  提交时间:2020/07/01
禽白血病及鸡白痢检测用标准物质的纯化及稳定 学位论文
: 中国科学院大学, 2019
作者:  尤星力
收藏  |  浏览/下载:19/0  |  提交时间:2020/06/17
The inhibitory mechanism of aurintricarboxylic acid targeting serine/threonine phosphatase Stp1 in Staphylococcus aureus: insights from molecular dynamics simulations 期刊论文
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 6, 页码: 850-858
作者:  Liu, Ting-ting;  Yang, Teng;  Gao, Mei-na;  Chen, Kai-xian;  Yang, Song
收藏  |  浏览/下载:11/0  |  提交时间:2020/07/01
An AIE-based self-assembled fluorescent probe for COX-2 imaging 期刊论文
NEW JOURNAL OF CHEMISTRY, 2019, 卷号: 43, 期号: 20, 页码: 7874-7880
作者:  Cao, Xiaozheng;  Gao, Tang;  Dong, Jie;  Jiang, Xinchen;  Zou, Hui
收藏  |  浏览/下载:5/0  |  提交时间:2020/07/01


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