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Discovery of (E)-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)propanamide (CHMFL-ABL-121) as a highly potent ABL kinase inhibitor capable of overcoming a variety of ABL mutants including T315I for chronic myeloid leukemia 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 160, 页码: 61-81
作者:  Liu, Xuesong;  Wang, Beilei;  Chen, Cheng;  Jiang, Zongru;  Hu, Chen
收藏  |  浏览/下载:14/0  |  提交时间:2019/01/11
PIDA/I-2-Mediated alpha- and beta-C(sp(3))-H Bond Dual Functionalization of Tertiary Amines 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2018, 卷号: 83, 期号: 17, 页码: 10166-10174
作者:  Zhu, Yu;  Shao, Li-Dong;  Deng, Zhen-Tao;  Bao, Ying;  Shi, Xin
收藏  |  浏览/下载:20/0  |  提交时间:2018/10/22
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFR alpha kinase inhibitor for PDGFR alpha driving chronic eosinophilic leukemia 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 期号: 无, 页码: 366-384
作者:  Wang, Qiang;  Liu, Feiyang;  Qi, Shuang;  Qi, Ziping;  Yan, Xiao-E.
收藏  |  浏览/下载:62/0  |  提交时间:2019/06/10
Comparison of Frequency and Sensitivity of BCR-ABL1 Kinase Domain Mutations in Asian and White Patients With Imatinib-resistant Chronice-Phase Chronic Myeloid Leukemia 期刊论文
CLINICAL LYMPHOMA MYELOMA & LEUKEMIA, 2018, 卷号: 18, 期号: 10
作者:  Cui, Jiu Wei;  Kim, Hawk;  Kim, SooHyun;  Kim, Hyeoung-Joon;  Kim, Yeo-Kyeoung
收藏  |  浏览/下载:13/0  |  提交时间:2019/12/05
THE ECONOMIC EVALUATION OF IMATINIB COMBINED WITH CHEMOTHERAPY FOR PEDIATRIC PHILADELPHIA CHROMOSOME-POSITIVE ACUTE LYMPHOBLASTIC LEUKEMIA IN CHINA 会议论文
作者:  Wang, V. W.;  Li, Z.
收藏  |  浏览/下载:8/0  |  提交时间:2019/12/05
To compare the efficacy of sunitinib and imatinib following cytoreductive resection in GIST patients with progression on imatinib: A multi-center controlled study. 会议论文
作者:  Zhang, Xinhua;  Zhou, Ye;  Wu, Xin;  Nie, Mingming;  Zhang, Bo
收藏  |  浏览/下载:7/0  |  提交时间:2019/12/05
Early BCR-ABL1 decline in imatinib-treated patients with chronic myeloid leukemia: results from a multicenter study of the Chinese CML alliance 期刊论文
Blood Cancer Journal, 2018, 卷号: Vol.8
作者:  Zhang, JR;  Wang, YQ;  Wang, JX;  Hu, JD;  Chen, SN
收藏  |  浏览/下载:49/0  |  提交时间:2019/02/25
Cytoreductive surgery for metastatic gastrointestinal stromal tumors followed by sunitinib compared to followed by imatinib-a multi-center cohort study 期刊论文
European Journal of Surgical Oncology, 2018
作者:  Xinhua Zhang;  Ye Zhou;  Xin Wu;  Mingming Nie;  Bo Zhang
收藏  |  浏览/下载:6/0  |  提交时间:2019/02/28
Co-delivery of doxorubicin and imatinib by pH sensitive cleavable PEGylated nanoliposomes with folate-mediated targeting to overcome multidrug resistance 期刊论文
INTERNATIONAL JOURNAL OF PHARMACEUTICS, 2018, 卷号: 542, 期号: 1-2
作者:  Chen, Yan;  Cheng, Yao;  Zhao, Pengxuan;  Zhang, Shasha;  Li, Minsi
收藏  |  浏览/下载:8/0  |  提交时间:2019/12/05
The c-Myc-regulated lncRNA NEAT1 and paraspeckles modulate imatinib-induced apoptosis in CML cells 期刊论文
2018, 卷号: 17
作者:  Zeng, Chengwu[1,2];  Liu, Sichu[1];  Lu, Shuai[1];  Yu, Xibao[1];  Lai, Jing[2]
收藏  |  浏览/下载:9/0  |  提交时间:2019/12/13


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