Design, synthesis and anticancer potential of NSC-319745 hydroxamic acid derivatives as DNMT and HDAC inhibitors | |
Yuan, Zigao[1,2]; Sun, Qinsheng[2,3]; Li, Dan[1,2]; Miao, Shuangshuang[2]; Chen, Shaopeng[2]; Song, Lu[1,2]; Gao, Chunmei[2,4]; Chen, Yuzong[4,5]; Tan, Chunyan[4]; Jiang, Yuyang[2,3,4] | |
刊名 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY |
2017 | |
卷号 | 134页码:281-292 |
关键词 | Epigenetic targets Multi-target Drug design Antitumor bioactivity DNMT HDAC |
URL标识 | 查看原文 |
内容类型 | 期刊论文 |
URI标识 | http://www.corc.org.cn/handle/1471x/2187619 |
专题 | 华南理工大学 |
作者单位 | 1.[1]Tsinghua Univ, Dept Chem, Beijing 100084, Peoples R China 2.[2]Tsinghua Univ, Grad Sch Shenzhen, Minist Prov Jointly Constructed Base State Key La, Shenzhen 518055, Peoples R China 3.[3]Tsinghua Univ, Sch Med, Dept Pharmacol & Pharmaceut Sci, Beijing 100084, Peoples R China 4.[4]Tsinghua Univ, Grad Sch Shenzhen, Natl & Local United Engn Lab Personalized Antitum, Shenzhen 518055, Peoples R China 5.[5]Natl Univ Singapore, Ctr Computat Sci & Engn, Dept Pharm, Bioinformat & Drug Design Grp, Singapore 117543, Singapore |
推荐引用方式 GB/T 7714 | Yuan, Zigao[1,2],Sun, Qinsheng[2,3],Li, Dan[1,2],et al. Design, synthesis and anticancer potential of NSC-319745 hydroxamic acid derivatives as DNMT and HDAC inhibitors[J]. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY,2017,134:281-292. |
APA | Yuan, Zigao[1,2].,Sun, Qinsheng[2,3].,Li, Dan[1,2].,Miao, Shuangshuang[2].,Chen, Shaopeng[2].,...&Jiang, Yuyang[2,3,4].(2017).Design, synthesis and anticancer potential of NSC-319745 hydroxamic acid derivatives as DNMT and HDAC inhibitors.EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY,134,281-292. |
MLA | Yuan, Zigao[1,2],et al."Design, synthesis and anticancer potential of NSC-319745 hydroxamic acid derivatives as DNMT and HDAC inhibitors".EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 134(2017):281-292. |
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