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A structure-guided optimization of pyrido[2,3-d]pyrimidin-7-ones as selective inhibitors of EGFR(L858R/T790M) mutant with improved pharmacokinetic properties
Yu, Lei[1,2]; Huang, Minhao[1,2]; Xu, Tianfeng[1,2]; Tong, Linjiang[4]; Yan, Xiao-e[5,6]; Zhang, Zhang[1]; Xu, Yong[1]; Yun, Caihong; Xie, Hua[4]; Ding, Ke[1,3]
2017
卷号126期号:[db:dc_citation_issue]页码:1107
DOI[db:dc_identifier_doi]
URL标识查看原文
WOS记录号[DB:DC_IDENTIFIER_WOSID]
内容类型期刊论文
URI标识http://www.corc.org.cn/handle/1471x/3353701
专题暨南大学
作者单位1.[1]Chinese Acad Sci, Guangzhou Inst Biomed & Hlth, 190 Kaiyuan Ave, Guangzhou 510530, Peoples R China
2.[2]Univ Chinese Acad Sci, 19 Yuquan Rd, Beijing 100049, Peoples R China
3.[3]Jinan Univ, Sch Pharm, 601 Huangpu Ave West, Guangzhou 510632, Peoples R China
4.[4]Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, 555 Zu Chong Zhi Rd,Zhangjiang Hi Tech Pk, Shanghai 201203, Peoples R China
5.[5]Peking Univ, Hlth Sci Ctr, Inst Syst Biomed, Beijing 100191, Peoples R China
6.[6]Peking Univ, Hlth Sci Ctr, Dept Biophys, Beijing 100191, Peoples R China
推荐引用方式
GB/T 7714
Yu, Lei[1,2],Huang, Minhao[1,2],Xu, Tianfeng[1,2],et al. A structure-guided optimization of pyrido[2,3-d]pyrimidin-7-ones as selective inhibitors of EGFR(L858R/T790M) mutant with improved pharmacokinetic properties[J],2017,126([db:dc_citation_issue]):1107.
APA Yu, Lei[1,2].,Huang, Minhao[1,2].,Xu, Tianfeng[1,2].,Tong, Linjiang[4].,Yan, Xiao-e[5,6].,...&Lu, Xiaoyun[3].(2017).A structure-guided optimization of pyrido[2,3-d]pyrimidin-7-ones as selective inhibitors of EGFR(L858R/T790M) mutant with improved pharmacokinetic properties.,126([db:dc_citation_issue]),1107.
MLA Yu, Lei[1,2],et al."A structure-guided optimization of pyrido[2,3-d]pyrimidin-7-ones as selective inhibitors of EGFR(L858R/T790M) mutant with improved pharmacokinetic properties".126.[db:dc_citation_issue](2017):1107.
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