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Design, Synthesis, and Pharmacological Evaluation of 2-(2,5-Dimethyl-5,6,7,8-tetrahydroquinolin-8-yl)-N-aryl Propanamides as Novel Smoothened (Smo) Antagonists 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 24, 页码: 11050-11068
作者:  Liu, Gang;  Xue, Ding;  Yang, Jun;  Wan, Juan;  Liu, Xiaohua
收藏  |  浏览/下载:54/0  |  提交时间:2019/01/08
Miltirone protects human EA.hy926 endothelial cells from oxidized low-density lipoprotein-derived oxidative stress via a heme oxygenase-1 and MAPK/Nrf2 dependent pathway 期刊论文
PHYTOMEDICINE, 2016, 卷号: 23, 期号: 14, 页码: 1806-1813
作者:  Zhang, Liu;  Zhang, Hui;  Li, Xueyan;  Jia, Bingjie;  Yang, Yuyu
收藏  |  浏览/下载:19/0  |  提交时间:2019/01/08
Molecular mechanism of R-bicalutamide switching from androgen receptor antagonist to agonist induced by amino acid mutations using molecular dynamics simulations and free energy calculation 期刊论文
JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN, 2016, 卷号: 30, 期号: 1-12, 页码: 1189-1200
作者:  Liu, HL;  Han, R;  Li, JZ;  Liu, HX;  Zheng, LF
收藏  |  浏览/下载:3/0  |  提交时间:2017/05/09
DESIGN, SYNTHESIS, IN VITRO ANTIPROLIFERATIVE ACTIVITY EVALUATION OF 2-ALICANOYLAMIDOTHIOPHENE-3-CARBOXAMIDE DERIVATIVES 期刊论文
HETEROCYCLES, 2016, 卷号: 92, 期号: 12, 页码: 2145-2165
作者:  Zhang, Jiefeng;  Guan, Fengjie;  Qiu, Jiakun;  Fang, Yanfen;  Yu, Lifang
收藏  |  浏览/下载:28/0  |  提交时间:2019/01/08
Challenges and strategies of oral insulin delivery 会议论文
作者:  Gan Y(甘勇)
收藏  |  浏览/下载:23/0  |  提交时间:2019/01/08
Ultra-deep tyrosine phosphoproteomics enabled by a phosphotyrosine superbinder 期刊论文
NATURE CHEMICAL BIOLOGY, 2016, 卷号: 12, 期号: 11, 页码: 959-+
作者:  Liu, Xuguang;  Bian, Yangyang;  Li, Lei;  Dong, Mingming;  Kaneko, Tomonori
收藏  |  浏览/下载:22/0  |  提交时间:2019/06/20
Design, Synthesis of Lithocholic Acid Mimics and Their Inhibitory Activities against Protein Tyrosine Phosphatase 1B 期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2016, 卷号: 36, 期号: 11, 页码: 2670-2676
作者:  He Haibing;  Dai Hong;  Gao Lixin;  Zhang Haijun;  Zou Zheng
收藏  |  浏览/下载:26/0  |  提交时间:2019/01/08
Design, Synthesis, and Biological Evaluation of Novel Tetrahydroprotoberberine Derivatives (THPBs) as Selective alpha(1A)-Adrenoceptor Antagonists 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 20, 页码: 9489-9502
作者:  Guo, Diliang;  Li, Jing;  Lin, Henry;  Zhou, Yu;  Chen, Ying
收藏  |  浏览/下载:28/0  |  提交时间:2019/01/08
Crystal Structure of the Human Cannabinoid Receptor CB1 期刊论文
CELL, 2016, 卷号: 167, 期号: 3, 页码: 750-+
作者:  Hua, Tian;  Vemuri, Kiran;  Pu, Mengchen;  Qu, Lu;  Han, Gye Won
收藏  |  浏览/下载:20/0  |  提交时间:2019/01/08
Design, Synthesis and Biological Evaluation of 6-(2,6-Dichloro-3,5-dimethoxyphenyl)-4-substituted-1H-indazoles as Potent Fibroblast Growth Factor Receptor Inhibitors 期刊论文
MOLECULES, 2016, 卷号: 21, 期号: 10
作者:  Zhang, Zhen;  Zhao, Dongmei;  Dai, Yang;  Cheng, Maosheng;  Geng, Meiyu
收藏  |  浏览/下载:16/0  |  提交时间:2019/01/08


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