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Discovery of new potent protein arginine methyltransferase 5 (PRMT5) inhibitors by assembly of key pharmacophores from known inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2018, 卷号: 28, 期号: 23-24, 页码: 3693-3699
作者:  Zhu, Kongkai;  Song, Jia-Li;  Tao, Hong-Rui;  Cheng, Zhi-Qiang;  Jiang, Cheng-Shi
收藏  |  浏览/下载:100/0  |  提交时间:2019/01/08
Identification of a cellularly active SIRT6 allosteric activator 期刊论文
NATURE CHEMICAL BIOLOGY, 2018, 卷号: 14, 期号: 12, 页码: 1118-+
作者:  Huang, Zhimin;  Zhao, Junxing;  Deng, Wei;  Chen, Yingyi;  Shang, Jialin
收藏  |  浏览/下载:88/0  |  提交时间:2019/01/08
18β-Glycyrrhetinic acid protects against alpha-naphthylisothiocyanate-induced cholestasis through activation of the Sirt1/FXR signaling pathway 期刊论文
Acta pharmacologica Sinica, 2018, 卷号: 39, 期号: 12, 页码: 1865-1873
作者:  Wu, Shou-Yan;  Cui, Shi-Chao;  Wang, Le;  Zhang, Yi-Ting;  Yan, Xiao-Xia
收藏  |  浏览/下载:93/0  |  提交时间:2019/01/08
18 beta-Glycyrrhetinic acid protects against alpha-naphthylisothiocyanate-induced cholestasis through activation of the Sirt1/FXR signaling pathway 期刊论文
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 12, 页码: 1865-1873
作者:  Wu, Shou-yan;  Cui, Shi-chao;  Wang, Le;  Zhang, Yi-ying;  Yan, Xiao-xia
收藏  |  浏览/下载:13/0  |  提交时间:2020/07/01
C11, a novel fibroblast growth factor receptor 1 (FGFR1) inhibitor, suppresses breast cancer metastasis and angiogenesis 期刊论文
Acta pharmacologica Sinica, 2018
作者:  Chen, Zhuo;  Tong, Lin-Jiang;  Tang, Bai-You;  Liu, Hong-Yan;  Wang, Xin
收藏  |  浏览/下载:101/0  |  提交时间:2019/01/08
Development of high potent and selective Bcl-2 inhibitors bearing the structural elements of natural product artemisinin 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 159, 页码: 149-165
作者:  Liu, Xiaohua;  Zhang, Yu;  Huang, Wenjing;  Luo, Jia;  Li, Yang
收藏  |  浏览/下载:37/0  |  提交时间:2019/01/08
Discovery of JND3229 as a New EGFR(C797S) Mutant Inhibitor with In Vivo Monodrug Efficacy 期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2018, 卷号: 9, 期号: 11, 页码: 1123-1127
作者:  Lu, Xiaoyun;  Zhang, Tao;  Zhu, Su-Jie;  Xun, Qiuju;  Tong, Lingjiang
收藏  |  浏览/下载:108/0  |  提交时间:2019/01/08
Identification of compound D2923 as a novel anti-tumor agent targeting CSF1R 期刊论文
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 11, 页码: 1768-1776
作者:  Liu, Ying-Qiang;  Wang, Ya-Nan;  Lu, Xiao-Yun;  Tong, Lin-Jiang;  Li, Yan
收藏  |  浏览/下载:110/0  |  提交时间:2019/01/08
Discovery of Potent Irreversible Pan-Fibroblast Growth Factor Receptor (FGFR) Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 20, 页码: 9085-9104
作者:  Wang, Yuming;  Li, Lijun;  Fan, Jun;  Dai, Yang;  Jiang, Alan
收藏  |  浏览/下载:29/0  |  提交时间:2019/01/08
Phosphodiesterase-4 Inhibitors for the Treatment of Inflammatory Diseases 期刊论文
FRONTIERS IN PHARMACOLOGY, 2018, 卷号: 9
作者:  Li, Heng;  Zuo, Jianping;  Tang, Wei
收藏  |  浏览/下载:55/0  |  提交时间:2019/01/08


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