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Positive Allosteric Modulation of AMPAR by PF-4778574 Produced Rapid Onset Antidepressant Actions in Mice 期刊论文
Cerebral cortex (New York, N.Y. : 1991), 2018
作者:  Shen, Mengxin;  Lv, Dan;  Li, Shuting;  Zhang, Yanhua;  Wang, Zhen
收藏  |  浏览/下载:104/0  |  提交时间:2019/01/08
Exploring molecular mechanism of allosteric inhibitor to relieve drug resistance of multiple mutations in HIV-1 protease by enhanced conformational sampling 期刊论文
PROTEINS-STRUCTURE FUNCTION AND BIOINFORMATICS, 2018, 卷号: 86, 期号: 12, 页码: 1294-1305
作者:  Chen, Jianzhong;  Peng, Cheng;  Wang, Jinan;  Zhu, Weiliang
收藏  |  浏览/下载:59/0  |  提交时间:2019/01/08
Druggable negative allosteric site of P2X3 receptors 期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2018, 卷号: 115, 期号: 19, 页码: 4939-4944
作者:  Wang, Jin;  Wang, Yao;  Cui, Wen-Wen;  Huang, Yichen;  Yang, Yang
收藏  |  浏览/下载:27/0  |  提交时间:2019/01/08
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFR alpha kinase inhibitor for PDGFR alpha driving chronic eosinophilic leukemia 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 期号: 无, 页码: 366-384
作者:  Wang, Qiang;  Liu, Feiyang;  Qi, Shuang;  Qi, Ziping;  Yan, Xiao-E.
收藏  |  浏览/下载:62/0  |  提交时间:2019/06/10
High-throughput identification of G protein-coupled receptor modulators through affinity mass spectrometry screening 期刊论文
CHEMICAL SCIENCE, 2018, 卷号: 9, 期号: 12, 页码: 3192-3199
作者:  Qin, Shanshan;  Meng, Mengmeng;  Yang, Dehua;  Bai, Wenwen;  Lu, Yan
收藏  |  浏览/下载:42/0  |  提交时间:2019/01/08
Structure Optimization and Structure-Activity Relationship Study of a Kind of Type II FAK Inhibitors with N-Phenylpyrazole Ureas 期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2018, 卷号: 38, 期号: 11
作者:  Gong Chaochao;  Tan Hanyi;  Zhang Qian
收藏  |  浏览/下载:2/0  |  提交时间:2019/12/05
Valepotriates From the Roots and Rhizomes of Valeriana jatamansi Jones as Novel N-Type Calcium Channel Antagonists 期刊论文
FRONTIERS IN PHARMACOLOGY, 2018, 卷号: 9, 页码: 885
作者:  Dong, Fa-Wu;  Jiang, He-Hai;  Yang, Liu;  Gong, Ye;  Zi, Cheng-Ting
收藏  |  浏览/下载:37/0  |  提交时间:2019/03/29
Valepotriates From the Roots and Rhizomes of Valeriana jatamansi Jones as Novel N-Type Calcium Channel Antagonists. 期刊论文
Frontiers in Pharmacology, 2018, 期号: 9, 页码: 885
作者:  Fa-Wu Dong;  Yin Nian;  Liu Yang;  Jun Zhou;  Ye Gong
收藏  |  浏览/下载:28/0  |  提交时间:2018/09/19


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