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Rational design of 5-((1H-imidazol-1-yl)methyl)quinolin-8-ol derivatives as novel bromodomain-containing protein 4 inhibitors 期刊论文
European journal of medicinal chemistry, 2018, 卷号: 163, 页码: 281-294
作者:  Xing, Jing;  Zhang, Rukang;  Jiang, Xiangrui;  Hu, Tianwen;  Wang, Xinjun
收藏  |  浏览/下载:88/0  |  提交时间:2019/01/08
Development and evaluation of a novel series of Nitroxoline-derived BET inhibitors with antitumor activity in renal cell carcinoma 期刊论文
ONCOGENESIS, 2018, 卷号: 7
作者:  Chen, Wei;  Zhang, Hao;  Chen, Zhifeng;  Jiang, Hao;  Liao, Liping
收藏  |  浏览/下载:108/0  |  提交时间:2019/01/08
Nut Directs p300-Dependent, Genome-Wide H4 Hyperacetylation in Male Germ Cells 期刊论文
CELL REPORTS, 2018, 卷号: 24, 期号: 13, 页码: 3477-+
作者:  Shiota, Hitoshi;  Barral, Sophie;  Buchou, Thierry;  Tan, Minjia;  Coute, Yohann
收藏  |  浏览/下载:66/0  |  提交时间:2019/01/08
Identification of small molecule inhibitors targeting the SMARCA2 bromodomain from a high-throughput screening assay 期刊论文
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 9, 页码: 1544-1552
作者:  Lu, Tian;  Hu, Jun-chi;  Lu, Wen-chao;  Han, Jie;  Ding, Hong
收藏  |  浏览/下载:33/0  |  提交时间:2019/01/08
Discovery of QCA570 as an Exceptionally Potent and Efficacious Proteolysis Targeting Chimera (PROTAC) Degrader of the Bromodomain and Extra-Terminal (BET) Proteins Capable of Inducing Complete and Durable Tumor Regression 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 15, 页码: 6685-6704
作者:  Qin, Chong;  Hu, Yang;  Zhou, Bing;  Fernandez-Salas, Ester;  Yang, Chao-Yie
收藏  |  浏览/下载:45/0  |  提交时间:2019/01/08
Structure-Based Discovery of CF53 as a Potent and Orally Bioavailable Bromodomain and Extra-Terminal (BET) Bromodomain Inhibitor 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 14, 页码: 6110-6120
作者:  Zhao, Yujun;  Zhou, Bing;  Bai, Longchuan;  Liu, Liu;  Yang, Chao-Yie
收藏  |  浏览/下载:49/0  |  提交时间:2019/01/08
Brd2调节I型干扰素机制研究和病毒感染转录组分析 学位论文
北京: 中国科学院大学, 2018
作者:  胡本霞
收藏  |  浏览/下载:73/0  |  提交时间:2019/09/30
Design, synthesis and biological evaluation of benzo[cd]indo1-2(1H)-ones derivatives as BRD4 inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 152, 页码: 264-273
作者:  Feng, Yuxin;  Xiao, Senhao;  Chen, Yantao;  Jiang, Hao;  Liu, Na
收藏  |  浏览/下载:35/0  |  提交时间:2019/01/08
Structure-based optimization of a series of selective BET inhibitors containing aniline or indoline groups 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 页码: 156-175
作者:  Hu, Jianping;  Wang, Yingqing;  Li, Yanlian;  Cao, Danyan;  Xu, Lin
收藏  |  浏览/下载:34/0  |  提交时间:2019/01/08
Computer-Aided Drug Design in Epigenetics 期刊论文
FRONTIERS IN CHEMISTRY, 2018, 卷号: 6
作者:  Lu, Wenchao;  Zhang, Rukang;  Jiang, Hao;  Zhang, Huimin;  Luo, Cheng
收藏  |  浏览/下载:27/0  |  提交时间:2019/01/08


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