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科研机构
上海药物研究所 [5]
兰州理工大学 [2]
昆明植物研究所 [1]
上海大学 [1]
上海健康医学院 [1]
兰州化学物理研究所 [1]
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期刊论文 [11]
发表日期
2019 [11]
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Design, synthesis and biological evaluation of novel copper-chelating acetylcholinesterase inhibitors with pyridine and N-benzylpiperidine fragments
期刊论文
BIOORGANIC CHEMISTRY, 2019, 卷号: 93, 页码: 13
作者:
Zhou, Yeheng
;
Sun, Wei
;
Peng, Jiale
;
Yan, Hui
;
Zhang, Li
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2020/03/18
Acetylcholinesterase
Drug design
N-acylhydrazone
Dementia
Copper-chelating
N-Benzylpiperidine
Donepezil, a drug for Alzheimer's disease, promotes oligodendrocyte generation and remyelination
期刊论文
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 11, 页码: 1386-1393
作者:
Cui, Xue
;
Guo, Yu-e
;
Fang, Jia-hui
;
Shi, Chang-jie
;
Suo, Na
收藏
  |  
浏览/下载:69/0
  |  
提交时间:2020/07/01
donepezil
aricept
oligodendrocyte
oligodendrocyte progenitor cell
differentiation
myelin sheaths
remyelination
CNS demyelinating disorders
multiple sclerosis
Quantitative visualization and detection of acetylcholinesterase activity and its inhibitor based on the oxidation character of ultrathin MnO2 nanosheets. Analytical Methods, Analytical Methods, 2019,
期刊论文
Analytical Methods, 2019, 卷号: 11, 期号: -, 页码: 4931–4938
作者:
Cai-Hong Li
;
Jun-Li Yang
;
Wei-Feng Wang
;
Won Keun Oh
;
Dang Lan Huong
收藏
  |  
浏览/下载:55/0
  |  
提交时间:2019/11/11
Acetylcholinesterase
AChE–MnO2–OPD
Discovery of New Selective Butyrylcholinesterase (BChE) Inhibitors with Anti-A beta Aggregation Activity: Structure-Based Virtual Screening, Hit Optimization and Biological Evaluation
期刊论文
MOLECULES, 2019, 卷号: 24, 期号: 14, 页码: 21
作者:
Jiang, Cheng-Shi
;
Ge, Yong-Xi
;
Cheng, Zhi-Qiang
;
Wang, Yin-Yin
;
Tao, Hong-Rui
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2020/07/01
selective BChE inhibitor
virtual screening
structural optimization
molecular dynamics
anti-A beta aggregation
Discovery of new multifunctional selective acetylcholinesterase inhibitors: structure-based virtual screening and biological evaluation
期刊论文
JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN, 2019, 卷号: 33, 期号: 5, 页码: 521-530
作者:
Jiang, Cheng-Shi
;
Ge, Yong-Xi
;
Cheng, Zhi-Qiang
;
Song, Jia-Li
;
Wang, Yin-Yin
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2020/07/01
AChE inhibitor
Pharmacophore model
Molecular docking
Anti-A aggregation
Neuroprotective activity
Colletotrichine B, a new sesquiterpenoid from Colletotrichum gloeosporioides GT-7, a fungal endophyte of Uncaria rhynchophylla
期刊论文
NATURAL PRODUCT RESEARCH, 2019, 卷号: 33, 期号: 1, 页码: 108-112
作者:
Chen, Xiao-Wei
;
Yang, Zhong-Duo
;
Li, Xiao-Fei
;
Sun, Jian-Hui
;
Yang, Li-Jun
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2019/11/15
Colletotrichum gloeosporioides
sesquiterpenoid
Uncaria rhynchophylla
acetylcholinesterase inhibitor
PI3K alpha inhibitor
Colletotrichine B, a new sesquiterpenoid from Colletotrichum gloeosporioides GT-7, a fungal endophyte of Uncaria rhynchophylla
期刊论文
NATURAL PRODUCT RESEARCH, 2019, 卷号: 33, 期号: 1, 页码: 108-112
作者:
Chen, Xiao-Wei
;
Yang, Zhong-Duo
;
Li, Xiao-Fei
;
Sun, Jian-Hui
;
Yang, Li-Jun
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2022/03/01
Colletotrichum gloeosporioides
sesquiterpenoid
Uncaria rhynchophylla
acetylcholinesterase inhibitor
PI3K alpha inhibitor
Synthesis, preliminarily biological evaluation and molecular docking study of new Olaparib analogues as multifunctional PARP-1 and cholinesterase inhibitors
期刊论文
Journal of enzyme inhibition and medicinal chemistry, 2019, 卷号: 34, 页码: 150-162
作者:
Gao Cheng-Zhi[1]
;
Dong Wei[2]
;
Cui Zhi-Wen[3]
;
Yuan Qiong[4]
;
Hu Xia-Min[5]
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2019/04/22
AChE
Alzheimer's Disease
BChE
Olaparib
PARP-1 inhibitor
Synthesis, preliminarily biological evaluation and molecular docking study of new Olaparib analogues as multifunctional PARP-1 and cholinesterase inhibitors
期刊论文
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2019, 卷号: 34, 期号: 1
作者:
Gao, Cheng-Zhi
;
Dong, Wei
;
Cui, Zhi-Wen
;
Yuan, Qiong
;
Hu, Xia-Min
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/06
PARP-1 inhibitor
Olaparib
AChE
BChE
Alzheimer's Disease
donepeziladrugforalzheimersdiseasepromotesoligodendrocytegenerationandremyelination
期刊论文
actapharmacologicasinica, 2019, 卷号: 40, 期号: 11, 页码: 1386
作者:
Cui Xue
;
Guo Yue
;
Fang Jiahui
;
Shi Changjie
;
Suo Na
收藏
  |  
浏览/下载:57/0
  |  
提交时间:2020/07/01
EXPERIMENTAL AUTOIMMUNE ENCEPHALOMYELITIS
NICOTINIC ACETYLCHOLINE-RECEPTORS
CENTRAL-NERVOUS-SYSTEM
THYROID-HORMONE
MYELINATION
INHIBITORS
NEUROPROTECTION
CELL
ACTIVATION
GROWTH
donepezil
aricept
oligodendrocyte
oligodendrocyte progenitor cell
differentiation
myelin sheaths
remyelination
CNS demyelinating disorders
multiple sclerosis
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