Synthesis and Fungicidal Activity of Novel 2,5-Disubstituted-1,3,4-oxadiazole Derivatives

doi:10.1021/jf303807a

	Synthesis and Fungicidal Activity of Novel 2,5-Disubstituted-1,3,4-oxadiazole Derivatives
	Cui, Zi-Ning 1,3; Shi, Yan-Xia 2; Zhang, Li 1; Ling, Yun 1; Li, Bao-Ju 2; Nishida, Yoshihiro 3; Yang, Xin-Ling 1
刊名	JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY
	2012
卷号	60 期号:47 页码:11649-11656
关键词	2,5-disubstituted-1,3,4-oxadiazole 5-phenyl-2-furan fungicidal activity microwave irradiation synthesis
ISSN号	0021-8561
DOI	10.1021/jf303807a
通讯作者	Cui, Zi-Ning
英文摘要	A novel series of 1,3,4-oxadiazole derivatives containing a 5-phenyl-2-furan moiety were synthesized from the intermediates diacylhydrazine 3 and acylhydrazone 5 via an efficient approach under microwave irradiation in good yields. Their structures were characterized by IR, H-1 NMR, and elemental analysis. The antifungal tests indicated that the title compounds showed in vivo fungicidal activity against Botrytis cinerea and Rhizoctonia solanii at 500 mu g/mL obviously. Some tested compounds even had a superiority effect over the commercial fungicides 40% Pyrimethanil SC and 3% Validamycin AS. The activity between the title compound and their precursors diacylhydrazine 3 and acylhydrazone 5 was also compared and discussed.
学科主题	Agriculture, Multidisciplinary ; Chemistry, Applied ; Food Science & Technology ; AGRICULTURE, MULTIDISCIPLINARY ; CHEMISTRY, APPLIED ; FOOD SCIENCE & TECHNOLOGY
语种	英语
出版者	AMER CHEMICAL SOC
WOS记录号	WOS:000313769500001
内容类型	期刊论文
源URL	[http://111.203.20.206/handle/2HMLN22E/101084]
专题	蔬菜花卉研究所_植物保护研究室
作者单位	1.China Agr Univ, Dept Appl Chem, Coll Sci, Beijing 100193, Peoples R China 2.Chinese Acad Agr Sci, Inst Vegetables & Flowers, Beijing 100081, Peoples R China 3.Chiba Univ, Dept Nanobiol, Grad Sch Adv Integrat Sci, Matsudo, Chiba 2718510, Japan
推荐引用方式 GB/T 7714	Cui, Zi-Ning,Shi, Yan-Xia,Zhang, Li,et al. Synthesis and Fungicidal Activity of Novel 2,5-Disubstituted-1,3,4-oxadiazole Derivatives[J]. JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY,2012,60(47):11649-11656.
APA	Cui, Zi-Ning.,Shi, Yan-Xia.,Zhang, Li.,Ling, Yun.,Li, Bao-Ju.,...&Yang, Xin-Ling.(2012).Synthesis and Fungicidal Activity of Novel 2,5-Disubstituted-1,3,4-oxadiazole Derivatives.JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY,60(47),11649-11656.
MLA	Cui, Zi-Ning,et al."Synthesis and Fungicidal Activity of Novel 2,5-Disubstituted-1,3,4-oxadiazole Derivatives".JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY 60.47(2012):11649-11656.